SG11201507033RA - Tripeptide epoxy ketone protease inhibitors - Google Patents

Tripeptide epoxy ketone protease inhibitors

Info

Publication number
SG11201507033RA
SG11201507033RA SG11201507033RA SG11201507033RA SG11201507033RA SG 11201507033R A SG11201507033R A SG 11201507033RA SG 11201507033R A SG11201507033R A SG 11201507033RA SG 11201507033R A SG11201507033R A SG 11201507033RA SG 11201507033R A SG11201507033R A SG 11201507033RA
Authority
SG
Singapore
Prior art keywords
protease inhibitors
epoxy ketone
ketone protease
tripeptide epoxy
tripeptide
Prior art date
Application number
SG11201507033RA
Other languages
English (en)
Inventor
Dustin Mcminn
Henry Johnson
Simeon Bowers
David C Moebius
Original Assignee
Onyx Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51581125&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201507033R(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Onyx Therapeutics Inc filed Critical Onyx Therapeutics Inc
Publication of SG11201507033RA publication Critical patent/SG11201507033RA/en

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0821Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06Tripeptides
    • AHUMAN NECESSITIES
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • C07D303/12Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
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SG11201507033RA 2013-03-14 2014-03-14 Tripeptide epoxy ketone protease inhibitors SG11201507033RA (en)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US201361786086P 2013-03-14 2013-03-14
US201361785608P 2013-03-14 2013-03-14
US201361847780P 2013-07-18 2013-07-18
US201361856847P 2013-07-22 2013-07-22
US201361883843P 2013-09-27 2013-09-27
US201361883798P 2013-09-27 2013-09-27
US201461941798P 2014-02-19 2014-02-19
ARP140100970A AR095426A1 (es) 2013-03-14 2014-03-13 Inhibidores tripeptídicos de la epoxicetona proteasa
PCT/US2014/026987 WO2014152134A1 (en) 2013-03-14 2014-03-14 Tripeptide epoxy ketone protease inhibitors

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SG11201507033RA true SG11201507033RA (en) 2015-10-29

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SG11201507033RA SG11201507033RA (en) 2013-03-14 2014-03-14 Tripeptide epoxy ketone protease inhibitors

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