SI21137A - Derivati azafenilalanina - Google Patents
Derivati azafenilalanina Download PDFInfo
- Publication number
- SI21137A SI21137A SI200200013A SI200200013A SI21137A SI 21137 A SI21137 A SI 21137A SI 200200013 A SI200200013 A SI 200200013A SI 200200013 A SI200200013 A SI 200200013A SI 21137 A SI21137 A SI 21137A
- Authority
- SI
- Slovenia
- Prior art keywords
- formula
- compound
- same meaning
- alkyl
- triphosgene
- Prior art date
Links
- DHTRYTBHUGJCJV-UHFFFAOYSA-N NC(c1ccc(CN(C(N2CCCCCC2)=O)NC(COc2cc3ccccc3cc2)=O)cc1)=N Chemical compound NC(c1ccc(CN(C(N2CCCCCC2)=O)NC(COc2cc3ccccc3cc2)=O)cc1)=N DHTRYTBHUGJCJV-UHFFFAOYSA-N 0.000 description 1
- DACCTOWVRVPJMC-UHFFFAOYSA-N O=C(N(Cc1ccc(CNCl)cc1)NS(C1=CC=C2C=CC=CC2C1)(=O)=O)N1CCCCC1 Chemical compound O=C(N(Cc1ccc(CNCl)cc1)NS(C1=CC=C2C=CC=CC2C1)(=O)=O)N1CCCCC1 DACCTOWVRVPJMC-UHFFFAOYSA-N 0.000 description 1
- ALPLIAPYWWEZCG-UHFFFAOYSA-N O=CC(N(Cc1ccc(CNCl)cc1)NS(c1cc2ccccc2cc1)(=O)=O)N1CCCCCC1 Chemical compound O=CC(N(Cc1ccc(CNCl)cc1)NS(c1cc2ccccc2cc1)(=O)=O)N1CCCCCC1 ALPLIAPYWWEZCG-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/48—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups having nitrogen atoms of sulfonamide groups further bound to another hetero atom
- C07C311/49—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups having nitrogen atoms of sulfonamide groups further bound to another hetero atom to nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
- C07D207/48—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D277/06—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/18—Systems containing only non-condensed rings with a ring being at least seven-membered
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hematology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SI200200013A SI21137A (sl) | 2002-01-24 | 2002-01-24 | Derivati azafenilalanina |
| CH01209/04A CH696724A5 (de) | 2002-01-24 | 2003-01-27 | Azaphenylalaninderivate. |
| AT0900103A AT503355A2 (de) | 2002-01-24 | 2003-01-27 | Azaphenylalanine derivatives |
| PCT/IB2003/000403 WO2004067522A1 (en) | 2002-01-24 | 2003-01-27 | Azaphenylalanine derivatives and their use as antithrombotic agents |
| DE10392134T DE10392134T5 (de) | 2002-01-24 | 2003-01-27 | Azaphenylalaninderivate |
| AU2003205963A AU2003205963A1 (en) | 2002-01-24 | 2003-01-27 | Azaphenylalanine derivatives and their use as antithrombotic agents |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SI200200013A SI21137A (sl) | 2002-01-24 | 2002-01-24 | Derivati azafenilalanina |
| PCT/IB2003/000403 WO2004067522A1 (en) | 2002-01-24 | 2003-01-27 | Azaphenylalanine derivatives and their use as antithrombotic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI21137A true SI21137A (sl) | 2003-08-31 |
Family
ID=39522234
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI200200013A SI21137A (sl) | 2002-01-24 | 2002-01-24 | Derivati azafenilalanina |
Country Status (6)
| Country | Link |
|---|---|
| AT (1) | AT503355A2 (de) |
| AU (1) | AU2003205963A1 (de) |
| CH (1) | CH696724A5 (de) |
| DE (1) | DE10392134T5 (de) |
| SI (1) | SI21137A (de) |
| WO (1) | WO2004067522A1 (de) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE502005007959D1 (de) | 2004-10-14 | 2009-10-01 | Wilex Ag | Verfahren zur reinigung von 3-hydroxy-amidino-phenylalanin-derivaten durch ausfällung und umkristallisation eines salzes mit einer aromatischen sulfonsäure |
| DE102004057195A1 (de) | 2004-11-26 | 2006-06-01 | Wilex Ag | Kristalline Modifikationen von N-Alpha-(2,4,6-Triisopropylphenylsulfonyl)-3-hydroxyamidino-(L)-phenylalanin-4-ethoxycarbonylpiperazid und/oder Salzen davon |
| GB0523539D0 (en) * | 2005-11-18 | 2005-12-28 | Lek Tovarna Farmacevtskih | New use of organic compounds |
| MY146638A (en) | 2007-04-10 | 2012-09-14 | Bayer Cropscience Ag | Insecticidal aryl isoxazoline derivatives |
| CN114040920A (zh) * | 2019-06-28 | 2022-02-11 | 富士胶片株式会社 | 肽化合物的制造方法、保护基形成用试剂及稠合多环芳香族烃化合物 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH05503300A (ja) * | 1990-11-15 | 1993-06-03 | ペンタファルム アクチェンゲゼルシャフト | メタ置換フェニルアラニン誘導体 |
| DE4111394A1 (de) * | 1991-04-09 | 1992-10-15 | Behringwerke Ag | Amidinophenylalaninderivate, verfahren zu deren herstellung, deren verwendung und diese enthaltende mittel |
| GB9322976D0 (en) * | 1993-11-08 | 1994-01-05 | Pfizer Ltd | Therapeutic agents |
| JP4414652B2 (ja) * | 2001-03-21 | 2010-02-10 | ヴィレックス アクチェンゲゼルシャフト | ウロキナーゼ阻害剤 |
-
2002
- 2002-01-24 SI SI200200013A patent/SI21137A/sl not_active IP Right Cessation
-
2003
- 2003-01-27 WO PCT/IB2003/000403 patent/WO2004067522A1/en not_active Application Discontinuation
- 2003-01-27 AU AU2003205963A patent/AU2003205963A1/en not_active Abandoned
- 2003-01-27 AT AT0900103A patent/AT503355A2/de not_active Application Discontinuation
- 2003-01-27 DE DE10392134T patent/DE10392134T5/de not_active Withdrawn
- 2003-01-27 CH CH01209/04A patent/CH696724A5/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE10392134T5 (de) | 2005-10-13 |
| AU2003205963A8 (en) | 2004-08-23 |
| AT503355A2 (de) | 2007-09-15 |
| CH696724A5 (de) | 2007-10-31 |
| WO2004067522A1 (en) | 2004-08-12 |
| AU2003205963A1 (en) | 2004-08-23 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US6638980B1 (en) | Inhibitors of factor Xa | |
| US6545055B1 (en) | Inhibitors of factor Xa | |
| DE69829879T2 (de) | Indolderivate als faktor xa inhibitoren | |
| US20040067938A1 (en) | Quaternary amines and related inhibitors of factor xa | |
| US20020065303A1 (en) | Bivalent phenylene inhibitors of factor Xa | |
| US7312235B2 (en) | Benzamide inhibitors of factor Xa | |
| US20020058677A1 (en) | Isoquinolone inhibitors of factor Xa | |
| US7417144B2 (en) | Factor Xa inhibitors | |
| US20020013314A1 (en) | 3,4-dihydro-2H-benzo[1,4]oxazine inhibitors of factor Xa | |
| CZ245994A3 (en) | Piperazides of substituted phenylalanine derivatives as thrombin inhibitors | |
| EP1185512A2 (de) | Faktor xa inhibitoren | |
| US20020052368A1 (en) | Oxindole inhibitors of factor Xa | |
| EP0190356B1 (de) | Amidinverbindungen | |
| US6924296B2 (en) | Antithrombotic agents | |
| US9708265B2 (en) | Urethanes, ureas, amidines and related inhibitors of factor Xa | |
| SI21137A (sl) | Derivati azafenilalanina | |
| AU2004279412A1 (en) | Thioether-substituted benzamides as inhibitors of Factor Xa | |
| US20080051388A1 (en) | Novel Compounds That Inhibit Factor Xa Activity | |
| US20020019394A1 (en) | Bicyclic sulfonyl amino inhibitors of factor Xa | |
| US20040077690A1 (en) | Quaternary amidino based inhibitors of factor xa | |
| SI21097A (sl) | Inhibitorji trombina | |
| US7285547B2 (en) | Amidinophenylalanine derivatives as thrombin inhibitors | |
| EP0486702A1 (de) | Derivate des phenyl-4-guanidinobenzoats, verfahren zu seiner herstellung und dieses enthaltender protease-inhibitor | |
| JP2004516317A5 (de) | ||
| SI20025A (sl) | Novi trombinski inhibitorji, njihova priprava in uporaba |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| IF | Valid on the prs date | ||
| KO00 | Lapse of patent |
Effective date: 20100901 |