SMT201700533T1 - Composti, composizioni e metodi utili per la mobilitazione del colesterolo - Google Patents

Composti, composizioni e metodi utili per la mobilitazione del colesterolo

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Publication number
SMT201700533T1
SMT201700533T1 SM20170533T SMT201700533T SMT201700533T1 SM T201700533 T1 SMT201700533 T1 SM T201700533T1 SM 20170533 T SM20170533 T SM 20170533T SM T201700533 T SMT201700533 T SM T201700533T SM T201700533 T1 SMT201700533 T1 SM T201700533T1
Authority
SM
San Marino
Prior art keywords
compositions
compounds
methods useful
mobilisation
cholesterol
Prior art date
Application number
SM20170533T
Other languages
English (en)
Italian (it)
Inventor
Daniela Carmen Oniciu
Jean-Louis Henri Dasseux
Ronald Barbaras
Valery Kochubey
Dmitry Kovalsky
Oleg Gennadievich Rodin
Otto Geoffroy
Anna Rzepiela
Original Assignee
Cerenis Therapeutics Holding Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cerenis Therapeutics Holding Sa filed Critical Cerenis Therapeutics Holding Sa
Publication of SMT201700533T1 publication Critical patent/SMT201700533T1/it

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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