TW201313726A - 製造合成之中間體之方法 - Google Patents

製造合成之中間體之方法 Download PDF

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Publication number
TW201313726A
TW201313726A TW101133871A TW101133871A TW201313726A TW 201313726 A TW201313726 A TW 201313726A TW 101133871 A TW101133871 A TW 101133871A TW 101133871 A TW101133871 A TW 101133871A TW 201313726 A TW201313726 A TW 201313726A
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TW
Taiwan
Prior art keywords
compound
formula
polar aprotic
mixture
aprotic solvent
Prior art date
Application number
TW101133871A
Other languages
English (en)
Chinese (zh)
Inventor
Stefan Abele
Eike J Bergner
Christian Bukovec
Jacques-Alexis Funel
Christian Hubschwerlen
Azely Mirre
Ivan Schindelholz
Jean-Philippe Surivet
Acklin Cornelia Zumbrunn
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of TW201313726A publication Critical patent/TW201313726A/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D497/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D497/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D497/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
TW101133871A 2011-09-16 2012-09-14 製造合成之中間體之方法 TW201313726A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IB2011054061 2011-09-16

Publications (1)

Publication Number Publication Date
TW201313726A true TW201313726A (zh) 2013-04-01

Family

ID=47080755

Family Applications (1)

Application Number Title Priority Date Filing Date
TW101133871A TW201313726A (zh) 2011-09-16 2012-09-14 製造合成之中間體之方法

Country Status (3)

Country Link
AR (1) AR087875A1 (es)
TW (1) TW201313726A (es)
WO (1) WO2013038374A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3936192A4 (en) 2019-03-06 2022-11-16 Daiichi Sankyo Company, Limited PYRROLOPYRAZOL DERIVATIVES

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009512695A (ja) 2005-10-21 2009-03-26 グラクソ グループ リミテッド 化合物
EP1963324B1 (en) 2005-12-22 2010-04-21 Glaxo Group Limited Heterocyclic compounds, their preparation and their use as antibacterials
GB0613208D0 (en) 2006-07-03 2006-08-09 Glaxo Group Ltd Compounds
EP1992628A1 (en) 2007-05-18 2008-11-19 Glaxo Group Limited Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
GB0705672D0 (en) 2007-03-23 2007-05-02 Glaxo Group Ltd Compounds
EP1980251A1 (en) 2007-04-13 2008-10-15 Glaxo Group Limited Pyrrolo[3,2,1-ij]quinoline-4-one derivatives for treating tuberculosis
ES1065649Y (es) 2007-06-22 2008-01-01 Gavalda Josep Sarmiento Disposicion perfeccionada de apertura de bozal para animales
WO2009128953A2 (en) 2008-04-18 2009-10-22 University Of Maryland, Baltimore Genetic variants in a hypertension susceptibility gene stk39 and uses thereof
EP2376497B1 (en) 2008-12-12 2013-09-18 Actelion Pharmaceuticals Ltd. 5-amino-2-(1-hydroxy-ethyl)-tetrahydropyran derivatives
AR076222A1 (es) 2009-04-09 2011-05-26 Actelion Pharmaceuticals Ltd Derivados 2-hidroxietil-1h-quinolin-ona y sus analogos azaisotericos con actividad antibacteriana y composiciones farmaceuticas que los contienen

Also Published As

Publication number Publication date
AR087875A1 (es) 2014-04-23
WO2013038374A1 (en) 2013-03-21

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