FI834698A0 - Karboxiamidoderivat av 5h-1,3,4-tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa - Google Patents

Karboxiamidoderivat av 5h-1,3,4-tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa

Info

Publication number
FI834698A0
FI834698A0 FI834698A FI834698A FI834698A0 FI 834698 A0 FI834698 A0 FI 834698A0 FI 834698 A FI834698 A FI 834698A FI 834698 A FI834698 A FI 834698A FI 834698 A0 FI834698 A0 FI 834698A0
Authority
FI
Finland
Prior art keywords
carboxiamider
thiadiazolo
derivatives
carboxiamider derivatives
Prior art date
Application number
FI834698A
Other languages
English (en)
Other versions
FI834698A (fi
Inventor
Gianfederico Doria
Carlo Passarotti
Ada Buttinoni
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838329746A external-priority patent/GB8329746D0/en
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of FI834698A0 publication Critical patent/FI834698A0/fi
Publication of FI834698A publication Critical patent/FI834698A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/1251,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI834698A 1982-12-23 1983-12-20 Karboxiamidoderivat av 5h-1,3,4- tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa. FI834698A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8236642 1982-12-23
GB838329746A GB8329746D0 (en) 1983-11-08 1983-11-08 Carboxamido-derivatives

Publications (2)

Publication Number Publication Date
FI834698A0 true FI834698A0 (fi) 1983-12-20
FI834698A FI834698A (fi) 1984-06-24

Family

ID=26284768

Family Applications (1)

Application Number Title Priority Date Filing Date
FI834698A FI834698A (fi) 1982-12-23 1983-12-20 Karboxiamidoderivat av 5h-1,3,4- tiadiazolo/3,2-a/ pyridiner och foerfarande foer framstaellning av dessa.

Country Status (15)

Country Link
US (1) US4522944A (fi)
AT (1) AT385036B (fi)
AU (1) AU558600B2 (fi)
CA (1) CA1211440A (fi)
CH (1) CH657136A5 (fi)
DE (1) DE3346223A1 (fi)
DK (1) DK593983A (fi)
FI (1) FI834698A (fi)
FR (1) FR2538392B1 (fi)
GR (1) GR79479B (fi)
IL (1) IL70522A (fi)
IT (1) IT1194521B (fi)
NL (1) NL8304340A (fi)
SE (1) SE454698B (fi)
SU (1) SU1297731A3 (fi)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3702758A1 (de) * 1987-01-30 1988-09-29 Hoechst Ag Substituierte 3-phenyl-7h-thiazolo (3,2-b) (1,2,4) triazin-7-one, verfahren zu ihrer herstellung, die sie enthaltenden arzneimittel und ihre verwendung, sowie einige bei der herstellung der genannten verbindungen gebildete zwischenprodukte
KR102065319B1 (ko) * 2007-03-12 2020-01-10 인트라-셀룰라 써래피스, 인코퍼레이티드. 치환된 헤테로환 융합 감마-카르볼린 합성
AU2013245702A1 (en) 2012-04-14 2014-11-13 Intra-Cellular Therapies, Inc. Organic compounds
WO2014145192A1 (en) 2013-03-15 2014-09-18 Intra-Cellular Therapies, Inc. Organic compounds
MX2021007665A (es) 2013-12-03 2022-09-09 Intra Cellular Therapies Inc Metodos novedosos.
EP3125892A4 (en) 2014-04-04 2017-12-27 Intra-Cellular Therapies, Inc. Organic compounds
JP2017509686A (ja) 2014-04-04 2017-04-06 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 有機化合物
JP6995761B2 (ja) 2016-01-26 2022-01-17 イントラ-セルラー・セラピーズ・インコーポレイテッド 有機化合物
JP2019513143A (ja) 2016-03-28 2019-05-23 イントラ−セルラー・セラピーズ・インコーポレイテッドIntra−Cellular Therapies, Inc. 新規塩類および結晶
EP3436016B1 (en) 2016-03-28 2022-04-27 Intra-Cellular Therapies, Inc. Novel co-crystals
WO2017172795A1 (en) 2016-03-28 2017-10-05 Intra-Cellular Therapies, Inc. Novel compositions and methods
JP7013454B2 (ja) 2016-10-12 2022-02-15 イントラ-セルラー・セラピーズ・インコーポレイテッド アモルファス固体分散体
WO2018126140A1 (en) 2016-12-29 2018-07-05 Intra-Cellular Therapies, Inc. Organic compounds
EP3562484B1 (en) 2016-12-29 2021-08-25 Intra-Cellular Therapies, Inc. Pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxaline derivatives useful in the treatment of cns disorders
EP3600325A4 (en) 2017-03-24 2021-01-06 Intra-Cellular Therapies, Inc. UNIQUE COMPOSITIONS AND PROCESSES
CA3071137A1 (en) 2017-07-26 2019-01-31 Intra-Cellular Therapies, Inc. Prodrugs of substituted heterocycle fused gamma-carbolines
WO2019023062A1 (en) 2017-07-26 2019-01-31 Intra-Cellular Therapies, Inc. ORGANIC COMPOUNDS
WO2019237037A1 (en) 2018-06-08 2019-12-12 Intra-Cellular Therapies, Inc. Novel methods
CA3106447A1 (en) 2018-06-11 2019-12-19 Intra-Cellular Therapies, Inc. Substituted heterocycle fused gamma-carbolines synthesis
AU2019328528A1 (en) 2018-08-31 2021-03-18 Intra-Cellular Therapies, Inc. Novel methods
KR20210052472A (ko) 2018-08-31 2021-05-10 인트라-셀룰라 써래피스, 인코퍼레이티드. 신규한 방법
WO2021007245A1 (en) 2019-07-07 2021-01-14 Intra-Cellular Therapies, Inc. Novel methods

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5129981B2 (fi) * 1973-07-17 1976-08-28
GB1568962A (en) * 1975-10-31 1980-06-11 Beecham Group Ltd Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p
JPS55115889A (en) * 1979-02-28 1980-09-06 Teijin Ltd 6-carbamoylthiazolo 3,2-a pyrimidine derivative and its preparation
JPS57142989A (en) * 1981-02-27 1982-09-03 Dai Ichi Seiyaku Co Ltd Thiazolopyrimidine derivative

Also Published As

Publication number Publication date
DK593983D0 (da) 1983-12-22
IL70522A0 (en) 1984-03-30
DK593983A (da) 1984-06-24
SU1297731A3 (ru) 1987-03-15
IL70522A (en) 1986-02-28
DE3346223A1 (de) 1984-06-28
IT8324207A0 (it) 1983-12-16
AU2252583A (en) 1984-06-28
AU558600B2 (en) 1987-02-05
CA1211440A (en) 1986-09-16
US4522944A (en) 1985-06-11
AT385036B (de) 1988-02-10
CH657136A5 (de) 1986-08-15
GR79479B (fi) 1984-10-30
FR2538392B1 (fr) 1987-01-16
FI834698A (fi) 1984-06-24
ATA438383A (de) 1987-07-15
IT1194521B (it) 1988-09-22
SE8307133L (sv) 1984-06-24
SE8307133D0 (sv) 1983-12-22
NL8304340A (nl) 1984-07-16
SE454698B (sv) 1988-05-24
FR2538392A1 (fr) 1984-06-29

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Legal Events

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FD Application lapsed

Owner name: FARMITALIA CARLO ERBA S.P.A