TW200524902A - 2-substituted benzimidazole piperidines analogs as selective melanin concentrating hormone receptor antagonists for the treatment of obesity and related disorders - Google Patents

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Publication number

TW200524902A

TW200524902A TW093125667A TW93125667A TW200524902A TW 200524902 A TW200524902 A TW 200524902A TW 093125667 A TW093125667 A TW 093125667A TW 93125667 A TW93125667 A TW 93125667A TW 200524902 A TW200524902 A TW 200524902A

Authority

TW

Taiwan

Prior art keywords

compound

group

doc

substituted

nr8r9

Prior art date

2003-08-29

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• 235000020824 obesity Nutrition 0.000 title claims abstract description 24
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• 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title claims description 20
• 102000029828 Melanin-concentrating hormone receptor Human genes 0.000 title description 4
• 108010047068 Melanin-concentrating hormone receptor Proteins 0.000 title description 4
• 229940123502 Hormone receptor antagonist Drugs 0.000 title 1
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• 150000003839 salts Chemical class 0.000 claims description 52
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• 125000003118 aryl group Chemical group 0.000 claims description 31
• 125000001072 heteroaryl group Chemical group 0.000 claims description 24
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