FI834698A0 - Karboxiamidoderivat av 5h-1,3,4-tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa - Google Patents

Karboxiamidoderivat av 5h-1,3,4-tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa

Info

Publication number
FI834698A0
FI834698A0 FI834698A FI834698A FI834698A0 FI 834698 A0 FI834698 A0 FI 834698A0 FI 834698 A FI834698 A FI 834698A FI 834698 A FI834698 A FI 834698A FI 834698 A0 FI834698 A0 FI 834698A0
Authority
FI
Finland
Prior art keywords
carboxiamider
thiadiazolo
derivatives
carboxiamider derivatives
Prior art date
Application number
FI834698A
Other languages
English (en)
Other versions
FI834698A (fi
Inventor
Gianfederico Doria
Carlo Passarotti
Ada Buttinoni
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838329746A external-priority patent/GB8329746D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of FI834698A0 publication Critical patent/FI834698A0/fi
Publication of FI834698A publication Critical patent/FI834698A/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI834698A 1982-12-23 1983-12-20 Karboxiamidoderivat av 5h-1,3,4- tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa. FI834698A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8236642 1982-12-23
GB838329746A GB8329746D0 (en) 1983-11-08 1983-11-08 Carboxamido-derivatives

Publications (2)

Publication Number Publication Date
FI834698A0 true FI834698A0 (fi) 1983-12-20
FI834698A FI834698A (fi) 1984-06-24

Family

ID=26284768

Family Applications (1)

Application Number Title Priority Date Filing Date
FI834698A FI834698A (fi) 1982-12-23 1983-12-20 Karboxiamidoderivat av 5h-1,3,4- tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa.

Country Status (15)

Country Link
US (1) US4522944A (fi)
AT (1) AT385036B (fi)
AU (1) AU558600B2 (fi)
CA (1) CA1211440A (fi)
CH (1) CH657136A5 (fi)
DE (1) DE3346223A1 (fi)
DK (1) DK593983A (fi)
FI (1) FI834698A (fi)
FR (1) FR2538392B1 (fi)
GR (1) GR79479B (fi)
IL (1) IL70522A (fi)
IT (1) IT1194521B (fi)
NL (1) NL8304340A (fi)
SE (1) SE454698B (fi)
SU (1) SU1297731A3 (fi)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3702758A1 (de) * 1987-01-30 1988-09-29 Hoechst Ag Substituierte 3-phenyl-7h-thiazolo (3,2-b) (1,2,4) triazin-7-one, verfahren zu ihrer herstellung, die sie enthaltenden arzneimittel und ihre verwendung, sowie einige bei der herstellung der genannten verbindungen gebildete zwischenprodukte
CN101796051B (zh) * 2007-03-12 2013-11-06 细胞内治疗公司 与取代的杂环稠合的γ-咔啉的合成
CA2870303A1 (en) 2012-04-14 2013-10-17 Intra-Cellular Therapies, Inc. Organic compounds
HUE053159T2 (hu) 2013-03-15 2021-06-28 Intra Cellular Therapies Inc Szerves vegyületek
DK3076967T3 (da) 2013-12-03 2021-10-25 Intra Cellular Therapies Inc Fremgangsmåder til behandling af residuelle symptomer på skizofreni
EP3125893B1 (en) 2014-04-04 2023-09-20 Intra-Cellular Therapies, Inc. Deuterated heterocycle fused gamma-carbolines as antagonists of 5-ht2a receptors
JP2017509677A (ja) 2014-04-04 2017-04-06 イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−Ｃｅｌｌｕｌａｒ Ｔｈｅｒａｐｉｅｓ， Ｉｎｃ． 有機化合物
CA3011983A1 (en) 2016-01-26 2017-08-03 Intra-Cellular Therapies, Inc. Organic compounds
WO2017172784A1 (en) 2016-03-28 2017-10-05 Intra-Cellular Therapies, Inc. Novel salts and crystals
EP3436083A4 (en) 2016-03-28 2019-11-27 Intra-Cellular Therapies, Inc. NEW COMPOSITIONS AND METHODS
US11014925B2 (en) 2016-03-28 2021-05-25 Intra-Cellular Therapies, Inc. Co-crystals of 1-(4-fluoro-phenyl)-4-((6bR,1OaS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H- pyrido[3′,4′:4,51_pyrrolo [1,2,3-delqcuinoxalin-8-yl)-butan-1-one with nicotinamide or isonicotinamide
CN110072518B (zh) 2016-10-12 2021-10-26 细胞内治疗公司 无定形固体分散体
US10961245B2 (en) 2016-12-29 2021-03-30 Intra-Cellular Therapies, Inc. Substituted heterocycle fused gamma-carbolines for treatment of central nervous system disorders
EP3562484B1 (en) 2016-12-29 2021-08-25 Intra-Cellular Therapies, Inc. Pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxaline derivatives useful in the treatment of cns disorders
US10716786B2 (en) 2017-03-24 2020-07-21 Intra-Cellular Therapies, Inc. Transmucosal and subcutaneous compositions
US11376249B2 (en) 2017-07-26 2022-07-05 Intra-Cellular Therapies, Inc. Organic compounds
WO2019023063A1 (en) 2017-07-26 2019-01-31 Intra-Cellular Therapies, Inc. ORGANIC COMPOUNDS
JP7483671B2 (ja) 2018-06-11 2024-05-15 イントラ－セルラー・セラピーズ・インコーポレイテッド 置換ヘテロ環縮合ガンマ－カルボリン類合成
BR112021003838A2 (pt) 2018-08-31 2021-05-18 Intra-Cellular Therapies, Inc. métodos novos
JP2021536453A (ja) 2018-08-31 2021-12-27 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 新規方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5129981B2 (fi) * 1973-07-17 1976-08-28
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
JPS55115889A (en) * 1979-02-28 1980-09-06 Teijin Ltd 6-carbamoylthiazolo 3,2-a pyrimidine derivative and its preparation
JPS57142989A (en) * 1981-02-27 1982-09-03 Dai Ichi Seiyaku Co Ltd Thiazolopyrimidine derivative

Also Published As

Publication number Publication date
FR2538392A1 (fr) 1984-06-29
SE8307133D0 (sv) 1983-12-22
IL70522A (en) 1986-02-28
FR2538392B1 (fr) 1987-01-16
AU558600B2 (en) 1987-02-05
US4522944A (en) 1985-06-11
GR79479B (fi) 1984-10-30
NL8304340A (nl) 1984-07-16
SE454698B (sv) 1988-05-24
IL70522A0 (en) 1984-03-30
DK593983D0 (da) 1983-12-22
SU1297731A3 (ru) 1987-03-15
IT8324207A0 (it) 1983-12-16
CA1211440A (en) 1986-09-16
ATA438383A (de) 1987-07-15
CH657136A5 (de) 1986-08-15
IT1194521B (it) 1988-09-22
DE3346223A1 (de) 1984-06-28
FI834698A (fi) 1984-06-24
AT385036B (de) 1988-02-10
AU2252583A (en) 1984-06-28
SE8307133L (sv) 1984-06-24
DK593983A (da) 1984-06-24

Similar Documents

Publication Publication Date Title
FI822266L (fi) Nya imidazo/1,2-a/pyridiner och pyraziner
FI810147L (fi) Imidazo/1,2-a/pyridiner foerfande foer deras framstaellning och dessa innehaollande farmaceutiska kompositioner
FI834698A0 (fi) Karboxiamidoderivat av 5h-1,3,4-tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa
MX6983E (es) Procedimiento de preparacion de derivados 1,3-dihidro-6-metil-7-hidroxifuro-(3,4-c)-piridina
FI831350A0 (fi) Framstaellning av imidazo /1,2- /pyridinderivat och terapeutisk anvaendning
FI880429A0 (fi) Foerfarande foer utbredning av ett eldfast skikt med hjaelp av sprutning pao en yta och ett pao detta saett bildat skikt.
FI822446A0 (fi) Foerfarande och anordning foer gjutning av en lista med sidoriktade utspraong
FI782527A (fi) Pyrido(1,2-a)pyrimidin-derivat foerfarande foer deras framstaellning och desamma innehaollande farmaceutiska blandningar
DE3376324D1 (de) Imidazo(1,5-a)pyridine derivatives
AR229519A1 (es) Procedimiento de preparacion de derivados de 2,3-dihidro-9-fenil-1h-pirazolo(1,2-a)-indazolio
FI803355L (fi) 3,6,7,8-substituerade-s-triazolo/4,3-b/pyridaziner och dessa innehaollande foereningar
FI821035A0 (fi) Imidazo/1,2-a/pyrimidinderivat, deras framstaellning och anvaendning vid sjukvaord
FI864891A0 (fi) Foerfarande foer framstaellning av 6,7,8,9-tetrahydro-10-metylpyrido/1,2-a/indol-9-aminer och deras derivat.
FI833818A (fi) Foerfarande foer framstaellning av foerbaettrade formmassor av finfoerdelade expanderbara styrenpolymerisat med belaeggning, och anvaendning av belaeggningsprodukterna
IT8021821A0 (it) Pirido [1,2-a] pirimidine sostituite
DE3373473D1 (de) Pyrido(2,1-b)quinazoline derivatives
FI853027L (fi) Imidazo/1,2-a/kinoliner, deras framstaellning och deras terapeutiska tillaempning.
FI822329L (fi) Foerfarande foer framstaellning av substituerade pyrrolo/2,1-b/ kinazoliner och pyrido /2,1-b/ kinatsoliner
FI821992A0 (fi) Nya 1,4,9,10-tetrahydro-pyratsolo/4,3-e/-pyrido/3,2-b//1,4/diazepin-10-oner, foerfarande foer deras framstaellning och dessa foereningar innehaollande laekemedel
FI811970L (fi) 6-hydrazono-pyrido/2,1-b/kinazolin-11-oner och deras framstaellningsfoerfarande
FI832944A (fi) Rotationsstaol och haollorgan foer faststaellning av staolet i en haollare
AR227683A1 (es) Procedimiento para la preparacion de derivados de 6,7,8,9-tetrahidro-5h-pirazino(2,3-d)azepina,5,6,7,8-tetrahidro-pirido(3,4-b)pirazina y 6,7-dihidro-5h-pirrolo(3,4-b)pirazina
FI843282A (fi) Foerbaettringar i och beroerande pyrimido /4,5-g/kinoliner och mellanprodukter.
FI801513A (fi) 9-hydrazono-6,7,8,9-tetrahydro-4h-pyrido /1,2-a/ pyrimidin-4-on-derivat och foerfarande foer deras framstaellning
SE7910255L (sv) Pyrazolo (1,5-c)kinazolinderivat

Legal Events

Date Code Title Description
FD Application lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A