TR200102680T2 - 1,3,4- Oksadiazol türevleri ve üretilmeleri için bir işlem - Google Patents

1,3,4- Oksadiazol türevleri ve üretilmeleri için bir işlem

Info

Publication number
TR200102680T2
TR200102680T2 TR2001/02680T TR200102680T TR200102680T2 TR 200102680 T2 TR200102680 T2 TR 200102680T2 TR 2001/02680 T TR2001/02680 T TR 2001/02680T TR 200102680 T TR200102680 T TR 200102680T TR 200102680 T2 TR200102680 T2 TR 200102680T2
Authority
TR
Turkey
Prior art keywords
oxadiazole derivatives
formula
group
production
derivatives represented
Prior art date
Application number
TR2001/02680T
Other languages
English (en)
Inventor
Kojima Tsutomu
Hachiya Katsutoshi
Ohmoto Kazuyuki
Original Assignee
Ono Pharmaceutical Co. Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ono Pharmaceutical Co. Ltd. filed Critical Ono Pharmaceutical Co. Ltd.
Publication of TR200102680T2 publication Critical patent/TR200102680T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Formül (I) ile temsil edilen oksadiazol türevleri: (buradaki R1, bir hidrojen atomunu veya amino-koruyucu bir grubu temsil eder; R2, R3 ve R4'ün herbiri bagumsiz olarak bir alkil grubunu, ikameli olabilen bir fenil grubunu veya bir 3,4-metilendioksifenil grubunu temsil eder), bunlari üretilmesi için bir islem ve yukarda kitürevi kullanarak, formül (II) ile temsil edilen oksadiazol türevlerinin üretilmesi için bir islem: (buradaki bütün semboller, yukarida tanimlananlarla ayni anlamara sahiptirler). Bulusa uygun olarak, formül (II) ile temsil edilen bilesik, daha az basamakla, yüksek bir verimle üretilir.
TR2001/02680T 1999-03-12 2000-03-10 1,3,4- Oksadiazol türevleri ve üretilmeleri için bir işlem TR200102680T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP6606599 1999-03-12

Publications (1)

Publication Number Publication Date
TR200102680T2 true TR200102680T2 (tr) 2002-07-22

Family

ID=13305090

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/02680T TR200102680T2 (tr) 1999-03-12 2000-03-10 1,3,4- Oksadiazol türevleri ve üretilmeleri için bir işlem

Country Status (16)

Country Link
US (2) US6534658B1 (tr)
EP (1) EP1162199A4 (tr)
KR (1) KR20010102569A (tr)
CN (1) CN1350525A (tr)
AU (1) AU2941200A (tr)
BR (1) BR0008936A (tr)
CA (1) CA2367418A1 (tr)
HU (1) HUP0200476A3 (tr)
MX (1) MXPA01009165A (tr)
NO (1) NO20014393L (tr)
NZ (1) NZ513921A (tr)
RU (1) RU2001124908A (tr)
TR (1) TR200102680T2 (tr)
TW (1) TW482763B (tr)
WO (1) WO2000055145A1 (tr)
ZA (1) ZA200107256B (tr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1253144A4 (en) * 2000-02-03 2003-02-12 Ono Pharmaceutical Co 1,3,4-OXADIAZOLE DERIVATIVES AND A METHOD FOR THE PRODUCTION THEREOF
JPWO2002014310A1 (ja) * 2000-08-10 2004-01-15 小野薬品工業株式会社 ２−［５−アミノ−６−オキソ−２−フェニル−１，６−ジヒドロ−１−ピリミジル］−Ｎ−［１−（２−［５−ｔ−ブチル−１，３，４−オキサジアゾリル］カルボニル）−２−（Ｒ，Ｓ）−メチルプロピル］アセトアミド・塩酸塩化合物
CA2421499A1 (en) * 2000-09-08 2003-03-06 Ono Pharmaceutical Co., Ltd. Novel crystals of 1,3,4-oxadiazole derivative, process for producing the same and pharmaceutical agent containing the same as active ingredient
HUP0303631A2 (hu) * 2000-12-26 2004-03-01 Ono Pharmaceutical Co., Ltd. Pirimidinszármazékok és eljárás előállításukra
CN1898215A (zh) * 2003-12-19 2007-01-17 默克公司 有丝分裂驱动蛋白抑制剂
KR20090086802A (ko) * 2008-02-11 2009-08-14 삼성전자주식회사 옥사디아졸렌기를 포함하는 디페노퀴논계 화합물을포함하는 전자사진 감광체 및 이를 채용한 전자사진화상형성장치

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6015791A (en) * 1994-11-21 2000-01-18 Cortech Inc. Serine protease inhibitors-cycloheptane derivatives
US5618792A (en) 1994-11-21 1997-04-08 Cortech, Inc. Substituted heterocyclic compounds useful as inhibitors of (serine proteases) human neutrophil elastase
US5591695A (en) * 1995-02-08 1997-01-07 American Cyanamid Co. Herbicidal [1,3,4]oxadiazoles and thiadiazoles
HUP0100669A3 (en) * 1996-12-06 2001-12-28 Cortech Inc Denver Peptide derivatives as serine protease inhibitors, their use and pharmaceutical compositions comprising thereof

Also Published As

Publication number Publication date
NZ513921A (en) 2001-09-28
EP1162199A4 (en) 2002-06-05
CA2367418A1 (en) 2000-09-21
US6534658B1 (en) 2003-03-18
US20030153758A1 (en) 2003-08-14
CN1350525A (zh) 2002-05-22
BR0008936A (pt) 2002-04-09
HUP0200476A3 (en) 2004-03-29
RU2001124908A (ru) 2004-02-27
EP1162199A1 (en) 2001-12-12
NO20014393D0 (no) 2001-09-10
TW482763B (en) 2002-04-11
ZA200107256B (en) 2002-12-02
KR20010102569A (ko) 2001-11-15
WO2000055145A1 (fr) 2000-09-21
HUP0200476A2 (en) 2002-08-28
AU2941200A (en) 2000-10-04
MXPA01009165A (es) 2002-08-20
NO20014393L (no) 2001-11-08

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