SK282848B6 - Premostené cyklické aminokyseliny, farmaceutická kompozícia obsahujúca tieto aminokyseliny - Google Patents

Premostené cyklické aminokyseliny, farmaceutická kompozícia obsahujúca tieto aminokyseliny Download PDF

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Publication number
SK282848B6
SK282848B6 SK1248-98A SK124898A SK282848B6 SK 282848 B6 SK282848 B6 SK 282848B6 SK 124898 A SK124898 A SK 124898A SK 282848 B6 SK282848 B6 SK 282848B6
Authority
SK
Slovakia
Prior art keywords
cyclic amino
bridged cyclic
amino acid
acid according
formula
Prior art date
Application number
SK1248-98A
Other languages
English (en)
Slovak (sk)
Other versions
SK124898A3 (en
Inventor
Justin Stephen Bryans
David Christopher Horwell
Clare Octavia Kneen
Andrew Ian Morrell
Giles Stuart Ratcliffe
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of SK124898A3 publication Critical patent/SK124898A3/sk
Publication of SK282848B6 publication Critical patent/SK282848B6/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/28—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and containing rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A61P25/12—Antiepileptics; Anticonvulsants for grand-mal
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/36—Systems containing two condensed rings the rings having more than two atoms in common
    • C07C2602/42—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing seven carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/36—Systems containing two condensed rings the rings having more than two atoms in common
    • C07C2602/46—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing nine carbon atoms
SK1248-98A 1996-03-14 1997-02-18 Premostené cyklické aminokyseliny, farmaceutická kompozícia obsahujúca tieto aminokyseliny SK282848B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1343396P 1996-03-14 1996-03-14
PCT/US1997/002401 WO1997033859A1 (en) 1996-03-14 1997-02-18 Novel bridged cyclic amino acids as pharmaceutical agents

Publications (2)

Publication Number Publication Date
SK124898A3 SK124898A3 (en) 1999-02-11
SK282848B6 true SK282848B6 (sk) 2002-12-03

Family

ID=21759944

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1248-98A SK282848B6 (sk) 1996-03-14 1997-02-18 Premostené cyklické aminokyseliny, farmaceutická kompozícia obsahujúca tieto aminokyseliny

Country Status (18)

Country Link
US (1) US6020370A (ko)
EP (1) EP0888285B1 (ko)
JP (1) JP2000506862A (ko)
KR (1) KR100487032B1 (ko)
AT (1) ATE210629T1 (ko)
AU (1) AU731279B2 (ko)
BR (1) BR9708180A (ko)
CZ (1) CZ287598A3 (ko)
DE (1) DE69709070T2 (ko)
EA (1) EA001214B1 (ko)
ES (1) ES2169848T3 (ko)
IL (1) IL125364A0 (ko)
NO (1) NO984204L (ko)
NZ (1) NZ331142A (ko)
PL (1) PL185990B1 (ko)
SK (1) SK282848B6 (ko)
WO (1) WO1997033859A1 (ko)
ZA (1) ZA972199B (ko)

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US6310098B1 (en) 1999-07-22 2001-10-30 University Of Rochester Method of treating symptoms of hormonal variation, including hot flashes
WO2001072311A1 (en) * 2000-03-28 2001-10-04 Delorenzo Robert J Inhibition of a novel calcium injury current that forms in neurons during injury prevents neuronal cell death
WO2002000209A2 (en) * 2000-06-26 2002-01-03 Warner-Lambert Company Gabapentin analogues for sleep disorders
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GB2374595A (en) * 2001-04-19 2002-10-23 Warner Lambert Co Fused bicyclic or tricyclic amino acids
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US7186855B2 (en) * 2001-06-11 2007-03-06 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
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US20040162351A1 (en) * 2002-12-11 2004-08-19 Gallop Mark A. Orally administered dosage forms of fused GABA analog prodrugs having reduced toxicity
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ES2341240T3 (es) 2002-12-13 2010-06-17 Warner-Lambert Company Llc Ligando alfa-2-delta para tratar los sintomas del tracto urinario inferior.
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JP2006522146A (ja) * 2003-03-31 2006-09-28 ゼノポート，インコーポレイティド Ｇａｂａ類似体のプロドラッグを使用するのぼせの治療または予防
NZ545884A (en) 2003-09-11 2010-01-29 Xenoport Inc Treating and/or preventing urinary incontinence using prodrugs of GABA analogs
KR100828218B1 (ko) 2003-09-12 2008-05-07 화이자 인코포레이티드 알파-2-델타 리간드 및 세로토닌/노르아드레날린 재흡수 억제제를 포함하는 조합물
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Also Published As

Publication number Publication date
NO984204D0 (no) 1998-09-11
PL185990B1 (pl) 2003-09-30
EP0888285B1 (en) 2001-12-12
NZ331142A (en) 2001-04-27
ATE210629T1 (de) 2001-12-15
JP2000506862A (ja) 2000-06-06
EA001214B1 (ru) 2000-12-25
US6020370A (en) 2000-02-01
PL328800A1 (en) 1999-02-15
EP0888285A1 (en) 1999-01-07
ZA972199B (en) 1997-09-17
EA199800797A1 (ru) 1999-04-29
ES2169848T3 (es) 2002-07-16
AU731279B2 (en) 2001-03-29
IL125364A0 (en) 1999-03-12
CZ287598A3 (cs) 1999-02-17
AU2127197A (en) 1997-10-01
SK124898A3 (en) 1999-02-11
BR9708180A (pt) 1999-07-27
DE69709070T2 (de) 2002-06-20
KR100487032B1 (ko) 2005-12-21
DE69709070D1 (de) 2002-01-24
NO984204L (no) 1998-09-11
WO1997033859A1 (en) 1997-09-18
KR19990087755A (ko) 1999-12-27

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