TR199902942T2 - Nikotinik ACh Reseptörlerinde kolinerjik ligandlar olarak 8-Azabisiklo(3.2.1)okt-ene ve okstan türevleri. - Google Patents

Nikotinik ACh Reseptörlerinde kolinerjik ligandlar olarak 8-Azabisiklo(3.2.1)okt-ene ve okstan türevleri.

Info

Publication number
TR199902942T2
TR199902942T2 TR1999/02942T TR9902942T TR199902942T2 TR 199902942 T2 TR199902942 T2 TR 199902942T2 TR 1999/02942 T TR1999/02942 T TR 1999/02942T TR 9902942 T TR9902942 T TR 9902942T TR 199902942 T2 TR199902942 T2 TR 199902942T2
Authority
TR
Turkey
Prior art keywords
azabicyclo
derivatives
oxtane
octene
ach receptors
Prior art date
Application number
TR1999/02942T
Other languages
English (en)
Inventor
Peters Dan
M. Olsen Gunnar
Feldbaek Nielsen Simon
Ostergaard Nielsen Elsebet
Original Assignee
Neurosearch A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurosearch A/S filed Critical Neurosearch A/S
Publication of TR199902942T2 publication Critical patent/TR199902942T2/tr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P1/12—Antidiarrhoeals
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Abstract

Bu bulus, ACh reseptörlerinde kolinerjik ligandlar olan yeni 8-Azabisiklo[3.2.1]okt-2-ene ve türevleri ile ilgilidir. Bu bulusun bilesikleri, merkezi sinir sisteminin kolinerjik sistemi ile ilgili hastaliklarin, agri, iltihabi hastaliklar, yumusak kas kasilmalarinin yol açtigi hastaliklarin tedavisinde ve kimyasal madde tacizinin kesilmesine yardimci madde olarak faydalidir.
TR1999/02942T 1997-05-30 1998-05-29 Nikotinik ACh Reseptörlerinde kolinerjik ligandlar olarak 8-Azabisiklo(3.2.1)okt-ene ve okstan türevleri. TR199902942T2 (tr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DK62797 1997-05-30
DK150297 1997-12-19
DK40898 1998-03-24
DK53498 1998-04-16

Publications (1)

Publication Number Publication Date
TR199902942T2 true TR199902942T2 (tr) 2000-04-21

Family

ID=27439314

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1999/02942T TR199902942T2 (tr) 1997-05-30 1998-05-29 Nikotinik ACh Reseptörlerinde kolinerjik ligandlar olarak 8-Azabisiklo(3.2.1)okt-ene ve okstan türevleri.

Country Status (23)

Country Link
US (2) US6645977B1 (tr)
EP (1) EP0984965B1 (tr)
JP (1) JP4447663B2 (tr)
KR (1) KR100589872B1 (tr)
CN (1) CN1157392C (tr)
AT (1) ATE267199T1 (tr)
AU (1) AU745964B2 (tr)
BR (1) BR9809697A (tr)
CA (1) CA2289574C (tr)
CZ (1) CZ298824B6 (tr)
DE (1) DE69823994T2 (tr)
DK (1) DK0984965T3 (tr)
EE (1) EE04057B1 (tr)
HK (1) HK1027353A1 (tr)
HU (1) HUP0002713A3 (tr)
IL (2) IL132437A0 (tr)
IS (1) IS2092B (tr)
NO (1) NO325513B1 (tr)
NZ (1) NZ500642A (tr)
RU (1) RU2186780C2 (tr)
SK (1) SK284994B6 (tr)
TR (1) TR199902942T2 (tr)
WO (1) WO1998054181A1 (tr)

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CA2289574A1 (en) 1998-12-03
DE69823994D1 (de) 2004-06-24
KR20010013154A (ko) 2001-02-26
CN1157392C (zh) 2004-07-14
HUP0002713A3 (en) 2001-02-28
US6645977B1 (en) 2003-11-11
IS2092B (is) 2006-04-12
HK1027353A1 (en) 2001-01-12
CA2289574C (en) 2007-04-24
SK162699A3 (en) 2000-07-11
EE9900529A (et) 2000-06-15
EP0984965A1 (en) 2000-03-15
IL132437A (en) 2006-12-10
IL132437A0 (en) 2001-03-19
NO995850D0 (no) 1999-11-29
CN1257499A (zh) 2000-06-21
JP4447663B2 (ja) 2010-04-07
US6964972B2 (en) 2005-11-15
HUP0002713A2 (hu) 2001-01-29
DE69823994T2 (de) 2009-09-24
US20040019207A1 (en) 2004-01-29
IS5243A (is) 1999-11-10
NO995850L (no) 1999-11-29
ATE267199T1 (de) 2004-06-15
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NO325513B1 (no) 2008-05-26
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AU745964B2 (en) 2002-04-11
CZ298824B6 (cs) 2008-02-20
CZ414799A3 (cs) 2000-02-16
WO1998054181A1 (en) 1998-12-03
AU7426198A (en) 1998-12-30
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