SI3252053T1 - Policiklične karbamoilpiridonske spojine in njihova uporaba za zdravljenje okužb s HIV - Google Patents

Policiklične karbamoilpiridonske spojine in njihova uporaba za zdravljenje okužb s HIV

Info

Publication number
SI3252053T1
SI3252053T1 SI201431750T SI201431750T SI3252053T1 SI 3252053 T1 SI3252053 T1 SI 3252053T1 SI 201431750 T SI201431750 T SI 201431750T SI 201431750 T SI201431750 T SI 201431750T SI 3252053 T1 SI3252053 T1 SI 3252053T1
Authority
SI
Slovenia
Prior art keywords
polycyclic
treatment
hiv infections
carbamoylpyridone compounds
carbamoylpyridone
Prior art date
Application number
SI201431750T
Other languages
English (en)
Slovenian (sl)
Inventor
Mingzhe Ji
Teresa Alejandra Trejo Martin
Manoj C. Desai
Haolun Jin
Hyung-Jung Pyun
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of SI3252053T1 publication Critical patent/SI3252053T1/sl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
SI201431750T 2013-07-12 2014-07-11 Policiklične karbamoilpiridonske spojine in njihova uporaba za zdravljenje okužb s HIV SI3252053T1 (sl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361845807P 2013-07-12 2013-07-12
EP17177428.4A EP3252053B1 (en) 2013-07-12 2014-07-11 Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections

Publications (1)

Publication Number Publication Date
SI3252053T1 true SI3252053T1 (sl) 2021-03-31

Family

ID=51257630

Family Applications (2)

Application Number Title Priority Date Filing Date
SI201430410T SI3019499T1 (sl) 2013-07-12 2014-07-11 Policiklične karbamoilpiridonske spojine in njihova uporaba za zdravljenje HIV infekcij
SI201431750T SI3252053T1 (sl) 2013-07-12 2014-07-11 Policiklične karbamoilpiridonske spojine in njihova uporaba za zdravljenje okužb s HIV

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SI201430410T SI3019499T1 (sl) 2013-07-12 2014-07-11 Policiklične karbamoilpiridonske spojine in njihova uporaba za zdravljenje HIV infekcij

Country Status (18)

Country Link
US (6) US9458159B2 (OSRAM)
EP (2) EP3019499B1 (OSRAM)
JP (1) JP6411492B2 (OSRAM)
AU (3) AU2014286995B2 (OSRAM)
CA (1) CA2918055C (OSRAM)
CY (1) CY1119545T1 (OSRAM)
DK (1) DK3019499T3 (OSRAM)
ES (2) ES2856867T3 (OSRAM)
HR (1) HRP20171807T1 (OSRAM)
HU (1) HUE037343T2 (OSRAM)
LT (1) LT3019499T (OSRAM)
NO (1) NO2865735T3 (OSRAM)
PL (1) PL3019499T3 (OSRAM)
PT (1) PT3019499T (OSRAM)
RS (1) RS56539B1 (OSRAM)
SI (2) SI3019499T1 (OSRAM)
SM (1) SMT201700525T1 (OSRAM)
WO (1) WO2015006733A1 (OSRAM)

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TW202222798A (zh) * 2020-09-30 2022-06-16 美商基利科學股份有限公司 橋接三環胺甲醯基吡啶酮化合物及其用途
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