TR200402754T4 - Yeni benzosultam oksazolidinon antibakteriyel maddeler. - Google Patents

Yeni benzosultam oksazolidinon antibakteriyel maddeler.

Info

Publication number
TR200402754T4
TR200402754T4 TR2004/02754T TR200402754T TR200402754T4 TR 200402754 T4 TR200402754 T4 TR 200402754T4 TR 2004/02754 T TR2004/02754 T TR 2004/02754T TR 200402754 T TR200402754 T TR 200402754T TR 200402754 T4 TR200402754 T4 TR 200402754T4
Authority
TR
Turkey
Prior art keywords
benzosultam
new
antibacterial agents
oxazolidinone antibacterial
oxazolidinone
Prior art date
Application number
TR2004/02754T
Other languages
English (en)
Inventor
L. Ciske Fred
J. Genin Michael
Original Assignee
Pharmacia & Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Company filed Critical Pharmacia & Upjohn Company
Publication of TR200402754T4 publication Critical patent/TR200402754T4/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Bu bulus M'nin- CH2-veya-CH2CH2-oldugu formül (I)'e sahip olan ve güçlü antibakteriyel etkiler sergileyen bir bilesik saglar.
TR2004/02754T 2000-03-31 2001-03-27 Yeni benzosultam oksazolidinon antibakteriyel maddeler. TR200402754T4 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19363100P 2000-03-31 2000-03-31

Publications (1)

Publication Number Publication Date
TR200402754T4 true TR200402754T4 (tr) 2004-12-21

Family

ID=22714397

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2004/02754T TR200402754T4 (tr) 2000-03-31 2001-03-27 Yeni benzosultam oksazolidinon antibakteriyel maddeler.

Country Status (21)

Country Link
US (1) US6365612B2 (tr)
EP (1) EP1268475B1 (tr)
JP (1) JP2003529600A (tr)
KR (1) KR20020084274A (tr)
CN (1) CN1406237A (tr)
AR (1) AR035481A1 (tr)
AT (1) ATE277040T1 (tr)
AU (2) AU4754001A (tr)
BR (1) BR0108810A (tr)
CA (1) CA2399275A1 (tr)
DE (1) DE60105786T2 (tr)
DK (1) DK1268475T3 (tr)
ES (1) ES2227166T3 (tr)
MX (1) MXPA02009317A (tr)
NZ (1) NZ521689A (tr)
PE (1) PE20011124A1 (tr)
PT (1) PT1268475E (tr)
SI (1) SI1268475T1 (tr)
TR (1) TR200402754T4 (tr)
WO (1) WO2001074812A1 (tr)
ZA (1) ZA200207003B (tr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ2002186A3 (cs) * 1999-07-16 2002-09-11 Basf Aktiengesellschaft Způsob přípravy substituovaných benzothiazolových sloučenin
US7012088B2 (en) * 2003-02-24 2006-03-14 Pharmacia & Upjohn Company Indolone oxazolidinones and derivatives thereof
DE102004026532A1 (de) * 2004-05-29 2006-01-05 Sanofi-Aventis Deutschland Gmbh Substituierte Oxazol-Benzoisothiazoldioxidderivate, Verfahren zu deren Herstellung und deren Verwendung
WO2006106426A1 (en) * 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc An oxindole oxazolidinone as antibacterial agent
US7956193B2 (en) * 2007-05-04 2011-06-07 University Of South Florida Intramolecular C-H amination with sulfonyl azides
WO2009146032A2 (en) * 2008-03-31 2009-12-03 University Of South Florida Metal porphyrin catalyzed olefin aziridination with sulfonyl azides

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3635964A (en) * 1969-02-10 1972-01-18 Colgate Palmolive Co 5-morpholinyl-2 1-benzisothiazolines
US5036093A (en) 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US5036092A (en) 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US5039690A (en) 1987-10-09 1991-08-13 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US4965268A (en) 1987-10-09 1990-10-23 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5032605A (en) 1987-10-09 1991-07-16 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US5164510A (en) * 1988-09-15 1992-11-17 The Upjohn Company 5'Indolinyl-5β-amidomethyloxazolidin-2-ones
DE4425609A1 (de) 1994-07-20 1996-01-25 Bayer Ag Benzofuranyl- und Benzothienyloxazolidinone
HRP960159A2 (en) * 1995-04-21 1997-08-31 Bayer Ag Benzocyclopentane oxazolidinones containing heteroatoms
DE19604223A1 (de) 1996-02-06 1997-08-07 Bayer Ag Neue substituierte Oxazolidinone
AR008331A1 (es) 1997-01-23 1999-12-29 Smithkline Beecham Corp Compuestos antagonistas de un receptor de il-8, uso de los mismos para la fabricacion de medicamentos, procedimiento para su obtencion, composicionesfarmaceuticas que los contienen
WO1998034929A1 (en) 1997-02-12 1998-08-13 Smithkline Beecham Corporation Il-8 receptor antagonists
AR015425A1 (es) 1997-09-05 2001-05-02 Smithkline Beecham Corp Compuestos de benzotiazol, composicion farmaceutica que los contiene, su uso en la manufactura de un medicamento, procedimiento para su preparacion,compuestos intermediarios y procedimiento para su preparacion
WO1999036069A1 (en) 1998-01-16 1999-07-22 Smithkline Beecham Corporation Il-8 receptor antagonists
DE19802239A1 (de) 1998-01-22 1999-07-29 Bayer Ag Neue mit Bicyclen substituierte Oxazolidinone

Also Published As

Publication number Publication date
ES2227166T3 (es) 2005-04-01
MXPA02009317A (es) 2003-03-12
EP1268475A1 (en) 2003-01-02
PT1268475E (pt) 2004-11-30
CN1406237A (zh) 2003-03-26
JP2003529600A (ja) 2003-10-07
PE20011124A1 (es) 2001-10-28
NZ521689A (en) 2004-05-28
WO2001074812A1 (en) 2001-10-11
AU4754001A (en) 2001-10-15
US20010047018A1 (en) 2001-11-29
ATE277040T1 (de) 2004-10-15
AR035481A1 (es) 2004-06-02
AU2001247540B2 (en) 2004-08-19
BR0108810A (pt) 2002-11-05
ZA200207003B (en) 2003-12-01
DE60105786D1 (de) 2004-10-28
EP1268475B1 (en) 2004-09-22
DE60105786T2 (de) 2006-02-23
SI1268475T1 (en) 2005-02-28
KR20020084274A (ko) 2002-11-04
CA2399275A1 (en) 2001-10-11
US6365612B2 (en) 2002-04-02
DK1268475T3 (da) 2004-12-20

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