SG11201401743RA - Modulators of the g protein-coupled mas receptor and the treatment of disorders related thereto - Google Patents

Modulators of the g protein-coupled mas receptor and the treatment of disorders related thereto

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Publication number
SG11201401743RA
SG11201401743RA SG11201401743RA SG11201401743RA SG11201401743RA SG 11201401743R A SG11201401743R A SG 11201401743RA SG 11201401743R A SG11201401743R A SG 11201401743RA SG 11201401743R A SG11201401743R A SG 11201401743RA SG 11201401743R A SG11201401743R A SG 11201401743RA
Authority
SG
Singapore
Prior art keywords
modulators
protein
treatment
disorders related
mas receptor
Prior art date
Application number
SG11201401743RA
Other languages
English (en)
Inventor
Thuy-Anh Tran
Anthony C Blackburn
Bryan A Kramer
Maiko Nagura
Carleton R Sage
Young-Jun Shin
Ning Zou
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of SG11201401743RA publication Critical patent/SG11201401743RA/en

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    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
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WO2015161011A1 (en) * 2014-04-17 2015-10-22 Merck Sharp & Dohme Corp. Benzamide cgrp receptor antagonists
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