TR199801432A3 - Rasemizasyona karsi stabilize edilmis farmakolojik silansetron karisimlari. - Google Patents

Rasemizasyona karsi stabilize edilmis farmakolojik silansetron karisimlari.

Info

Publication number
TR199801432A3
TR199801432A3 TR1998/01432A TR9801432A TR199801432A3 TR 199801432 A3 TR199801432 A3 TR 199801432A3 TR 1998/01432 A TR1998/01432 A TR 1998/01432A TR 9801432 A TR9801432 A TR 9801432A TR 199801432 A3 TR199801432 A3 TR 199801432A3
Authority
TR
Turkey
Prior art keywords
cilansetron
pharmacological
stabilized against
against racemization
mixtures stabilized
Prior art date
Application number
TR1998/01432A
Other languages
English (en)
Other versions
TR199801432A2 (tr
Inventor
Bonnacker Ingo
Koehn Hartmut
Kristen Gerhard
Reichel Christine
Original Assignee
Solvay Pharmaceuticals Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharmaceuticals Gmbh filed Critical Solvay Pharmaceuticals Gmbh
Publication of TR199801432A3 publication Critical patent/TR199801432A3/tr
Publication of TR199801432A2 publication Critical patent/TR199801432A2/tr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/475Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
TR1998/01432A 1997-08-01 1998-07-23 Rasemizasyona karsi stabilize edilmis farmakolojik silansetron karisimlari. TR199801432A2 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19733271 1997-08-01
DE19813661A DE19813661A1 (de) 1997-08-01 1998-03-27 Gegen Racemisierung stabilisierte pharmazeutische Zubereitungen von Cilansetron

Publications (2)

Publication Number Publication Date
TR199801432A3 true TR199801432A3 (tr) 1999-02-22
TR199801432A2 TR199801432A2 (tr) 1999-02-22

Family

ID=7837672

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1998/01432A TR199801432A2 (tr) 1997-08-01 1998-07-23 Rasemizasyona karsi stabilize edilmis farmakolojik silansetron karisimlari.

Country Status (29)

Country Link
US (1) US5977127A (tr)
EP (1) EP0895782B1 (tr)
JP (1) JP4324260B2 (tr)
KR (1) KR100515201B1 (tr)
CN (1) CN1117565C (tr)
AR (1) AR010178A1 (tr)
AT (1) ATE283706T1 (tr)
AU (1) AU743043B2 (tr)
BR (1) BR9803730A (tr)
CA (1) CA2244389C (tr)
CZ (1) CZ295072B6 (tr)
DE (2) DE19813661A1 (tr)
DK (1) DK0895782T3 (tr)
DZ (1) DZ2560A1 (tr)
ES (1) ES2234051T3 (tr)
HK (1) HK1017611A1 (tr)
HU (1) HUP9801712A3 (tr)
ID (1) ID20685A (tr)
IL (1) IL125403A (tr)
NO (1) NO323229B1 (tr)
NZ (1) NZ331083A (tr)
PL (1) PL191767B1 (tr)
PT (1) PT895782E (tr)
RU (1) RU2199318C2 (tr)
SK (1) SK284916B6 (tr)
TR (1) TR199801432A2 (tr)
TW (1) TW509570B (tr)
UA (1) UA62924C2 (tr)
ZA (1) ZA986715B (tr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7452545B2 (en) * 2001-11-13 2008-11-18 Yu Ruey J Oligosaccharide aldonic acids and their topical use
ES2261671T3 (es) * 2001-03-26 2006-11-16 Novartis Ag Mezcla farmaceutica que incluye una estaurosporina poco soluble en agua, un surfactante y un polimero soluble en agua.
US20040048874A1 (en) * 2001-05-22 2004-03-11 Bardsley Hazel Judith New therapeutic use of 4-(2-fluorophenyl)-6-methyl-2-(1-piperazinyl)thieno[2,3-D]pyrimidine
GB0216027D0 (en) * 2002-07-10 2002-08-21 Arachnova Therapeutics Ltd New therapeutic use
NZ541009A (en) * 2003-01-13 2007-09-28 Dynogen Pharmaceuticals Inc Method of treating nausea, vomiting, retching or any combination thereof
EP1558081A4 (en) * 2003-01-13 2006-06-14 Dynogen Pharmaceuticals Inc METHOD OF TREATING FUNCTIONAL INTESTINAL DISORDERS
AU2004227945B2 (en) * 2003-04-04 2006-10-26 Dynogen Pharmaceuticals, Inc. Method of treating lower urinary tract disorders
US7820690B2 (en) * 2004-03-19 2010-10-26 Solvay Pharmaceuticals Gmbh Method of treating or inhibiting a non-digestive tract derived abdominal disorder associated with pain using a 5-HT, receptor antagonist
US20060293309A1 (en) * 2005-03-28 2006-12-28 Dynogen Pharmaceuticals, Inc. Method of treating disorders and conditions using peripherally-restricted antagonists and inhibitors
KR20110044780A (ko) 2008-08-14 2011-04-29 교린 세이야꾸 가부시키 가이샤 안정화된 의약 조성물
JPWO2021100728A1 (tr) 2019-11-20 2021-05-27

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3885357T2 (de) * 1987-06-29 1994-03-24 Duphar Int Res Anellierte Indolderivate.
DE4238553A1 (de) * 1992-11-14 1994-05-19 Kali Chemie Pharma Gmbh Neue Imidazol-1-yl-Verbindungen enthaltende Arzneimittel
AU702594B2 (en) * 1995-10-13 1999-02-25 Duphar International Research B.V. Process for the preparation of enantiomerically pure imidazolyl compounds

Also Published As

Publication number Publication date
PL191767B1 (pl) 2006-06-30
CZ236798A3 (cs) 1999-02-17
AU7863098A (en) 1999-02-11
DK0895782T3 (da) 2005-01-03
US5977127A (en) 1999-11-02
SK284916B6 (sk) 2006-02-02
HUP9801712A2 (hu) 1999-04-28
HK1017611A1 (en) 1999-11-26
EP0895782A3 (de) 2001-01-31
CN1207292A (zh) 1999-02-10
CA2244389A1 (en) 1999-02-01
IL125403A0 (en) 1999-03-12
ID20685A (id) 1999-02-18
NZ331083A (en) 2000-01-28
DE59812317D1 (de) 2005-01-05
TR199801432A2 (tr) 1999-02-22
BR9803730A (pt) 2000-03-28
NO983540L (no) 1999-02-02
HUP9801712A3 (en) 2001-08-28
EP0895782A2 (de) 1999-02-10
ES2234051T3 (es) 2005-06-16
TW509570B (en) 2002-11-11
AU743043B2 (en) 2002-01-17
CA2244389C (en) 2008-01-15
KR100515201B1 (ko) 2005-12-09
SK100998A3 (en) 1999-02-11
CZ295072B6 (cs) 2005-05-18
JPH1192369A (ja) 1999-04-06
ZA986715B (en) 1999-02-04
RU2199318C2 (ru) 2003-02-27
HU9801712D0 (en) 1998-09-28
DE19813661A1 (de) 1999-02-04
KR19990023194A (ko) 1999-03-25
UA62924C2 (en) 2004-01-15
PT895782E (pt) 2005-02-28
IL125403A (en) 2001-11-25
PL327786A1 (en) 1999-02-15
DZ2560A1 (fr) 2003-02-15
EP0895782B1 (de) 2004-12-01
JP4324260B2 (ja) 2009-09-02
CN1117565C (zh) 2003-08-13
NO323229B1 (no) 2007-02-05
NO983540D0 (no) 1998-07-31
AR010178A1 (es) 2000-05-17
ATE283706T1 (de) 2004-12-15

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