SI1476141T1 - Naprave za transdermalno dajanje opoida, zaščitene pred nedovoljenimi posegi - Google Patents
Naprave za transdermalno dajanje opoida, zaščitene pred nedovoljenimi posegiInfo
- Publication number
- SI1476141T1 SI1476141T1 SI200331243T SI200331243T SI1476141T1 SI 1476141 T1 SI1476141 T1 SI 1476141T1 SI 200331243 T SI200331243 T SI 200331243T SI 200331243 T SI200331243 T SI 200331243T SI 1476141 T1 SI1476141 T1 SI 1476141T1
- Authority
- SI
- Slovenia
- Prior art keywords
- tamper
- patient
- pharmaceutically acceptable
- acceptable salt
- opioid
- Prior art date
Links
- 150000003839 salts Chemical class 0.000 abstract 3
- 230000037317 transdermal delivery Effects 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 1
- 239000003887 narcotic antagonist Substances 0.000 abstract 1
- 239000003401 opiate antagonist Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Emergency Medicine (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35713902P | 2002-02-19 | 2002-02-19 | |
| US35714102P | 2002-02-19 | 2002-02-19 | |
| PCT/US2003/004999 WO2003070191A2 (en) | 2002-02-19 | 2003-02-19 | Tamper-resistant transdermal opioid delivery devices |
| EP03742830A EP1476141B1 (en) | 2002-02-19 | 2003-02-19 | Tamper-resistant transdermal opioid delivery devices |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI1476141T1 true SI1476141T1 (sl) | 2008-08-31 |
Family
ID=27760456
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI200331243T SI1476141T1 (sl) | 2002-02-19 | 2003-02-19 | Naprave za transdermalno dajanje opoida, zaščitene pred nedovoljenimi posegi |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20040033253A1 (cg-RX-API-DMAC7.html) |
| EP (1) | EP1476141B1 (cg-RX-API-DMAC7.html) |
| JP (3) | JP4874523B2 (cg-RX-API-DMAC7.html) |
| AT (1) | ATE392892T1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU2003216321A1 (cg-RX-API-DMAC7.html) |
| CY (1) | CY1108201T1 (cg-RX-API-DMAC7.html) |
| DE (1) | DE60320530T2 (cg-RX-API-DMAC7.html) |
| DK (1) | DK1476141T3 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2305480T3 (cg-RX-API-DMAC7.html) |
| PT (1) | PT1476141E (cg-RX-API-DMAC7.html) |
| SI (1) | SI1476141T1 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2003070191A2 (cg-RX-API-DMAC7.html) |
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| KR101159828B1 (ko) * | 2003-04-30 | 2012-07-04 | 퍼듀 퍼머 엘피 | 활성제 구성요소 및 활성제 층의 원위부에 억제제 구성요소를 포함하는 내변조성 경피제형 |
| DE102005005446A1 (de) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Bruchfeste Darreichungsformen mit retardierter Freisetzung |
| US20070048228A1 (en) | 2003-08-06 | 2007-03-01 | Elisabeth Arkenau-Maric | Abuse-proofed dosage form |
| DE10361596A1 (de) | 2003-12-24 | 2005-09-29 | Grünenthal GmbH | Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform |
| DE10336400A1 (de) | 2003-08-06 | 2005-03-24 | Grünenthal GmbH | Gegen Missbrauch gesicherte Darreichungsform |
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| US8252321B2 (en) | 2004-09-13 | 2012-08-28 | Chrono Therapeutics, Inc. | Biosynchronous transdermal drug delivery for longevity, anti-aging, fatigue management, obesity, weight loss, weight management, delivery of nutraceuticals, and the treatment of hyperglycemia, alzheimer's disease, sleep disorders, parkinson's disease, aids, epilepsy, attention deficit disorder, nicotine addiction, cancer, headache and pain control, asthma, angina, hypertension, depression, cold, flu and the like |
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-
2003
- 2003-02-14 US US10/366,394 patent/US20040033253A1/en not_active Abandoned
- 2003-02-19 AU AU2003216321A patent/AU2003216321A1/en not_active Abandoned
- 2003-02-19 PT PT03742830T patent/PT1476141E/pt unknown
- 2003-02-19 WO PCT/US2003/004999 patent/WO2003070191A2/en not_active Ceased
- 2003-02-19 ES ES03742830T patent/ES2305480T3/es not_active Expired - Lifetime
- 2003-02-19 EP EP03742830A patent/EP1476141B1/en not_active Expired - Lifetime
- 2003-02-19 DE DE60320530T patent/DE60320530T2/de not_active Expired - Lifetime
- 2003-02-19 AT AT03742830T patent/ATE392892T1/de active
- 2003-02-19 DK DK03742830T patent/DK1476141T3/da active
- 2003-02-19 SI SI200331243T patent/SI1476141T1/sl unknown
- 2003-02-19 JP JP2003569151A patent/JP4874523B2/ja not_active Expired - Fee Related
-
2008
- 2008-07-17 CY CY20081100746T patent/CY1108201T1/el unknown
-
2010
- 2010-03-29 JP JP2010075835A patent/JP5453151B2/ja not_active Expired - Fee Related
-
2013
- 2013-08-02 JP JP2013160887A patent/JP2013237692A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JP2006502967A (ja) | 2006-01-26 |
| JP4874523B2 (ja) | 2012-02-15 |
| EP1476141A2 (en) | 2004-11-17 |
| JP5453151B2 (ja) | 2014-03-26 |
| EP1476141B1 (en) | 2008-04-23 |
| ES2305480T3 (es) | 2008-11-01 |
| WO2003070191A2 (en) | 2003-08-28 |
| US20040033253A1 (en) | 2004-02-19 |
| AU2003216321A8 (en) | 2003-09-09 |
| DE60320530T2 (de) | 2009-06-10 |
| WO2003070191A3 (en) | 2004-09-10 |
| AU2003216321A1 (en) | 2003-09-09 |
| DK1476141T3 (da) | 2008-08-18 |
| DE60320530D1 (de) | 2008-06-05 |
| ATE392892T1 (de) | 2008-05-15 |
| JP2010189403A (ja) | 2010-09-02 |
| CY1108201T1 (el) | 2014-02-12 |
| JP2013237692A (ja) | 2013-11-28 |
| PT1476141E (pt) | 2008-07-03 |
| WO2003070191A8 (en) | 2004-06-10 |
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