HUP9801712A3 - Pharmaceutical compositions containing cilansetron stabilized against racemisation, their production and use of stobilizing additive agents - Google Patents
Pharmaceutical compositions containing cilansetron stabilized against racemisation, their production and use of stobilizing additive agentsInfo
- Publication number
- HUP9801712A3 HUP9801712A3 HU9801712A HUP9801712A HUP9801712A3 HU P9801712 A3 HUP9801712 A3 HU P9801712A3 HU 9801712 A HU9801712 A HU 9801712A HU P9801712 A HUP9801712 A HU P9801712A HU P9801712 A3 HUP9801712 A3 HU P9801712A3
- Authority
- HU
- Hungary
- Prior art keywords
- stobilizing
- racemisation
- production
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
- 239000000654 additive Substances 0.000 title 1
- 230000000996 additive effect Effects 0.000 title 1
- 239000003795 chemical substances by application Substances 0.000 title 1
- NCNFDKWULDWJDS-OAHLLOKOSA-N cilansetron Chemical compound CC1=NC=CN1C[C@@H]1C(=O)C(C=2C=3N4CCCC=3C=CC=2)=C4CC1 NCNFDKWULDWJDS-OAHLLOKOSA-N 0.000 title 1
- 229960002099 cilansetron Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/475—Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19733271 | 1997-08-01 | ||
| DE19813661A DE19813661A1 (en) | 1997-08-01 | 1998-03-27 | Pharmaceutical preparations from Cilansetron stabilized against racemization |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| HU9801712D0 HU9801712D0 (en) | 1998-09-28 |
| HUP9801712A2 HUP9801712A2 (en) | 1999-04-28 |
| HUP9801712A3 true HUP9801712A3 (en) | 2001-08-28 |
Family
ID=7837672
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU9801712A HUP9801712A3 (en) | 1997-08-01 | 1998-07-29 | Pharmaceutical compositions containing cilansetron stabilized against racemisation, their production and use of stobilizing additive agents |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US5977127A (en) |
| EP (1) | EP0895782B1 (en) |
| JP (1) | JP4324260B2 (en) |
| KR (1) | KR100515201B1 (en) |
| CN (1) | CN1117565C (en) |
| AR (1) | AR010178A1 (en) |
| AT (1) | ATE283706T1 (en) |
| AU (1) | AU743043B2 (en) |
| BR (1) | BR9803730A (en) |
| CA (1) | CA2244389C (en) |
| CZ (1) | CZ295072B6 (en) |
| DE (2) | DE19813661A1 (en) |
| DK (1) | DK0895782T3 (en) |
| DZ (1) | DZ2560A1 (en) |
| ES (1) | ES2234051T3 (en) |
| HK (1) | HK1017611A1 (en) |
| HU (1) | HUP9801712A3 (en) |
| ID (1) | ID20685A (en) |
| IL (1) | IL125403A (en) |
| NO (1) | NO323229B1 (en) |
| NZ (1) | NZ331083A (en) |
| PL (1) | PL191767B1 (en) |
| PT (1) | PT895782E (en) |
| RU (1) | RU2199318C2 (en) |
| SK (1) | SK284916B6 (en) |
| TR (1) | TR199801432A3 (en) |
| TW (1) | TW509570B (en) |
| UA (1) | UA62924C2 (en) |
| ZA (1) | ZA986715B (en) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7452545B2 (en) * | 2001-11-13 | 2008-11-18 | Yu Ruey J | Oligosaccharide aldonic acids and their topical use |
| AU2002304784A1 (en) * | 2001-03-26 | 2002-10-08 | Novartis Pharma Gmbh | Pharmaceutical composition comprising a poorly water-soluble active ingredient, a surfactant and a water-soluble polymer |
| GB0216027D0 (en) * | 2002-07-10 | 2002-08-21 | Arachnova Therapeutics Ltd | New therapeutic use |
| US20040048874A1 (en) * | 2001-05-22 | 2004-03-11 | Bardsley Hazel Judith | New therapeutic use of 4-(2-fluorophenyl)-6-methyl-2-(1-piperazinyl)thieno[2,3-D]pyrimidine |
| DE602004005814T2 (en) * | 2003-01-13 | 2008-01-10 | Dynogen Pharmaceuticals Inc., Waltham | PROCEDURE FOR TREATING EVILNESS, INFRINGEMENT, ORGANIZATION OR ANY COMBINATION THEREOF |
| AU2004204825B2 (en) * | 2003-01-13 | 2007-07-19 | Dynogen Pharmaceuticals, Inc. | Method of treating functional bowel disorders |
| EP1539181B1 (en) * | 2003-04-04 | 2007-06-27 | Dynogen Pharmaceuticals Inc. | Method of treating lower urinary tract disorders |
| US7820690B2 (en) * | 2004-03-19 | 2010-10-26 | Solvay Pharmaceuticals Gmbh | Method of treating or inhibiting a non-digestive tract derived abdominal disorder associated with pain using a 5-HT, receptor antagonist |
| US20060293309A1 (en) * | 2005-03-28 | 2006-12-28 | Dynogen Pharmaceuticals, Inc. | Method of treating disorders and conditions using peripherally-restricted antagonists and inhibitors |
| EP2327406A4 (en) * | 2008-08-14 | 2014-04-09 | Kyorin Seiyaku Kk | Stabilized pharmaceutical composition |
| WO2021100728A1 (en) | 2019-11-20 | 2021-05-27 | 塩野義製薬株式会社 | 6,7-unsaturated-7-carbamoyl morphinan derivative-containing solid formulation |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0297651B1 (en) * | 1987-06-29 | 1993-11-03 | Duphar International Research B.V | Anellated indole derivatives |
| DE4238553A1 (en) * | 1992-11-14 | 1994-05-19 | Kali Chemie Pharma Gmbh | New drugs containing imidazol-1-yl compounds |
| AU702594B2 (en) * | 1995-10-13 | 1999-02-25 | Duphar International Research B.V. | Process for the preparation of enantiomerically pure imidazolyl compounds |
-
1998
- 1998-03-27 DE DE19813661A patent/DE19813661A1/en not_active Withdrawn
- 1998-06-05 CN CN98109652A patent/CN1117565C/en not_active Expired - Fee Related
- 1998-06-17 TW TW087109651A patent/TW509570B/en not_active IP Right Cessation
- 1998-06-18 AR ARP980102904A patent/AR010178A1/en active IP Right Grant
- 1998-07-11 KR KR10-1998-0028014A patent/KR100515201B1/en not_active IP Right Cessation
- 1998-07-15 DZ DZ980170A patent/DZ2560A1/en active
- 1998-07-20 IL IL12540398A patent/IL125403A/en not_active IP Right Cessation
- 1998-07-22 AT AT98113643T patent/ATE283706T1/en active
- 1998-07-22 DE DE59812317T patent/DE59812317D1/en not_active Expired - Lifetime
- 1998-07-22 EP EP98113643A patent/EP0895782B1/en not_active Expired - Lifetime
- 1998-07-22 ES ES98113643T patent/ES2234051T3/en not_active Expired - Lifetime
- 1998-07-22 PT PT98113643T patent/PT895782E/en unknown
- 1998-07-22 DK DK98113643T patent/DK0895782T3/en active
- 1998-07-23 TR TR1998/01432A patent/TR199801432A3/en unknown
- 1998-07-24 SK SK1009-98A patent/SK284916B6/en not_active IP Right Cessation
- 1998-07-24 NZ NZ331083A patent/NZ331083A/en not_active IP Right Cessation
- 1998-07-27 CZ CZ19982367A patent/CZ295072B6/en not_active IP Right Cessation
- 1998-07-28 ZA ZA986715A patent/ZA986715B/en unknown
- 1998-07-29 HU HU9801712A patent/HUP9801712A3/en unknown
- 1998-07-29 RU RU98114668/14A patent/RU2199318C2/en not_active IP Right Cessation
- 1998-07-31 BR BR9803730-7A patent/BR9803730A/en not_active Application Discontinuation
- 1998-07-31 JP JP21707598A patent/JP4324260B2/en not_active Expired - Fee Related
- 1998-07-31 CA CA002244389A patent/CA2244389C/en not_active Expired - Fee Related
- 1998-07-31 AU AU78630/98A patent/AU743043B2/en not_active Ceased
- 1998-07-31 UA UA98074202A patent/UA62924C2/en unknown
- 1998-07-31 PL PL327786A patent/PL191767B1/en not_active IP Right Cessation
- 1998-07-31 NO NO19983540A patent/NO323229B1/en not_active IP Right Cessation
- 1998-07-31 US US09/126,751 patent/US5977127A/en not_active Expired - Lifetime
- 1998-08-03 ID IDP981075A patent/ID20685A/en unknown
-
1999
- 1999-06-30 HK HK99102775A patent/HK1017611A1/en not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA9A | Lapse of provisional patent protection due to relinquishment or protection considered relinquished |