EA200970487A1 - Применение пролекарств аналогов гамк для лечения заболеваний - Google Patents

Применение пролекарств аналогов гамк для лечения заболеваний

Info

Publication number
EA200970487A1
EA200970487A1 EA200970487A EA200970487A EA200970487A1 EA 200970487 A1 EA200970487 A1 EA 200970487A1 EA 200970487 A EA200970487 A EA 200970487A EA 200970487 A EA200970487 A EA 200970487A EA 200970487 A1 EA200970487 A1 EA 200970487A1
Authority
EA
Eurasian Patent Office
Prior art keywords
treatment
diseases
application
disease
gaba analogue
Prior art date
Application number
EA200970487A
Other languages
English (en)
Inventor
Рональд В. Барретт
Кеннет К. Канди
Original Assignee
Ксенопорт, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ксенопорт, Инк. filed Critical Ксенопорт, Инк.
Publication of EA200970487A1 publication Critical patent/EA200970487A1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid, pantothenic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/04—Drugs for disorders of the respiratory system for throat disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/14—Antitussive agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Описаны способы применения пролекарств аналогов ГАМК и их фармацевтических композиций для лечения мигрени, фибромиалгии, бокового амиотрофического склероза, синдрома раздраженного кишечника, социальной фобии, болезни Паркинсона, астмы, кашля или хронического обструктивного легочного заболевания и фармацевтические композиции пролекарств аналогов ГАМК, применяемых при лечении мигрени, фибромиалгии, бокового амиотрофического склероза, синдрома раздраженного кишечника, социальной фобии, болезни Паркинсона, астмы, кашля или хронического обструктивного легочного заболевания.
EA200970487A 2006-12-08 2007-12-06 Применение пролекарств аналогов гамк для лечения заболеваний EA200970487A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US87356106P 2006-12-08 2006-12-08
PCT/US2007/024944 WO2008073257A1 (en) 2006-12-08 2007-12-06 Use of prodrugs of gaba analogs for treating diseases

Publications (1)

Publication Number Publication Date
EA200970487A1 true EA200970487A1 (ru) 2009-12-30

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
EA200970487A EA200970487A1 (ru) 2006-12-08 2007-12-06 Применение пролекарств аналогов гамк для лечения заболеваний

Country Status (13)

Country Link
US (2) US20080161393A1 (ru)
EP (1) EP2101752A1 (ru)
JP (1) JP2010512314A (ru)
CN (1) CN101652133A (ru)
AR (1) AR064212A1 (ru)
AU (1) AU2007332904A1 (ru)
BR (1) BRPI0720252A2 (ru)
CA (1) CA2672044A1 (ru)
EA (1) EA200970487A1 (ru)
MX (1) MX2009006080A (ru)
PE (1) PE20081389A1 (ru)
TW (1) TW200845959A (ru)
WO (1) WO2008073257A1 (ru)

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PE20081389A1 (es) 2008-11-19
US20120041061A1 (en) 2012-02-16
MX2009006080A (es) 2009-07-14
CA2672044A1 (en) 2008-06-19
JP2010512314A (ja) 2010-04-22
EP2101752A1 (en) 2009-09-23
CN101652133A (zh) 2010-02-17
BRPI0720252A2 (pt) 2014-01-07
US20080161393A1 (en) 2008-07-03
TW200845959A (en) 2008-12-01
AU2007332904A1 (en) 2008-06-19
AR064212A1 (es) 2009-03-18
WO2008073257A1 (en) 2008-06-19

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