SE8307133L - Karboxamidoderivat av 5h-1,3,4-tiadiazolo/3,2-a/pyrimider och forfarande for deras framstellning - Google Patents

Karboxamidoderivat av 5h-1,3,4-tiadiazolo/3,2-a/pyrimider och forfarande for deras framstellning

Info

Publication number
SE8307133L
SE8307133L SE8307133A SE8307133A SE8307133L SE 8307133 L SE8307133 L SE 8307133L SE 8307133 A SE8307133 A SE 8307133A SE 8307133 A SE8307133 A SE 8307133A SE 8307133 L SE8307133 L SE 8307133L
Authority
SE
Sweden
Prior art keywords
alkyl
unsubstituted
substituted
ring
alkoxy
Prior art date
Application number
SE8307133A
Other languages
English (en)
Other versions
SE8307133D0 (sv
SE454698B (sv
Inventor
G Doria
C Passarotti
A Buttinoni
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838329746A external-priority patent/GB8329746D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of SE8307133D0 publication Critical patent/SE8307133D0/sv
Publication of SE8307133L publication Critical patent/SE8307133L/sv
Publication of SE454698B publication Critical patent/SE454698B/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/1251,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE8307133A 1982-12-23 1983-12-22 6-karboxamidoderivat av 5-oxo-5h-1,3,4-tiadiazolo/3,2-a/pyrimidiner, forfarande for deras framstellning samt farmaceutiska kompositioner innehallande desamma SE454698B (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8236642 1982-12-23
GB838329746A GB8329746D0 (en) 1983-11-08 1983-11-08 Carboxamido-derivatives

Publications (3)

Publication Number Publication Date
SE8307133D0 SE8307133D0 (sv) 1983-12-22
SE8307133L true SE8307133L (sv) 1984-06-24
SE454698B SE454698B (sv) 1988-05-24

Family

ID=26284768

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8307133A SE454698B (sv) 1982-12-23 1983-12-22 6-karboxamidoderivat av 5-oxo-5h-1,3,4-tiadiazolo/3,2-a/pyrimidiner, forfarande for deras framstellning samt farmaceutiska kompositioner innehallande desamma

Country Status (15)

Country Link
US (1) US4522944A (sv)
AT (1) AT385036B (sv)
AU (1) AU558600B2 (sv)
CA (1) CA1211440A (sv)
CH (1) CH657136A5 (sv)
DE (1) DE3346223A1 (sv)
DK (1) DK593983A (sv)
FI (1) FI834698A (sv)
FR (1) FR2538392B1 (sv)
GR (1) GR79479B (sv)
IL (1) IL70522A (sv)
IT (1) IT1194521B (sv)
NL (1) NL8304340A (sv)
SE (1) SE454698B (sv)
SU (1) SU1297731A3 (sv)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3702758A1 (de) * 1987-01-30 1988-09-29 Hoechst Ag Substituierte 3-phenyl-7h-thiazolo (3,2-b) (1,2,4) triazin-7-one, verfahren zu ihrer herstellung, die sie enthaltenden arzneimittel und ihre verwendung, sowie einige bei der herstellung der genannten verbindungen gebildete zwischenprodukte
JP5567349B2 (ja) 2007-03-12 2014-08-06 イントラ−セルラー・セラピーズ・インコーポレイテッド 置換ヘテロ環縮合ガンマ−カルボリンの合成
ES2727815T3 (es) 2012-04-14 2019-10-18 Intra Cellular Therapies Inc Tratamiento del TEPT y de trastornos del control de impulsos
PL2968320T3 (pl) 2013-03-15 2021-05-17 Intra-Cellular Therapies, Inc. Związki organiczne
KR102495941B1 (ko) 2013-12-03 2023-02-06 인트라-셀룰라 써래피스, 인코퍼레이티드. 신규한 방법
EP3125892A4 (en) 2014-04-04 2017-12-27 Intra-Cellular Therapies, Inc. Organic compounds
CA2944512C (en) 2014-04-04 2018-04-24 Intra-Cellular Therapies, Inc. Heterocycle fused gamma-carbolines for treatment of central nervous system disorders
HUE053737T2 (hu) 2016-01-26 2021-07-28 Intra Cellular Therapies Inc Piridopirrolokinoxalin vegyületek, készítményeik és alkalmazásaik
WO2017172795A1 (en) 2016-03-28 2017-10-05 Intra-Cellular Therapies, Inc. Novel compositions and methods
EP3436016B1 (en) 2016-03-28 2022-04-27 Intra-Cellular Therapies, Inc. Novel co-crystals
US10654854B2 (en) 2016-03-28 2020-05-19 Intra-Cellular Therapies, Inc. Salts and crystals of ITI-007
JP7013454B2 (ja) 2016-10-12 2022-02-15 イントラ-セルラー・セラピーズ・インコーポレイテッド アモルファス固体分散体
JP6987868B2 (ja) 2016-12-29 2022-01-05 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 有機化合物
WO2018126140A1 (en) 2016-12-29 2018-07-05 Intra-Cellular Therapies, Inc. Organic compounds
MX2019011329A (es) 2017-03-24 2019-12-02 Intra Celular Therapies Inc Composiciones novedosas y metodos.
KR102667268B1 (ko) 2017-07-26 2024-05-17 인트라-셀룰라 써래피스, 인코퍼레이티드. 유기 화합물
US11376249B2 (en) 2017-07-26 2022-07-05 Intra-Cellular Therapies, Inc. Organic compounds
AU2019287460B2 (en) 2018-06-11 2024-02-15 Intra-Cellular Therapies, Inc. Substituted heterocycle fused gamma-carbolines synthesis
EP3843739A4 (en) 2018-08-31 2022-06-01 Intra-Cellular Therapies, Inc. NEW METHODS
EP3843738A4 (en) 2018-08-31 2022-06-01 Intra-Cellular Therapies, Inc. NEW METHODS

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5129981B2 (sv) * 1973-07-17 1976-08-28
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
JPS55115889A (en) * 1979-02-28 1980-09-06 Teijin Ltd 6-carbamoylthiazolo 3,2-a pyrimidine derivative and its preparation
JPS57142989A (en) * 1981-02-27 1982-09-03 Dai Ichi Seiyaku Co Ltd Thiazolopyrimidine derivative

Also Published As

Publication number Publication date
SU1297731A3 (ru) 1987-03-15
FR2538392B1 (fr) 1987-01-16
NL8304340A (nl) 1984-07-16
SE8307133D0 (sv) 1983-12-22
DK593983A (da) 1984-06-24
FR2538392A1 (fr) 1984-06-29
FI834698A0 (fi) 1983-12-20
US4522944A (en) 1985-06-11
SE454698B (sv) 1988-05-24
FI834698A (fi) 1984-06-24
AT385036B (de) 1988-02-10
CA1211440A (en) 1986-09-16
IT8324207A0 (it) 1983-12-16
CH657136A5 (de) 1986-08-15
GR79479B (sv) 1984-10-30
IL70522A (en) 1986-02-28
AU2252583A (en) 1984-06-28
IL70522A0 (en) 1984-03-30
IT1194521B (it) 1988-09-22
ATA438383A (de) 1987-07-15
AU558600B2 (en) 1987-02-05
DK593983D0 (da) 1983-12-22
DE3346223A1 (de) 1984-06-28

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