SK281511B6 - Estery bi- a tricyklických aminoalkoholov, farmaceutický prostriedok s ich obsahom a ich použitie - Google Patents

Estery bi- a tricyklických aminoalkoholov, farmaceutický prostriedok s ich obsahom a ich použitie Download PDF

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Publication number
SK281511B6
SK281511B6 SK949-93A SK94993A SK281511B6 SK 281511 B6 SK281511 B6 SK 281511B6 SK 94993 A SK94993 A SK 94993A SK 281511 B6 SK281511 B6 SK 281511B6
Authority
SK
Slovakia
Prior art keywords
tropanyl
methobromide
thienyl
methyl
formula
Prior art date
Application number
SK949-93A
Other languages
English (en)
Slovak (sk)
Other versions
SK94993A3 (en
Inventor
Rolf Banholzer
Rudolf Bauer
Richard Reichl
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of SK94993A3 publication Critical patent/SK94993A3/sk
Publication of SK281511B6 publication Critical patent/SK281511B6/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
SK949-93A 1991-03-15 1992-03-05 Estery bi- a tricyklických aminoalkoholov, farmaceutický prostriedok s ich obsahom a ich použitie SK281511B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4108393A DE4108393A1 (de) 1991-03-15 1991-03-15 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln
PCT/EP1992/000489 WO1992016528A1 (de) 1991-03-15 1992-03-05 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln

Publications (2)

Publication Number Publication Date
SK94993A3 SK94993A3 (en) 1994-04-06
SK281511B6 true SK281511B6 (sk) 2001-04-09

Family

ID=6427349

Family Applications (1)

Application Number Title Priority Date Filing Date
SK949-93A SK281511B6 (sk) 1991-03-15 1992-03-05 Estery bi- a tricyklických aminoalkoholov, farmaceutický prostriedok s ich obsahom a ich použitie

Country Status (26)

Country Link
US (1) US5654314A (es)
EP (1) EP0579615B1 (es)
JP (1) JP3352684B2 (es)
KR (1) KR100307274B1 (es)
AT (1) ATE202778T1 (es)
AU (1) AU662128B2 (es)
CA (1) CA2105575C (es)
CZ (1) CZ281509B6 (es)
DE (2) DE4108393A1 (es)
DK (1) DK0579615T3 (es)
ES (1) ES2160577T3 (es)
FI (1) FI120235B (es)
GR (1) GR3036792T3 (es)
HU (1) HU224210B1 (es)
IE (1) IE920815A1 (es)
IL (1) IL101225A (es)
MX (1) MX9201139A (es)
NO (1) NO304266B1 (es)
NZ (1) NZ241961A (es)
PL (1) PL179673B1 (es)
PT (1) PT100234B (es)
SG (1) SG43037A1 (es)
SK (1) SK281511B6 (es)
UA (1) UA29406C2 (es)
WO (1) WO1992016528A1 (es)
ZA (1) ZA921875B (es)

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US7309707B2 (en) * 2002-03-20 2007-12-18 Boehringer Ingelheim Pharma Gmbh & Co. Kg Crystalline micronisate, process for the manufacture thereof and use thereof for the preparation of a medicament
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Also Published As

Publication number Publication date
JP3352684B2 (ja) 2002-12-03
AU1345792A (en) 1992-10-21
EP0579615B1 (de) 2001-07-04
SK94993A3 (en) 1994-04-06
IL101225A0 (en) 1992-11-15
HU224210B1 (hu) 2005-06-28
CA2105575C (en) 2000-04-25
US5654314A (en) 1997-08-05
MX9201139A (es) 1992-10-01
HU9302611D0 (en) 1993-12-28
PL179673B1 (pl) 2000-10-31
NO304266B1 (no) 1998-11-23
JPH06505718A (ja) 1994-06-30
FI120235B (fi) 2009-08-14
KR100307274B1 (ko) 2001-12-05
FI934000A (fi) 1993-09-13
UA29406C2 (uk) 2000-11-15
DK0579615T3 (da) 2001-09-17
PT100234B (pt) 1999-06-30
SG43037A1 (en) 1997-10-17
IE920815A1 (en) 1992-09-23
WO1992016528A1 (de) 1992-10-01
ES2160577T3 (es) 2001-11-16
CA2105575A1 (en) 1992-09-16
NO933274L (no) 1993-11-12
CZ191793A3 (en) 1994-05-18
GR3036792T3 (en) 2002-01-31
DE59209907D1 (de) 2001-08-09
DE4108393A1 (de) 1992-09-17
ZA921875B (en) 1993-09-13
EP0579615A1 (de) 1994-01-26
NZ241961A (en) 1995-07-26
NO933274D0 (no) 1993-09-14
FI934000A0 (fi) 1993-09-13
AU662128B2 (en) 1995-08-24
ATE202778T1 (de) 2001-07-15
HUT65132A (en) 1994-04-28
PT100234A (pt) 1993-07-30
IL101225A (en) 1996-05-14
CZ281509B6 (cs) 1996-10-16

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