SK5072003A3 - Polysubstituted imidazopyridines as gastric secretion inhibitors - Google Patents
Polysubstituted imidazopyridines as gastric secretion inhibitors Download PDFInfo
- Publication number
- SK5072003A3 SK5072003A3 SK507-2003A SK5072003A SK5072003A3 SK 5072003 A3 SK5072003 A3 SK 5072003A3 SK 5072003 A SK5072003 A SK 5072003A SK 5072003 A3 SK5072003 A3 SK 5072003A3
- Authority
- SK
- Slovakia
- Prior art keywords
- alkoxy
- alkyl
- hydrogen
- halogen
- hydroxyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00123133 | 2000-10-25 | ||
| PCT/EP2001/012207 WO2002034749A1 (en) | 2000-10-25 | 2001-10-23 | Polysubstituted imidazopyridines as gastric secretion inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK5072003A3 true SK5072003A3 (en) | 2003-09-11 |
Family
ID=8170193
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK507-2003A SK5072003A3 (en) | 2000-10-25 | 2001-10-23 | Polysubstituted imidazopyridines as gastric secretion inhibitors |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US6869949B2 (pt) |
| EP (1) | EP1332143A1 (pt) |
| JP (1) | JP2004512338A (pt) |
| KR (1) | KR20040011423A (pt) |
| CN (1) | CN1692113A (pt) |
| AU (2) | AU2002210563B2 (pt) |
| BR (1) | BR0114873A (pt) |
| CA (1) | CA2426616A1 (pt) |
| EA (1) | EA008151B1 (pt) |
| HR (1) | HRP20030323A2 (pt) |
| HU (1) | HUP0302308A2 (pt) |
| IL (1) | IL154850A0 (pt) |
| MX (1) | MXPA03003706A (pt) |
| NO (1) | NO325736B1 (pt) |
| NZ (1) | NZ525281A (pt) |
| PL (1) | PL360412A1 (pt) |
| SK (1) | SK5072003A3 (pt) |
| WO (1) | WO2002034749A1 (pt) |
| ZA (1) | ZA200302038B (pt) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2426616A1 (en) * | 2000-10-25 | 2002-05-02 | Altana Pharma Ag | Polysubstituted imidazopyridines as gastric secretion inhibitors |
| DE10145457A1 (de) * | 2001-09-14 | 2003-04-03 | Basf Ag | Substituierte Imidazo[1,2-a]-5,6,7,8-tetrahydropyridin-8-one, Verfahren zu ihrer Herstellung, sowie deren Verwendung zur Herstellung von Imidazo[1,2,-a]pyridinen |
| JP2005519933A (ja) | 2002-02-15 | 2005-07-07 | アルタナ ファルマ アクチエンゲゼルシャフト | 三環式ｎ−アシル化合物 |
| TWI295575B (en) * | 2002-04-24 | 2008-04-11 | Altana Pharma Ag | Nitrosated imidazopyridines |
| PL375933A1 (en) * | 2002-12-20 | 2005-12-12 | Altana Pharma Ag | 8-trialkylsiloxy-2-methyl-9-phenyl-7-oxo-7,8,9,10-tetrahydroimidazo[1,2-h][1,7]naphthyridines |
| WO2004071391A2 (en) * | 2003-02-17 | 2004-08-26 | Altana Pharma Ag | Imidazopyridines containing combinations and their use in treating gastrointestinal inflammatory disorders |
| CN1764665A (zh) * | 2003-04-03 | 2006-04-26 | 奥坦纳医药公司 | 咪唑并吡啶－8－酮的生产方法 |
| AR044129A1 (es) * | 2003-05-06 | 2005-08-24 | Altana Pharma Ag | Compuestos intermedios de imidazopiridina. proceso de preparacion. |
| CN1874772A (zh) | 2003-11-03 | 2006-12-06 | 阿斯利康(瑞典)有限公司 | 治疗隐匿性胃食管反流的咪唑并[1,2－a]吡啶衍生物 |
| AR046893A1 (es) * | 2003-12-16 | 2005-12-28 | Altana Pharma Ag | Bencimidazoles triciclicos |
| WO2005058894A1 (en) | 2003-12-19 | 2005-06-30 | Altana Pharma Ag | Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives |
| AR046941A1 (es) * | 2003-12-19 | 2006-01-04 | Altana Pharma Ag | Imidazopiridinas triciclicas y su uso como inhibidores de secrecion de acido gastrico |
| CA2582256A1 (en) * | 2004-10-01 | 2006-04-13 | Altana Pharma Ag | Substituted tricyclic benzimidazoles |
| AR051375A1 (es) * | 2004-10-15 | 2007-01-10 | Altana Pharma Ag | Imidazopiridinas difluoro substituidas |
| WO2008058990A1 (en) * | 2006-11-16 | 2008-05-22 | Nycomed Gmbh | 7,7-disubstituted pyrano-[2,3-c]-imidazo-[1,2-a]-pyridine derivatives and their use as gastric acid secretion inhibitors |
| WO2012027240A1 (en) * | 2010-08-23 | 2012-03-01 | Schering Corporation | Fused tricyclic inhibitors of mammalian target of rapamycin |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4468400A (en) * | 1982-12-20 | 1984-08-28 | Schering Corporation | Antiulcer tricyclic imidazo [1,2-a]pyridines |
| US4673679A (en) * | 1986-05-14 | 1987-06-16 | E. I. Du Pont De Nemours And Company | Use of prodrugs of 3-hydroxymorphinans to prevent bitter taste upon buccal, nasal or sublingual administration |
| WO1992021341A1 (en) * | 1991-05-31 | 1992-12-10 | Pfizer Inc. | Use of rapamycin prodrugs as immunosuppressant agents |
| DE4308095A1 (de) * | 1993-03-13 | 1994-09-15 | Hoechst Ag | Prodrug-Derivate von Arzneimittelwirkstoffen mit Hydroxylgruppen, Verfahren zu deren Herstellung und ihre Verwendung |
| SE9401197D0 (sv) * | 1994-04-11 | 1994-04-11 | Astra Ab | Active compounds |
| EA002402B1 (ru) * | 1997-03-24 | 2002-04-25 | Бык Гульден Ломберг Хемише Фабрик Гмбх | Тетрагидропиридо-соединения |
| ZA982445B (en) * | 1997-03-24 | 1998-09-24 | Byk Gulden Lomberg Chem Fab | Tetrahydropyrido compounds |
| CA2289542A1 (en) * | 1997-05-28 | 1998-12-03 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Fused dihydropyrans |
| HUP0001555A3 (en) * | 1997-10-30 | 2001-01-29 | Altana Pharma Ag | Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation |
| PL193616B1 (pl) * | 1998-09-23 | 2007-02-28 | Altana Pharma Ag | Tetrahydropirydoetery |
| EP1127059B1 (en) * | 1998-11-03 | 2008-02-20 | Nycomed GmbH | Imidazonaphthyridines |
| SI1173439T1 (en) * | 1999-04-17 | 2003-10-31 | Altana Pharma Ag | Haloalkoxy imidazonaphthyridines |
| BR0109483A (pt) | 2000-03-29 | 2003-06-10 | Altana Pharma Ag | Pró-drogas de derivados de imidazopiridina |
| MXPA02009550A (es) * | 2000-03-29 | 2004-05-14 | Altana Pharma Ag | Derivados de pirano (2,3,c)imidazo(1,2-a]piridina para el tratamiento de trastornos gastrointestinales. |
| AU783764B2 (en) * | 2000-03-29 | 2005-12-01 | Altana Pharma Ag | Alkylated imidazopyridine derivatives |
| ATE356131T1 (de) * | 2000-03-29 | 2007-03-15 | Altana Pharma Ag | Tricyclische imidazopyridine |
| CA2426616A1 (en) * | 2000-10-25 | 2002-05-02 | Altana Pharma Ag | Polysubstituted imidazopyridines as gastric secretion inhibitors |
-
2001
- 2001-10-23 CA CA002426616A patent/CA2426616A1/en not_active Abandoned
- 2001-10-23 MX MXPA03003706A patent/MXPA03003706A/es active IP Right Grant
- 2001-10-23 AU AU2002210563A patent/AU2002210563B2/en not_active Ceased
- 2001-10-23 IL IL15485001A patent/IL154850A0/xx unknown
- 2001-10-23 CN CNA018177808A patent/CN1692113A/zh active Pending
- 2001-10-23 JP JP2002537739A patent/JP2004512338A/ja active Pending
- 2001-10-23 BR BR0114873-7A patent/BR0114873A/pt not_active IP Right Cessation
- 2001-10-23 EP EP01978447A patent/EP1332143A1/en not_active Withdrawn
- 2001-10-23 WO PCT/EP2001/012207 patent/WO2002034749A1/en active IP Right Grant
- 2001-10-23 PL PL36041201A patent/PL360412A1/xx not_active Application Discontinuation
- 2001-10-23 EA EA200300478A patent/EA008151B1/ru not_active IP Right Cessation
- 2001-10-23 SK SK507-2003A patent/SK5072003A3/sk not_active Application Discontinuation
- 2001-10-23 AU AU1056302A patent/AU1056302A/xx active Pending
- 2001-10-23 KR KR10-2003-7005620A patent/KR20040011423A/ko not_active Application Discontinuation
- 2001-10-23 NZ NZ525281A patent/NZ525281A/en unknown
- 2001-10-23 HU HU0302308A patent/HUP0302308A2/hu unknown
- 2001-10-23 US US10/380,624 patent/US6869949B2/en not_active Expired - Fee Related
-
2003
- 2003-03-13 ZA ZA200302038A patent/ZA200302038B/en unknown
- 2003-04-24 NO NO20031830A patent/NO325736B1/no unknown
- 2003-04-24 HR HR20030323A patent/HRP20030323A2/hr not_active Application Discontinuation
-
2004
- 2004-05-24 US US10/851,092 patent/US7141567B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP1332143A1 (en) | 2003-08-06 |
| US7141567B2 (en) | 2006-11-28 |
| PL360412A1 (en) | 2004-09-06 |
| NZ525281A (en) | 2004-11-26 |
| US20040214852A1 (en) | 2004-10-28 |
| US20040106642A1 (en) | 2004-06-03 |
| BR0114873A (pt) | 2003-07-01 |
| MXPA03003706A (es) | 2005-01-25 |
| ZA200302038B (en) | 2004-04-22 |
| US6869949B2 (en) | 2005-03-22 |
| EA008151B1 (ru) | 2007-04-27 |
| NO20031830D0 (no) | 2003-04-24 |
| EA200300478A1 (ru) | 2003-12-25 |
| JP2004512338A (ja) | 2004-04-22 |
| NO325736B1 (no) | 2008-07-14 |
| CN1692113A (zh) | 2005-11-02 |
| AU2002210563B2 (en) | 2007-03-01 |
| HUP0302308A2 (hu) | 2003-11-28 |
| NO20031830L (no) | 2003-04-24 |
| AU1056302A (en) | 2002-05-06 |
| HRP20030323A2 (hr) | 2005-04-30 |
| IL154850A0 (en) | 2003-10-31 |
| CA2426616A1 (en) | 2002-05-02 |
| WO2002034749A1 (en) | 2002-05-02 |
| KR20040011423A (ko) | 2004-02-05 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AU2002210563B2 (en) | Polysubstituted imidazopyridines as gastric secretion inhibitors | |
| AU2002210563A1 (en) | Polysubstituted imidazopyridines as gastric secretion inhibitors | |
| SK13872002A3 (sk) | Alkylové imidazopyridínové deriváty, farmaceutický prostriedok s ich obsahom a ich použitie | |
| KR20070009614A (ko) | 7ｈ-8,9-디히드로-피라노(2,3-ｃ)이미다조(1,2-ａ)피리딘유도체 및 이의 위산 분비 억제제로서의 용도 | |
| CA2582294A1 (en) | Condensed tricyclic benzimidazoles for the treatment of gastrointestinal disorders | |
| US20060035892A1 (en) | Nitrosated imidazopyridines | |
| US20040235883A1 (en) | Alkyl-substituted imidazopyridines for the treatment of gastrointestinal disorders | |
| US20040235882A1 (en) | Amino-substituted imidazopyridines for the treatment of gastrointestial diseases | |
| EP1797089A1 (en) | Substituted tricyclic benzimidazoles | |
| US20070244173A1 (en) | 6,7-Dihydroxy-8-Phenyl-3,6,7,8-Tetrahydro-Chromeno [7,8-d] Imidazole Derivatives and Their Use as Gastric Acid Secretion Inhibitors | |
| EP1718648B1 (en) | Tricyclic imidazopyridines and intermediates for the synthesis thereof | |
| AU2002328995A1 (en) | Alkyl-substituted imidazopyridines for the treatment of gastrointestinal disorders |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC9A | Refused patent application |