SG11201700703XA - Salt of monocyclic pyridine derivative and crystal thereof - Google Patents
Salt of monocyclic pyridine derivative and crystal thereofInfo
- Publication number
- SG11201700703XA SG11201700703XA SG11201700703XA SG11201700703XA SG11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA
- Authority
- SG
- Singapore
- Prior art keywords
- salt
- crystal
- pyridine derivative
- monocyclic pyridine
- monocyclic
- Prior art date
Links
- 239000013078 crystal Substances 0.000 title 1
- -1 monocyclic pyridine derivative Chemical class 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
- C07C55/10—Succinic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014166118 | 2014-08-18 | ||
| PCT/JP2015/073047 WO2016027781A1 (ja) | 2014-08-18 | 2015-08-17 | 単環ピリジン誘導体の塩およびその結晶 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG11201700703XA true SG11201700703XA (en) | 2017-03-30 |
Family
ID=55350725
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG11201700703XA SG11201700703XA (en) | 2014-08-18 | 2015-08-17 | Salt of monocyclic pyridine derivative and crystal thereof |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US9951047B2 (de) |
| EP (1) | EP3184520B1 (de) |
| JP (1) | JP5925978B1 (de) |
| KR (1) | KR102344105B1 (de) |
| CN (1) | CN106660997B (de) |
| AU (1) | AU2015304465B2 (de) |
| BR (1) | BR112017002268B1 (de) |
| CA (1) | CA2956270C (de) |
| ES (1) | ES2914072T3 (de) |
| IL (1) | IL250290B (de) |
| MX (1) | MX369646B (de) |
| RU (1) | RU2658821C1 (de) |
| SG (1) | SG11201700703XA (de) |
| WO (1) | WO2016027781A1 (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2016374441B2 (en) * | 2015-12-17 | 2021-10-21 | Eisai R&D Management Co., Ltd. | Therapeutic agent for breast cancer |
| MX2020002083A (es) * | 2017-10-12 | 2020-03-24 | Eisai R&D Man Co Ltd | Composicion farmaceutica que comprende un inhibidor tirosina cinasa selectivo para receptores del factor de crecimiento de fibroblastos (fgfr). |
| MX2020008610A (es) | 2018-03-28 | 2020-09-21 | Eisai R&D Man Co Ltd | Agente terapeutico para carcinoma hepatocelular. |
| BR112022020786A2 (pt) | 2020-04-17 | 2022-11-29 | Eisai R&D Man Co Ltd | Agente terapêutico de câncer de mama |
| AU2021315234A1 (en) | 2020-07-31 | 2023-01-19 | Eisai R&D Management Co., Ltd. | Therapeutic agent for breast cancer |
| CN116390757A (zh) | 2020-10-28 | 2023-07-04 | 卫材R&D管理有限公司 | 用于治疗肿瘤的药物组合物 |
| CA3227445A1 (en) * | 2021-08-31 | 2023-03-09 | Eisai R&D Management Co., Ltd. | Production method for synthetic intermediate of monocyclic pyridine derivative |
| MX2024001504A (es) | 2021-08-31 | 2024-02-27 | Eisai R&D Man Co Ltd | Metodo para producir un derivado de piridina monociclico. |
| AU2023236231A1 (en) * | 2022-03-18 | 2024-09-05 | Shanghai Institute Of Materia Medica , Chinese Academy Of Sciences | Salt of substituted amino six-membered nitric heterocyclic compound, crystal form thereof, method for preparing same, and use thereof |
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| US20050256154A1 (en) | 2004-05-04 | 2005-11-17 | Kin-Chun Luk | 4-Amino-thieno[3,2-c]pyridine-7-carboxylic acid amides |
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| FR2883286B1 (fr) | 2005-03-16 | 2008-10-03 | Sanofi Aventis Sa | NOUVEAUX DERIVES D'IMIDAZO[1,5-a]PYRIDINES, INHIBITEURS DE FGFs, LEUR PROCEDE DE PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES LES CONTENANT |
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| CL2008003675A1 (es) | 2007-12-13 | 2009-03-20 | Wyeth Corp | Compuestos derivados de 5-alquil o alquenil 3-cianopiridinas, procedimiento de preparacion, composicion farmaceutica, util para reducir la actividad incrementada de una enzima en un mamifero, en donde dicha enzima es una proteina quinasa, destinado al tratamiento de la inflamacion, asma, colitis, esclerosis multiple, soriasis, artritis reumatoide. |
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| BR112012008094A2 (pt) | 2009-08-07 | 2020-08-18 | Chugai Seiyaku Kabushiki Kaisha | derivado de aminopirazol, seu uso, composição farmacêutica que o compreende, agentes para inibir a atividade de fgfr e para prevenir ou tratar câncer |
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| AR094812A1 (es) * | 2013-02-20 | 2015-08-26 | Eisai R&D Man Co Ltd | Derivado de piridina monocíclico como inhibidor del fgfr |
| TWI628176B (zh) | 2013-04-04 | 2018-07-01 | 奧利安公司 | 蛋白質激酶抑制劑 |
-
2015
- 2015-08-17 JP JP2015560425A patent/JP5925978B1/ja active Active
- 2015-08-17 KR KR1020177002791A patent/KR102344105B1/ko active IP Right Grant
- 2015-08-17 US US15/500,429 patent/US9951047B2/en active Active
- 2015-08-17 CN CN201580042132.3A patent/CN106660997B/zh active Active
- 2015-08-17 WO PCT/JP2015/073047 patent/WO2016027781A1/ja active Application Filing
- 2015-08-17 MX MX2017001624A patent/MX369646B/es active IP Right Grant
- 2015-08-17 EP EP15834302.0A patent/EP3184520B1/de active Active
- 2015-08-17 BR BR112017002268-0A patent/BR112017002268B1/pt active IP Right Grant
- 2015-08-17 CA CA2956270A patent/CA2956270C/en active Active
- 2015-08-17 ES ES15834302T patent/ES2914072T3/es active Active
- 2015-08-17 AU AU2015304465A patent/AU2015304465B2/en active Active
- 2015-08-17 SG SG11201700703XA patent/SG11201700703XA/en unknown
- 2015-08-17 RU RU2017103439A patent/RU2658821C1/ru active
-
2017
- 2017-01-25 IL IL250290A patent/IL250290B/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| MX369646B (es) | 2019-11-15 |
| CN106660997A (zh) | 2017-05-10 |
| EP3184520A4 (de) | 2018-04-18 |
| WO2016027781A1 (ja) | 2016-02-25 |
| AU2015304465A1 (en) | 2017-02-23 |
| BR112017002268A2 (pt) | 2017-11-21 |
| US20170217935A1 (en) | 2017-08-03 |
| IL250290A0 (en) | 2017-03-30 |
| ES2914072T3 (es) | 2022-06-07 |
| CA2956270A1 (en) | 2016-02-25 |
| JP5925978B1 (ja) | 2016-05-25 |
| JPWO2016027781A1 (ja) | 2017-04-27 |
| KR102344105B1 (ko) | 2021-12-29 |
| MX2017001624A (es) | 2017-04-27 |
| BR112017002268B1 (pt) | 2022-11-08 |
| KR20170035927A (ko) | 2017-03-31 |
| CA2956270C (en) | 2022-08-09 |
| CN106660997B (zh) | 2019-05-21 |
| EP3184520B1 (de) | 2022-03-23 |
| US9951047B2 (en) | 2018-04-24 |
| IL250290B (en) | 2020-06-30 |
| EP3184520A1 (de) | 2017-06-28 |
| RU2658821C1 (ru) | 2018-06-25 |
| AU2015304465B2 (en) | 2019-05-09 |
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