SG10201602311XA - Orally disintegrating tablet - Google Patents

Orally disintegrating tablet

Info

Publication number
SG10201602311XA
SG10201602311XA SG10201602311XA SG10201602311XA SG10201602311XA SG 10201602311X A SG10201602311X A SG 10201602311XA SG 10201602311X A SG10201602311X A SG 10201602311XA SG 10201602311X A SG10201602311X A SG 10201602311XA SG 10201602311X A SG10201602311X A SG 10201602311XA
Authority
SG
Singapore
Prior art keywords
orally disintegrating
disintegrating tablet
tablet
orally
disintegrating
Prior art date
Application number
SG10201602311XA
Other languages
English (en)
Inventor
Shiro Ishii
Yutaka Ebisawa
Takayuki Okabe
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45509604&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10201602311X(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of SG10201602311XA publication Critical patent/SG10201602311XA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5015—Organic compounds, e.g. fats, sugars
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SG10201602311XA 2010-12-27 2011-12-26 Orally disintegrating tablet SG10201602311XA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201061427384P 2010-12-27 2010-12-27

Publications (1)

Publication Number Publication Date
SG10201602311XA true SG10201602311XA (en) 2016-04-28

Family

ID=45509604

Family Applications (2)

Application Number Title Priority Date Filing Date
SG2013040944A SG190905A1 (en) 2010-12-27 2011-12-26 Orally disintegrating tablet
SG10201602311XA SG10201602311XA (en) 2010-12-27 2011-12-26 Orally disintegrating tablet

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SG2013040944A SG190905A1 (en) 2010-12-27 2011-12-26 Orally disintegrating tablet

Country Status (23)

Country Link
US (1) US20130273157A1 (fr)
EP (1) EP2658530A2 (fr)
JP (1) JP2014501224A (fr)
KR (1) KR20140007364A (fr)
CN (1) CN103402500A (fr)
AR (1) AR084610A1 (fr)
AU (1) AU2011350396A1 (fr)
BR (1) BR112013014875A2 (fr)
CA (1) CA2823166C (fr)
CL (1) CL2013001793A1 (fr)
CO (1) CO6731132A2 (fr)
CR (1) CR20130327A (fr)
EA (1) EA028217B1 (fr)
EC (1) ECSP13012718A (fr)
MA (1) MA34768B1 (fr)
MX (1) MX2013007588A (fr)
PE (1) PE20141115A1 (fr)
SG (2) SG190905A1 (fr)
TN (1) TN2013000220A1 (fr)
TW (1) TW201304823A (fr)
UY (1) UY33841A (fr)
WO (1) WO2012091153A2 (fr)
ZA (1) ZA201304617B (fr)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104127368A (zh) 2008-03-11 2014-11-05 武田药品工业株式会社 口腔崩解固体制剂
SI2797416T1 (sl) 2011-12-28 2017-12-29 Global Blood Therapeutics, Inc. Substituirane spojine benzaldehida in metode njihove uporabe pri povečanju oksigenacije tkiva
US9012450B2 (en) 2011-12-28 2015-04-21 Global Blood Therapeutics, Inc. Substituted heteroaryl aldehyde compounds and methods for their use in increasing tissue oxygenation
GB201303781D0 (en) 2013-03-04 2013-04-17 Gauthier Pierre Pascal Oral timer device and method of using same
AP2015008721A0 (en) 2013-03-15 2015-09-30 Global Blood Therapeutics Inc Compounds and uses thereof for the modulation of hemoglobin
US9458139B2 (en) 2013-03-15 2016-10-04 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
EP2968299B1 (fr) 2013-03-15 2021-01-20 Global Blood Therapeutics, Inc. Composés et leurs utilisations pour la modulation de l'hémoglobine
BR112015021982B1 (pt) 2013-03-15 2022-12-13 Global Blood Therapeutics, Inc Compostos e seus usos para a modulação de hemoglobina
US8952171B2 (en) 2013-03-15 2015-02-10 Global Blood Therapeutics, Inc. Compounds and uses thereof for the modulation of hemoglobin
EA202092627A1 (ru) 2013-11-18 2021-09-30 Глобал Блад Терапьютикс, Инк. Соединения и их применения для модуляции гемоглобина
CN114181195A (zh) 2014-02-07 2022-03-15 全球血液疗法股份有限公司 一种化合物的结晶多晶型物
RU2017118432A (ru) 2014-11-14 2018-12-14 Джемфир Терапьютикс Инк. СПОСОБЫ И ПРОМЕЖУТОЧНЫЕ СОЕДИНЕНИЯ ДЛЯ ПОЛУЧЕНИЯ ДИАЛКАНОВЫХ ЭФИРОВ, СОДЕРЖАЩИХ КОНЦЕВУЮ α,ω-ДИКАРБОНОВОКИСЛОТНУЮ ГРУППУ
US20170042806A1 (en) 2015-04-29 2017-02-16 Dexcel Pharma Technologies Ltd. Orally disintegrating compositions
SG11201804647TA (en) 2015-12-04 2018-06-28 Global Blood Therapeutics Inc Dosing regimens for 2-hydroxy-6-((2-(1-isopropyl-1h-pyrazol-5-yl)pyridin-3-yl)methoxy)benzaldehyde
TWI752307B (zh) 2016-05-12 2022-01-11 美商全球血液治療公司 新穎化合物及製造化合物之方法
US10076494B2 (en) 2016-06-16 2018-09-18 Dexcel Pharma Technologies Ltd. Stable orally disintegrating pharmaceutical compositions
TW202332423A (zh) * 2016-10-12 2023-08-16 美商全球血液治療公司 包含2-羥基-6-((2-(1-異丙基-1h-吡唑-5-基)吡啶-3-基)甲氧基)-苯甲醛之片劑
US20190008779A1 (en) * 2017-05-11 2019-01-10 Gemphire Therapeutics Inc. Gemcabene compositions and methods of use thereof
ES2921931T3 (es) 2017-07-10 2022-09-02 Takeda Pharmaceuticals Co Preparación que comprende vonoprazán
CN108576205B (zh) * 2018-03-22 2022-01-04 湖北省农业科学院农产品加工与核农技术研究所 一种草莓联合干燥的处理方法
US11014884B2 (en) 2018-10-01 2021-05-25 Global Blood Therapeutics, Inc. Modulators of hemoglobin

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6150978A (ja) 1984-08-16 1986-03-13 Takeda Chem Ind Ltd ピリジン誘導体およびその製造法
JPH072761B2 (ja) 1985-03-20 1995-01-18 不二パウダル株式会社 微結晶セルロ−ス球形顆粒及びその製造法
JPS62277322A (ja) 1986-02-13 1987-12-02 Takeda Chem Ind Ltd 安定化された腸溶性抗潰瘍固形組成物
FR2679451B1 (fr) 1991-07-22 1994-09-09 Prographarm Laboratoires Comprime multiparticulaire a delitement rapide.
ATE216577T1 (de) 1992-01-29 2002-05-15 Takeda Chemical Industries Ltd Schnellösliche tablette und ihre herstellung
JP2919771B2 (ja) 1995-04-17 1999-07-19 佐藤製薬株式会社 速溶解性錠剤の製造方法及び該製造方法により製造した速溶解性錠剤
JPH0948726A (ja) 1995-08-07 1997-02-18 Tanabe Seiyaku Co Ltd 口腔内速崩壊性製剤およびその製法
TW385306B (en) 1996-11-14 2000-03-21 Takeda Chemical Industries Ltd Method for producing crystals of benzimidazole derivatives
JP3828648B2 (ja) 1996-11-14 2006-10-04 武田薬品工業株式会社 ２−（２−ピリジルメチルスルフィニル）ベンズイミダゾール系化合物の結晶およびその製造法
ES2559766T3 (es) 1998-05-18 2016-02-15 Takeda Pharmaceutical Company Limited Comprimidos disgregables en la boca
DE69942777D1 (de) 1998-07-28 2010-10-28 Takeda Pharmaceutical Leicht zerfallende feste Zubereitung
TWI275587B (en) 1999-06-17 2007-03-11 Takeda Chemical Industries Ltd A crystal of (R)-2-[[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridyl]methyl]sulfinyl]-1H-benzimidazole
CN1193024C (zh) 2000-04-28 2005-03-16 武田药品工业株式会社 生产旋光的亚砜衍生物的方法
US7169799B2 (en) 2000-05-15 2007-01-30 Takeda Pharmaceutical Company Limited Process for producing crystal
EP1337525B8 (fr) 2000-12-01 2011-10-05 Takeda Pharmaceutical Company Limited Procede de cristallisation du (r)- ou du (s)-lansoprazole
JP4493970B2 (ja) 2002-10-16 2010-06-30 武田薬品工業株式会社 持続性製剤
US20050214372A1 (en) * 2004-03-03 2005-09-29 Simona Di Capua Stable pharmaceutical composition comprising an acid labile drug
CA2630235A1 (fr) * 2005-12-20 2007-07-12 Teva Pharmaceutical Industries Ltd. Comprimes a desintegration orale de lansoprazole
US20070141151A1 (en) * 2005-12-20 2007-06-21 Silver David I Lansoprazole orally disintegrating tablets
EP1837016A3 (fr) * 2006-03-08 2008-01-02 KRKA, tovarna zdravil, d.d., Novo mesto Composition pharmaceutique en multiple-unité
EP2098250B1 (fr) * 2006-12-28 2016-09-28 Takeda Pharmaceutical Company Limited Préparation solide se désintégrant oralement
CN104127368A (zh) * 2008-03-11 2014-11-05 武田药品工业株式会社 口腔崩解固体制剂
WO2010008569A1 (fr) * 2008-07-17 2010-01-21 Barr Laboratories, Inc. Formes posologiques pharmaceutiques solides à désintégration orale comprenant du lansoprazole à libération retardée et leurs méthodes de production et d'utilisation

Also Published As

Publication number Publication date
CO6731132A2 (es) 2013-08-15
SG190905A1 (en) 2013-07-31
EA201390981A1 (ru) 2014-07-30
TN2013000220A1 (en) 2014-11-10
AU2011350396A1 (en) 2013-07-11
UY33841A (es) 2012-07-31
US20130273157A1 (en) 2013-10-17
CL2013001793A1 (es) 2013-12-06
BR112013014875A2 (pt) 2016-10-18
CA2823166C (fr) 2019-04-09
JP2014501224A (ja) 2014-01-20
ZA201304617B (en) 2014-08-27
CN103402500A (zh) 2013-11-20
EA028217B1 (ru) 2017-10-31
MA34768B1 (fr) 2013-12-03
AR084610A1 (es) 2013-05-29
ECSP13012718A (es) 2013-12-31
CR20130327A (es) 2013-08-22
WO2012091153A3 (fr) 2012-09-07
EP2658530A2 (fr) 2013-11-06
KR20140007364A (ko) 2014-01-17
PE20141115A1 (es) 2014-09-12
MX2013007588A (es) 2013-08-09
WO2012091153A2 (fr) 2012-07-05
CA2823166A1 (fr) 2012-07-05
TW201304823A (zh) 2013-02-01

Similar Documents

Publication Publication Date Title
ZA201304617B (en) Orally disintegrating tablet
ZA201304366B (en) Orally disintegrating tablet
PL2415466T3 (pl) Tabletka powlekana ulegająca rozpadowi w jamie ustnej
EP2429586A4 (fr) Excipient se désintégrant par voie orale
EP2572995A4 (fr) Cassette de comprimés
PL2368704T3 (pl) Wylot tabletek
ZA201305567B (en) Orally dispersible tablet
EP2510950A4 (fr) Comprimé enrobé à sec à désintégration orale
GB2489658B (en) Tablet press
EP2382971A4 (fr) Comprimé à désintégration orale comportant un noyau intérieur
ZA201200761B (en) Tablet
EP2409688A4 (fr) Comprimé se délitant par voie orale
EP2810659A4 (fr) Comprimé à désintégration par voie orale contenant des granules masquant l'amertume
IL222368A0 (en) Orally disintegrating tablet containing acarbose
IL222754A0 (en) Enteric tablet
EP2612657A4 (fr) Comprimé à désintégration orale
AU330360S (en) Tablet
IL222753A0 (en) Enteric tablet
GB0920041D0 (en) Tablet
PL2428202T3 (pl) Kompozycje ulegające rozpadowi w jamie ustnej
PL2521819T3 (pl) Przestrzeń sanitarna
ZA201201059B (en) Tablet manufacture
AU335048S (en) Tablet
AU331949S (en) Tablet
AU330359S (en) Tablet