SE444679B - Sett att framstella 5(6)-substituerad bensimidazol-(2)-metylkarbamat med antihelmintisk verkan - Google Patents
Sett att framstella 5(6)-substituerad bensimidazol-(2)-metylkarbamat med antihelmintisk verkanInfo
- Publication number
- SE444679B SE444679B SE7804305A SE7804305A SE444679B SE 444679 B SE444679 B SE 444679B SE 7804305 A SE7804305 A SE 7804305A SE 7804305 A SE7804305 A SE 7804305A SE 444679 B SE444679 B SE 444679B
- Authority
- SE
- Sweden
- Prior art keywords
- general formula
- give
- substituted benzimidazole
- antihelmintic
- make
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
- C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT22645/77A IT1076022B (it) | 1977-04-20 | 1977-04-20 | Benzimidazolcarbammati antielmintici |
Publications (2)
Publication Number | Publication Date |
---|---|
SE7804305L SE7804305L (sv) | 1978-10-21 |
SE444679B true SE444679B (sv) | 1986-04-28 |
Family
ID=11198787
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE7804305A SE444679B (sv) | 1977-04-20 | 1978-04-17 | Sett att framstella 5(6)-substituerad bensimidazol-(2)-metylkarbamat med antihelmintisk verkan |
Country Status (19)
Country | Link |
---|---|
US (1) | US4182893A (es) |
AR (1) | AR219526A1 (es) |
AT (1) | AT356672B (es) |
AU (1) | AU520133B2 (es) |
BE (1) | BE866195A (es) |
BR (1) | BR7802445A (es) |
CA (1) | CA1104142A (es) |
CH (1) | CH639077A5 (es) |
DE (1) | DE2816694C2 (es) |
DK (1) | DK154076C (es) |
FR (1) | FR2387965A1 (es) |
GB (1) | GB1581517A (es) |
IE (1) | IE46869B1 (es) |
IT (1) | IT1076022B (es) |
NL (1) | NL7804049A (es) |
NZ (1) | NZ187003A (es) |
SE (1) | SE444679B (es) |
SU (1) | SU764609A3 (es) |
ZA (1) | ZA782250B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4174400A (en) * | 1978-09-13 | 1979-11-13 | Merck & Co., Inc. | Anthelmintic benzimidazoles |
DE2845537A1 (de) * | 1978-10-19 | 1980-04-30 | Bayer Ag | Benzimidazolylcarbamidsaeureester, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
NL7908719A (nl) * | 1978-12-06 | 1980-06-10 | Montedison Spa | Benzimidazoolcarbamaten. |
US4299837A (en) | 1979-12-05 | 1981-11-10 | Montedison S.P.A. | Anthelmintic benzimidazole-carbamates |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK131821C (da) * | 1967-03-22 | 1976-03-08 | Smith Kline French Lab | Analogifremgangsmade til fremstilling af en 2-karbalkoksyaminobenzimidazol |
US3657267A (en) * | 1969-06-20 | 1972-04-18 | Janssen Pharmaceutica Nv | Benzimidazole carbamates |
BE793358A (fr) * | 1971-12-27 | 1973-06-27 | Hoechst Ag | Nouveaux derives de 2-carbalcoxy-amino-benzimidazole presentantune activite anthelmintique et leur procede de preparation |
US3929821A (en) * | 1972-12-29 | 1975-12-30 | Syntex Inc | 5 (6)-Benzene ring substituted benzimidazole-2-carbamate derivatives |
US3929824A (en) * | 1972-12-29 | 1975-12-30 | Syntex Inc | 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity |
US3929823A (en) * | 1973-11-21 | 1975-12-30 | Syntex Inc | 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity |
US3915986A (en) * | 1974-06-19 | 1975-10-28 | Smithkline Corp | Methyl 5-propylthio-2-benzimidazolecarbamate |
-
1977
- 1977-04-20 IT IT22645/77A patent/IT1076022B/it active
-
1978
- 1978-04-17 SE SE7804305A patent/SE444679B/sv not_active IP Right Cessation
- 1978-04-17 DK DK166278A patent/DK154076C/da not_active IP Right Cessation
- 1978-04-17 CH CH410378A patent/CH639077A5/it not_active IP Right Cessation
- 1978-04-17 NL NL7804049A patent/NL7804049A/xx not_active Application Discontinuation
- 1978-04-18 AR AR271814A patent/AR219526A1/es active
- 1978-04-18 AT AT272878A patent/AT356672B/de not_active IP Right Cessation
- 1978-04-18 DE DE2816694A patent/DE2816694C2/de not_active Expired
- 1978-04-18 NZ NZ187003A patent/NZ187003A/xx unknown
- 1978-04-18 AU AU35193/78A patent/AU520133B2/en not_active Expired
- 1978-04-19 BR BR7802445A patent/BR7802445A/pt unknown
- 1978-04-19 GB GB15476/78A patent/GB1581517A/en not_active Expired
- 1978-04-19 FR FR7811486A patent/FR2387965A1/fr active Granted
- 1978-04-19 ZA ZA00782250A patent/ZA782250B/xx unknown
- 1978-04-19 SU SU782608100A patent/SU764609A3/ru active
- 1978-04-19 IE IE769/78A patent/IE46869B1/en unknown
- 1978-04-19 US US05/897,853 patent/US4182893A/en not_active Expired - Lifetime
- 1978-04-20 CA CA301,605A patent/CA1104142A/en not_active Expired
- 1978-04-20 BE BE186963A patent/BE866195A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DE2816694C2 (de) | 1986-02-06 |
AR219526A1 (es) | 1980-08-29 |
CH639077A5 (it) | 1983-10-31 |
FR2387965B1 (es) | 1980-10-10 |
NL7804049A (nl) | 1978-10-24 |
DK166278A (da) | 1978-10-21 |
DE2816694A1 (de) | 1978-10-26 |
DK154076C (da) | 1989-02-27 |
ATA272878A (de) | 1979-10-15 |
CA1104142A (en) | 1981-06-30 |
FR2387965A1 (fr) | 1978-11-17 |
SE7804305L (sv) | 1978-10-21 |
US4182893A (en) | 1980-01-08 |
DK154076B (da) | 1988-10-10 |
BE866195A (fr) | 1978-10-20 |
IE780769L (en) | 1978-10-20 |
BR7802445A (pt) | 1978-12-19 |
IT1076022B (it) | 1985-04-22 |
ZA782250B (en) | 1979-04-25 |
AT356672B (de) | 1980-05-12 |
NZ187003A (en) | 1981-03-16 |
GB1581517A (en) | 1980-12-17 |
IE46869B1 (en) | 1983-10-19 |
AU3519378A (en) | 1979-10-25 |
SU764609A3 (ru) | 1980-09-15 |
AU520133B2 (en) | 1982-01-14 |
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Legal Events
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NUG | Patent has lapsed |
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