SG11201506100XA - Pyridazinone-amides derivatives - Google Patents

Pyridazinone-amides derivatives

Info

Publication number
SG11201506100XA
SG11201506100XA SG11201506100XA SG11201506100XA SG11201506100XA SG 11201506100X A SG11201506100X A SG 11201506100XA SG 11201506100X A SG11201506100X A SG 11201506100XA SG 11201506100X A SG11201506100X A SG 11201506100XA SG 11201506100X A SG11201506100X A SG 11201506100XA
Authority
SG
Singapore
Prior art keywords
pyridazinone
amides derivatives
amides
derivatives
Prior art date
Application number
SG11201506100XA
Other languages
English (en)
Inventor
Catherine Jorand-Lebrun
Santosh Kulkarni
Stefano Crosignani
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SG11201506100XA publication Critical patent/SG11201506100XA/en

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    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • Neurology (AREA)
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  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
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  • Gynecology & Obstetrics (AREA)
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SG11201506100XA 2013-02-07 2014-02-06 Pyridazinone-amides derivatives SG11201506100XA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP13154390 2013-02-07
PCT/EP2014/000316 WO2014121931A1 (en) 2013-02-07 2014-02-06 Pyridazinone-amides derivatives

Publications (1)

Publication Number Publication Date
SG11201506100XA true SG11201506100XA (en) 2015-09-29

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201506100XA SG11201506100XA (en) 2013-02-07 2014-02-06 Pyridazinone-amides derivatives

Country Status (23)

Country Link
US (2) US9567320B2 (ko)
EP (1) EP2953944B1 (ko)
JP (1) JP6483624B2 (ko)
KR (1) KR102293952B1 (ko)
CN (1) CN104968658B (ko)
AU (1) AU2014214321B2 (ko)
BR (1) BR112015018663A2 (ko)
CA (1) CA2900431C (ko)
DK (1) DK2953944T3 (ko)
ES (1) ES2634627T3 (ko)
HK (1) HK1215708A1 (ko)
HR (1) HRP20171076T1 (ko)
HU (1) HUE032863T2 (ko)
IL (1) IL240290B (ko)
LT (1) LT2953944T (ko)
MX (1) MX364486B (ko)
PL (1) PL2953944T3 (ko)
PT (1) PT2953944T (ko)
RS (1) RS56331B1 (ko)
RU (1) RU2666899C2 (ko)
SG (1) SG11201506100XA (ko)
SI (1) SI2953944T1 (ko)
WO (1) WO2014121931A1 (ko)

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JP6920202B2 (ja) * 2015-02-06 2021-08-18 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングＭｅｒｃｋ Ｐａｔｅｎｔ Ｇｅｓｅｌｌｓｃｈａｆｔ ｍｉｔ ｂｅｓｃｈｒａｅｎｋｔｅｒ Ｈａｆｔｕｎｇ Ｉｒａｋ阻害剤としてのピリダジノン大環状化合物及びその使用
KR102677905B1 (ko) 2015-04-22 2024-06-24 리겔 파마슈티칼스, 인크. 피라졸 화합물 및 이러한 화합물을 제조하고 사용하는 방법
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US11512080B2 (en) 2018-01-12 2022-11-29 Kymera Therapeutics, Inc. CRBN ligands and uses thereof
US11485743B2 (en) 2018-01-12 2022-11-01 Kymera Therapeutics, Inc. Protein degraders and uses thereof
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