TW200924770A - Novel compounds 089 - Google Patents
Novel compounds 089 Download PDFInfo
- Publication number
- TW200924770A TW200924770A TW097142665A TW97142665A TW200924770A TW 200924770 A TW200924770 A TW 200924770A TW 097142665 A TW097142665 A TW 097142665A TW 97142665 A TW97142665 A TW 97142665A TW 200924770 A TW200924770 A TW 200924770A
- Authority
- TW
- Taiwan
- Prior art keywords
- phenyl
- methyl
- compound
- pharmaceutically acceptable
- trifluoromethyl
- Prior art date
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Classifications
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
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- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
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|---|---|---|---|
| US98571307P | 2007-11-06 | 2007-11-06 |
Publications (1)
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| TW200924770A true TW200924770A (en) | 2009-06-16 |
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| EP (1) | EP2217591A4 (enExample) |
| JP (1) | JP2011502982A (enExample) |
| KR (1) | KR20100096131A (enExample) |
| CN (1) | CN101918391B (enExample) |
| AR (1) | AR069206A1 (enExample) |
| AU (1) | AU2008325288B2 (enExample) |
| BR (1) | BRPI0819258A2 (enExample) |
| CA (1) | CA2703996A1 (enExample) |
| CL (1) | CL2008003301A1 (enExample) |
| CO (1) | CO6270241A2 (enExample) |
| CR (1) | CR11416A (enExample) |
| DO (1) | DOP2010000134A (enExample) |
| EA (1) | EA017297B1 (enExample) |
| IL (1) | IL205209A0 (enExample) |
| MX (1) | MX2010004673A (enExample) |
| NI (1) | NI201000079A (enExample) |
| PE (1) | PE20091565A1 (enExample) |
| SV (1) | SV2010003559A (enExample) |
| TW (1) | TW200924770A (enExample) |
| UY (1) | UY31456A1 (enExample) |
| WO (1) | WO2009061271A1 (enExample) |
| ZA (1) | ZA201002853B (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| SE0302486D0 (sv) * | 2003-09-18 | 2003-09-18 | Astrazeneca Ab | Novel compounds |
| TW200808771A (en) | 2006-05-08 | 2008-02-16 | Astrazeneca Ab | Novel compounds II |
| TW200808763A (en) | 2006-05-08 | 2008-02-16 | Astrazeneca Ab | Novel compounds I |
| EP2217591A4 (en) | 2007-11-06 | 2011-10-26 | Astrazeneca Ab | CERTAIN 2-PYRAZINONE DERIVATIVES AND THEIR USE AS NEUTROPHILES ELASTASE INHIBITORS |
| TW201036957A (en) | 2009-02-20 | 2010-10-16 | Astrazeneca Ab | Novel salt 628 |
| CA2773618A1 (en) | 2009-10-02 | 2011-04-07 | Astrazeneca Ab | 2-pyridone compounds used as inhibitors of neutrophil elastase |
| WO2011110852A1 (en) | 2010-03-10 | 2011-09-15 | Astrazeneca Ab | Polymorphic forms of 6- [2- (4 -cyanophenyl) - 2h - pyrazol - 3 - yl] - 5 -methyl - 3 - oxo - 4 - (trifluoromethyl - phenyl) 3,4-dihydropyrazine-2-carboxylic acid ethylamide |
| DE102010030187A1 (de) | 2010-06-16 | 2011-12-22 | Bayer Schering Pharma Aktiengesellschaft | 4-Cyan-2-sulfonylphenyl)pyrazolyl-substituierte Pyridinone und Pyrazinone und ihre Verwendung |
| TW201247631A (en) | 2011-04-28 | 2012-12-01 | Du Pont | Herbicidal pyrazinones |
| CA2878792A1 (en) * | 2012-07-12 | 2014-01-16 | Chiesi Farmaceutici S.P.A. | Inhibition of enzymes |
| US9102624B2 (en) | 2012-08-23 | 2015-08-11 | Boehringer Ingelheim International Gmbh | Substituted 4-pyridones and their use as inhibitors of neutrophil elastase activity |
| US20140057920A1 (en) | 2012-08-23 | 2014-02-27 | Boehringer Ingelheim International Gmbh | Substituted 4-pyridones and their use as inhibitors of neutrophil elastase activity |
| US20140057926A1 (en) | 2012-08-23 | 2014-02-27 | Boehringer Ingelheim International Gmbh | Substituted 4-pyridones and their use as inhibitors of neutrophil elastase activity |
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2008
- 2008-11-05 EP EP08847756A patent/EP2217591A4/en not_active Withdrawn
- 2008-11-05 BR BRPI0819258A patent/BRPI0819258A2/pt not_active IP Right Cessation
- 2008-11-05 AR ARP080104851A patent/AR069206A1/es unknown
- 2008-11-05 WO PCT/SE2008/051263 patent/WO2009061271A1/en not_active Ceased
- 2008-11-05 AU AU2008325288A patent/AU2008325288B2/en not_active Ceased
- 2008-11-05 US US12/740,136 patent/US8466284B2/en not_active Expired - Fee Related
- 2008-11-05 CA CA2703996A patent/CA2703996A1/en not_active Abandoned
- 2008-11-05 PE PE2008001893A patent/PE20091565A1/es not_active Application Discontinuation
- 2008-11-05 TW TW097142665A patent/TW200924770A/zh unknown
- 2008-11-05 EA EA201000702A patent/EA017297B1/ru not_active IP Right Cessation
- 2008-11-05 JP JP2010531996A patent/JP2011502982A/ja not_active Ceased
- 2008-11-05 MX MX2010004673A patent/MX2010004673A/es active IP Right Grant
- 2008-11-05 CL CL2008003301A patent/CL2008003301A1/es unknown
- 2008-11-05 KR KR1020107012294A patent/KR20100096131A/ko not_active Ceased
- 2008-11-05 CN CN2008801241402A patent/CN101918391B/zh not_active Expired - Fee Related
- 2008-11-06 UY UY31456A patent/UY31456A1/es not_active Application Discontinuation
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2010
- 2010-04-19 IL IL205209A patent/IL205209A0/en unknown
- 2010-04-20 CO CO10046222A patent/CO6270241A2/es not_active Application Discontinuation
- 2010-04-22 ZA ZA2010/02853A patent/ZA201002853B/en unknown
- 2010-05-06 NI NI201000079A patent/NI201000079A/es unknown
- 2010-05-06 SV SV2010003559A patent/SV2010003559A/es not_active Application Discontinuation
- 2010-05-06 CR CR11416A patent/CR11416A/es not_active Application Discontinuation
- 2010-05-06 DO DO2010000134A patent/DOP2010000134A/es unknown
Also Published As
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|---|---|
| AR069206A1 (es) | 2010-01-06 |
| ZA201002853B (en) | 2011-10-26 |
| BRPI0819258A2 (pt) | 2017-05-02 |
| IL205209A0 (en) | 2010-12-30 |
| KR20100096131A (ko) | 2010-09-01 |
| PE20091565A1 (es) | 2009-11-06 |
| CO6270241A2 (es) | 2011-04-20 |
| MX2010004673A (es) | 2010-05-27 |
| AU2008325288B2 (en) | 2011-12-22 |
| JP2011502982A (ja) | 2011-01-27 |
| UY31456A1 (es) | 2009-07-17 |
| CN101918391A (zh) | 2010-12-15 |
| EP2217591A4 (en) | 2011-10-26 |
| NI201000079A (es) | 2011-03-24 |
| EA201000702A1 (ru) | 2010-12-30 |
| CA2703996A1 (en) | 2009-05-14 |
| WO2009061271A1 (en) | 2009-05-14 |
| EP2217591A1 (en) | 2010-08-18 |
| CR11416A (es) | 2010-08-27 |
| US20100280048A1 (en) | 2010-11-04 |
| SV2010003559A (es) | 2010-09-13 |
| DOP2010000134A (es) | 2010-10-15 |
| AU2008325288A1 (en) | 2009-05-14 |
| CN101918391B (zh) | 2013-06-05 |
| CL2008003301A1 (es) | 2009-10-16 |
| EA017297B1 (ru) | 2012-11-30 |
| US8466284B2 (en) | 2013-06-18 |
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