SK480890A3 - (endo)-n-[[(8-methyl-8-azabicyclo[3.2.1]octan- -3-yl)amino]carbonyl]-2-(cyclopropylmethoxy)benzamide, process for its preparation and pharmaceutical compositions containing the same - Google Patents

(endo)-n-[[(8-methyl-8-azabicyclo[3.2.1]octan- -3-yl)amino]carbonyl]-2-(cyclopropylmethoxy)benzamide, process for its preparation and pharmaceutical compositions containing the same Download PDF

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Publication number
SK480890A3
SK480890A3 SK4808-90A SK480890A SK480890A3 SK 480890 A3 SK480890 A3 SK 480890A3 SK 480890 A SK480890 A SK 480890A SK 480890 A3 SK480890 A3 SK 480890A3
Authority
SK
Slovakia
Prior art keywords
endo
azabicyclo
methyl
octan
cyclopropylmethoxy
Prior art date
Application number
SK4808-90A
Other languages
English (en)
Slovak (sk)
Other versions
SK279469B6 (sk
Inventor
Terence J Ward
Janet C White
Gerald Bradley
Original Assignee
Wyeth John & Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth John & Brother Ltd filed Critical Wyeth John & Brother Ltd
Publication of SK279469B6 publication Critical patent/SK279469B6/sk
Publication of SK480890A3 publication Critical patent/SK480890A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Glass Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Removal Of Specific Substances (AREA)
SK4808-90A 1989-10-07 1990-10-03 (endo)-n-[[(8-methyl-8-azabicyclo[3.2.1]octan- -3-yl)amino]carbonyl]-2-(cyclopropylmethoxy)benzamide, process for its preparation and pharmaceutical compositions containing the same SK480890A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898922622A GB8922622D0 (en) 1989-10-07 1989-10-07 Aroylureas

Publications (2)

Publication Number Publication Date
SK279469B6 SK279469B6 (sk) 1998-11-04
SK480890A3 true SK480890A3 (en) 1998-11-04

Family

ID=10664224

Family Applications (1)

Application Number Title Priority Date Filing Date
SK4808-90A SK480890A3 (en) 1989-10-07 1990-10-03 (endo)-n-[[(8-methyl-8-azabicyclo[3.2.1]octan- -3-yl)amino]carbonyl]-2-(cyclopropylmethoxy)benzamide, process for its preparation and pharmaceutical compositions containing the same

Country Status (22)

Country Link
EP (1) EP0422846B1 (de)
JP (1) JP2960141B2 (de)
KR (1) KR100196263B1 (de)
CN (1) CN1042534C (de)
AT (1) ATE101607T1 (de)
AU (1) AU634584B2 (de)
CA (1) CA2027041C (de)
CZ (1) CZ280228B6 (de)
DE (1) DE69006675T2 (de)
DK (1) DK0422846T3 (de)
ES (1) ES2062398T3 (de)
FI (1) FI96419C (de)
GB (2) GB8922622D0 (de)
HU (1) HU204821B (de)
IE (1) IE64043B1 (de)
IL (1) IL95892A (de)
MX (1) MX22719A (de)
NZ (1) NZ235583A (de)
PT (1) PT95490B (de)
RU (2) RU1817778C (de)
SK (1) SK480890A3 (de)
ZA (1) ZA907993B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8922622D0 (en) * 1989-10-07 1989-11-22 Wyeth John & Brother Ltd Aroylureas
GB9106571D0 (en) * 1991-03-27 1991-05-15 Erba Carlo Spa Derivatives of substituted imidazol-2-one and process for their preparation
GB9217629D0 (en) * 1992-08-19 1992-09-30 Wyeth John & Brother Ltd Aroylureas
GB2269747B (en) * 1992-08-19 1996-06-05 Wyeth John & Brother Ltd Aroyl-ureas as pharmaceuticals, particularly 5-ht3 antagonists
GB9314174D0 (en) * 1993-07-08 1993-08-18 American Home Prod 5-ht3-antagonists

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU611976B2 (en) * 1987-12-24 1991-06-27 John Wyeth & Brother Limited Aroyl urea and carbamic acid derivatives of azabicyclo compounds
DK443489D0 (da) * 1989-09-08 1989-09-08 Ferrosan As Substituerede urinstofforbindelser, deres fremstilling og anvendelse
GB8922622D0 (en) * 1989-10-07 1989-11-22 Wyeth John & Brother Ltd Aroylureas

Also Published As

Publication number Publication date
GB9021695D0 (en) 1990-11-21
FI96419B (fi) 1996-03-15
CA2027041A1 (en) 1991-04-08
PT95490A (pt) 1991-07-05
FI96419C (fi) 1996-06-25
NZ235583A (en) 1991-12-23
IL95892A (en) 1994-06-24
SK279469B6 (sk) 1998-11-04
GB2236528A (en) 1991-04-10
PT95490B (pt) 1997-11-28
ZA907993B (en) 1992-06-24
CA2027041C (en) 2000-08-08
DK0422846T3 (da) 1994-03-14
FI904912A0 (fi) 1990-10-05
CZ480890A3 (en) 1995-07-12
IE903583A1 (en) 1991-04-10
AU634584B2 (en) 1993-02-25
EP0422846B1 (de) 1994-02-16
CN1050875A (zh) 1991-04-24
DE69006675D1 (de) 1994-03-24
KR100196263B1 (ko) 1999-06-15
RU1817778C (ru) 1993-05-23
CZ280228B6 (cs) 1995-12-13
IE64043B1 (en) 1995-06-28
MX22719A (es) 1993-09-01
IL95892A0 (en) 1991-07-18
AU6374990A (en) 1991-04-11
GB8922622D0 (en) 1989-11-22
ATE101607T1 (de) 1994-03-15
RU2036923C1 (ru) 1995-06-09
EP0422846A2 (de) 1991-04-17
DE69006675T2 (de) 1994-05-26
JPH03133986A (ja) 1991-06-07
ES2062398T3 (es) 1994-12-16
GB2236528B (en) 1993-06-30
HU906355D0 (en) 1991-04-29
CN1042534C (zh) 1999-03-17
HU204821B (en) 1992-02-28
KR910007871A (ko) 1991-05-30
JP2960141B2 (ja) 1999-10-06
EP0422846A3 (en) 1991-12-04
HUT55391A (en) 1991-05-28

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