SG145748A1 - 6-substituted anilino purines as rtk inhibitors - Google Patents
6-substituted anilino purines as rtk inhibitorsInfo
- Publication number
- SG145748A1 SG145748A1 SG200806062-6A SG2008060626A SG145748A1 SG 145748 A1 SG145748 A1 SG 145748A1 SG 2008060626 A SG2008060626 A SG 2008060626A SG 145748 A1 SG145748 A1 SG 145748A1
- Authority
- SG
- Singapore
- Prior art keywords
- purines
- substituted anilino
- rtk inhibitors
- rtk
- inhibitors
- Prior art date
Links
- -1 6-substituted anilino purines Chemical class 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/16—Emollients or protectives, e.g. against radiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Toxicology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US49540603P | 2003-08-15 | 2003-08-15 | |
US52435703P | 2003-11-21 | 2003-11-21 | |
US56536704P | 2004-04-26 | 2004-04-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
SG145748A1 true SG145748A1 (en) | 2008-09-29 |
Family
ID=34198974
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG200806062-6A SG145748A1 (en) | 2003-08-15 | 2004-08-13 | 6-substituted anilino purines as rtk inhibitors |
Country Status (16)
Country | Link |
---|---|
US (2) | US20050124637A1 (de) |
EP (1) | EP1656378A4 (de) |
JP (1) | JP2007502776A (de) |
AU (2) | AU2004264419B2 (de) |
BR (1) | BRPI0413563A (de) |
CA (1) | CA2535620A1 (de) |
CO (1) | CO5680404A2 (de) |
EC (1) | ECSP066365A (de) |
IL (1) | IL173392A0 (de) |
IS (1) | IS8345A (de) |
MA (1) | MA27997A1 (de) |
MX (1) | MXPA06001758A (de) |
NO (1) | NO20061074L (de) |
SG (1) | SG145748A1 (de) |
TN (1) | TNSN06053A1 (de) |
WO (1) | WO2005016528A2 (de) |
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AU2006261527B2 (en) * | 2005-05-16 | 2012-11-22 | Prometic Pharma Smt Limited | Purine derivatives and their use for treatment of autoimmune diseases |
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DE69613211T2 (de) * | 1995-11-14 | 2001-11-15 | Pharmacia & Upjohn Spa | Aryl- und heteroaryl- purin- und pyridopyrimidin- derivate |
GB9613021D0 (en) * | 1996-06-21 | 1996-08-28 | Pharmacia Spa | Bicyclic 4-aralkylaminopyrimidine derivatives as tyrosine kinase inhibitors |
US5866702A (en) * | 1996-08-02 | 1999-02-02 | Cv Therapeutics, Incorporation | Purine inhibitors of cyclin dependent kinase 2 |
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GB9918035D0 (en) * | 1999-07-30 | 1999-09-29 | Novartis Ag | Organic compounds |
EP1206559A2 (de) * | 1999-08-26 | 2002-05-22 | Plant Research International B.V. | Bedingte hemmung der vegetativen vermehrung |
US6506762B1 (en) * | 1999-09-30 | 2003-01-14 | Neurogen Corporation | Certain alkylene diamine-substituted heterocycles |
BR0207302A (pt) * | 2001-02-08 | 2004-02-10 | Memory Pharm Corp | Trifluorometilpurinas como inibidores da fosfodiesterase 4 |
CZ294535B6 (cs) * | 2001-08-02 | 2005-01-12 | Ústav Experimentální Botaniky Avčr | Heterocyklické sloučeniny na bázi N6-substituovaného adeninu, způsoby jejich přípravy, jejich použití pro přípravu léčiv, kosmetických přípravků a růstových regulátorů, farmaceutické přípravky, kosmetické přípravky a růstové regulátory tyto sloučeniny obsahující |
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EP1444982A1 (de) * | 2003-02-06 | 2004-08-11 | Merckle Gmbh | Verwendung von Purinderivaten als selektive Kinase-Inhibitoren |
BRPI0807182A2 (pt) * | 2007-01-26 | 2014-05-27 | Irm Llc | Compostos e composições como inibidores de cinase |
-
2004
- 2004-08-13 MX MXPA06001758A patent/MXPA06001758A/es not_active Application Discontinuation
- 2004-08-13 EP EP04781114A patent/EP1656378A4/de not_active Withdrawn
- 2004-08-13 JP JP2006523409A patent/JP2007502776A/ja active Pending
- 2004-08-13 WO PCT/US2004/026373 patent/WO2005016528A2/en active Application Filing
- 2004-08-13 SG SG200806062-6A patent/SG145748A1/en unknown
- 2004-08-13 CA CA002535620A patent/CA2535620A1/en not_active Abandoned
- 2004-08-13 US US10/917,578 patent/US20050124637A1/en not_active Abandoned
- 2004-08-13 BR BRPI0413563-6A patent/BRPI0413563A/pt not_active IP Right Cessation
- 2004-08-13 AU AU2004264419A patent/AU2004264419B2/en not_active Ceased
-
2006
- 2006-01-26 IL IL173392A patent/IL173392A0/en unknown
- 2006-02-14 EC EC2006006365A patent/ECSP066365A/es unknown
- 2006-02-14 TN TNP2006000053A patent/TNSN06053A1/en unknown
- 2006-02-17 MA MA28818A patent/MA27997A1/fr unknown
- 2006-02-20 CO CO06016491A patent/CO5680404A2/es not_active Application Discontinuation
- 2006-03-06 NO NO20061074A patent/NO20061074L/no not_active Application Discontinuation
- 2006-03-09 IS IS8345A patent/IS8345A/is unknown
-
2009
- 2009-04-15 AU AU2009201480A patent/AU2009201480A1/en not_active Abandoned
-
2010
- 2010-12-22 US US12/976,187 patent/US20110092491A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
NO20061074L (no) | 2006-03-06 |
CO5680404A2 (es) | 2006-09-29 |
IS8345A (is) | 2006-03-09 |
EP1656378A4 (de) | 2011-05-11 |
WO2005016528A3 (en) | 2005-05-12 |
AU2004264419A1 (en) | 2005-02-24 |
WO2005016528A2 (en) | 2005-02-24 |
AU2009201480A1 (en) | 2009-05-14 |
IL173392A0 (en) | 2006-06-11 |
JP2007502776A (ja) | 2007-02-15 |
US20110092491A1 (en) | 2011-04-21 |
AU2004264419B2 (en) | 2009-01-15 |
CA2535620A1 (en) | 2005-02-24 |
US20050124637A1 (en) | 2005-06-09 |
BRPI0413563A (pt) | 2006-10-17 |
EP1656378A2 (de) | 2006-05-17 |
MA27997A1 (fr) | 2006-07-03 |
ECSP066365A (es) | 2006-08-30 |
TNSN06053A1 (en) | 2007-10-03 |
MXPA06001758A (es) | 2006-08-11 |
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