FI782527A - Pyrido(1,2-a)pyrimidin-derivat foerfarande foer deras framstaellning och desamma innehaollande farmaceutiska blandningar - Google Patents

Pyrido(1,2-a)pyrimidin-derivat foerfarande foer deras framstaellning och desamma innehaollande farmaceutiska blandningar

Info

Publication number
FI782527A
FI782527A FI782527A FI782527A FI782527A FI 782527 A FI782527 A FI 782527A FI 782527 A FI782527 A FI 782527A FI 782527 A FI782527 A FI 782527A FI 782527 A FI782527 A FI 782527A
Authority
FI
Finland
Prior art keywords
pyrido
pyrimidine derivatives
pyrimidine
derivatives
Prior art date
Application number
FI782527A
Other languages
English (en)
Other versions
FI66864B (fi
FI66864C (fi
Inventor
Jozsef Knoll
Zoltan Meszaros
Istvan Hermecz
Ferenc Fueloep
Gabor Bernath
Sandor Virag
Gabor Nagy
Peter Szentmiklosi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of FI782527A publication Critical patent/FI782527A/fi
Publication of FI66864B publication Critical patent/FI66864B/fi
Application granted granted Critical
Publication of FI66864C publication Critical patent/FI66864C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
FI782527A 1977-08-19 1978-08-18 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-oxo-4h-pyrido(1,2-a)pyrimidinderivat FI66864C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HUCI001765 1977-08-19
HU77CI1765A HU178910B (en) 1977-08-19 1977-08-19 Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines

Publications (3)

Publication Number Publication Date
FI782527A true FI782527A (fi) 1979-02-20
FI66864B FI66864B (fi) 1984-08-31
FI66864C FI66864C (fi) 1984-12-10

Family

ID=10994667

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782527A FI66864C (fi) 1977-08-19 1978-08-18 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4-oxo-4h-pyrido(1,2-a)pyrimidinderivat

Country Status (22)

Country Link
US (2) US4219649A (fi)
JP (1) JPS5448795A (fi)
AT (1) AT368156B (fi)
AU (1) AU518364B2 (fi)
BE (1) BE869832A (fi)
CA (1) CA1152989A (fi)
CH (1) CH637541A5 (fi)
CS (1) CS238901B1 (fi)
DD (1) DD138320A5 (fi)
DE (1) DE2835004A1 (fi)
DK (1) DK160045C (fi)
ES (1) ES473181A1 (fi)
FI (1) FI66864C (fi)
FR (1) FR2416892A1 (fi)
GB (1) GB2006187B (fi)
GR (1) GR64913B (fi)
HU (1) HU178910B (fi)
IL (1) IL55338A (fi)
NL (1) NL7808570A (fi)
SE (1) SE435383B (fi)
SU (1) SU906378A3 (fi)
YU (1) YU40985B (fi)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU179143B (en) * 1977-12-29 1982-08-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydroxy-groops-containing 6,7-dihydro-pyrido-square bracket-1,2-a-square bracket closed-pyrimidin derivatives and esters thereof
HU180701B (en) * 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
FR2449689A1 (fr) * 1979-02-20 1980-09-19 Logeais Labor Jacques Nouveaux derives condenses de pyrrolidine ou de piperidine, leur procede de preparation et leurs applications en therapeutique
IL59802A (en) 1979-05-08 1983-07-31 Erba Farmitalia Substituted pyrido(1,2-a)pyrimidine carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
PL129375B1 (en) * 1980-07-24 1984-05-31 Rhone Poulenc Ind Process for preparing novel derivatives of 2,3,6,7-tetrahydro-thiazole-/3,2-a/-pyrimidin-5-one
HU183408B (en) * 1981-04-28 1984-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing oral ratard pharmaceutical compositions
CA1211111A (en) * 1982-02-15 1986-09-09 Isao Yanagisawa Process for preparing novel pyrimidone compounds
US5252572A (en) * 1988-02-03 1993-10-12 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt. Pyridopyrimidine derivatives, pharmaceutical compositions containing them and process for preparing same
WO1991016894A1 (en) * 1990-05-02 1991-11-14 Abbott Laboratories Quinolizinone type compounds
DE10050661A1 (de) * 2000-10-13 2002-04-18 Gruenenthal Gmbh Substituierte 3,4-Dihydro-pyrimido[1,2-a]pyrimidine und 3,4-Dihydro-pyrazino[1,2-a]pyrimidine
DE10050662A1 (de) * 2000-10-13 2002-04-18 Gruenenthal Gmbh Substituierte 3,4-Dihydro-pyrido[1,2-a]pyrimidine
DE20202183U1 (de) 2002-02-01 2002-06-06 Kretzschmar Michael Baukasten
CA2500952C (en) * 2002-10-04 2011-04-26 Prana Biotechnology Limited Neurologically-active compounds
EP2012789B1 (en) 2006-04-14 2013-09-25 Prana Biotechnology Limited Method of treatment of age-related macular degeneration (AMD)
US7955155B2 (en) 2007-07-09 2011-06-07 Mega Brands International Magnetic and electronic toy construction systems and elements
JP5649304B2 (ja) * 2007-11-13 2015-01-07 国立大学法人 東京大学 クオラムセンシング阻害剤
CA2727651C (en) * 2008-06-17 2016-04-05 Priscille Brodin Anti-infective compounds
CA2968090A1 (en) * 2014-12-02 2016-06-09 Prana Biotechnology Limited 4h-pyrido[1,2-a]pyrimidin-4-one compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT302311B (de) * 1966-11-02 1972-09-15 Chinoin Gyogyszer Es Vegyeszet Verfahren zur herstellung von homopyrimidazol-derivaten und deren saeureadditionssalzen und quaternaeren ammoniumsalzen
HU169230B (fi) * 1972-03-29 1976-10-28
HU168014B (fi) * 1973-03-30 1976-02-28
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
HU168541B (fi) * 1973-11-24 1976-05-28
US4022897A (en) * 1974-03-04 1977-05-10 E. R. Squibb & Sons, Inc. CNS active compounds
US3898224A (en) * 1974-09-09 1975-08-05 Squibb & Sons Inc 1,6,7,8-Tetrahydro-4-oxo-4H-pyrido {8 1,2-A{9 pyrimidine-9-carboalkoxy compounds
US3935197A (en) * 1975-05-16 1976-01-27 E. R. Squibb & Sons, Inc. 2-Styryl-4H-pyrido(1,2-a)pyrimidin-4-ones

Also Published As

Publication number Publication date
FR2416892A1 (fr) 1979-09-07
CS238901B1 (en) 1985-12-16
DE2835004C2 (fi) 1989-06-29
CS541778A1 (en) 1985-05-15
AU518364B2 (en) 1981-09-24
BE869832A (fr) 1978-12-18
FI66864B (fi) 1984-08-31
GB2006187A (en) 1979-05-02
NL7808570A (nl) 1979-02-21
JPS5448795A (en) 1979-04-17
IL55338A0 (en) 1978-10-31
IL55338A (en) 1985-10-31
ES473181A1 (es) 1979-04-01
JPS626554B2 (fi) 1987-02-12
CH637541A5 (de) 1983-08-15
DK367478A (da) 1979-02-20
SU906378A3 (ru) 1982-02-15
GB2006187B (en) 1982-10-06
SE435383B (sv) 1984-09-24
DE2835004A1 (de) 1979-03-01
DD138320A5 (de) 1979-10-24
GR64913B (en) 1980-06-09
HU178910B (en) 1982-07-28
US4219649A (en) 1980-08-26
AT368156B (de) 1982-09-27
DK160045C (da) 1991-06-10
US4291036A (en) 1981-09-22
DK160045B (da) 1991-01-21
FI66864C (fi) 1984-12-10
AU3900978A (en) 1980-02-21
ATA585278A (de) 1982-01-15
FR2416892B1 (fi) 1983-11-18
YU40985B (en) 1986-10-31
SE7808770L (sv) 1979-02-20
YU196678A (en) 1983-10-31
CA1152989A (en) 1983-08-30

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: CHINOIN GYOGUSZER ES VEGYESZETI TERMEKEK