RU95110939A - Ингибирующие орнитиндекарбоксилазу разветвленные аминооксиаминоалкан производные - Google Patents

Ингибирующие орнитиндекарбоксилазу разветвленные аминооксиаминоалкан производные

Info

Publication number
RU95110939A
RU95110939A RU95110939/04A RU95110939A RU95110939A RU 95110939 A RU95110939 A RU 95110939A RU 95110939/04 A RU95110939/04 A RU 95110939/04A RU 95110939 A RU95110939 A RU 95110939A RU 95110939 A RU95110939 A RU 95110939A
Authority
RU
Russia
Prior art keywords
radicals
aminooxyaminoalkane
derivatives
ornithine decarboxylase
compounds
Prior art date
Application number
RU95110939/04A
Other languages
English (en)
Inventor
Фрай Йорг
Ch]
Станек Ярослав
Original Assignee
Циба-Гейги АГ (CH)
Циба-Гейги АГ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Циба-Гейги АГ (CH), Циба-Гейги АГ filed Critical Циба-Гейги АГ (CH)
Publication of RU95110939A publication Critical patent/RU95110939A/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C239/00Compounds containing nitrogen-to-halogen bonds; Hydroxylamino compounds or ethers or esters thereof
    • C07C239/08Hydroxylamino compounds or their ethers or esters
    • C07C239/20Hydroxylamino compounds or their ethers or esters having oxygen atoms of hydroxylamino groups etherified
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)

Abstract

Описаны соединения формулы I, указанной в описании, или их соли. Соединения формулы I и их соли ингибируют орнитиндекарбоксилазу.

Claims (1)

  1. Описаны соединения формулы I, указанной в описании, или их соли. Соединения формулы I и их соли ингибируют орнитиндекарбоксилазу.
RU95110939/04A 1993-04-13 1994-04-02 Ингибирующие орнитиндекарбоксилазу разветвленные аминооксиаминоалкан производные RU95110939A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH112993 1993-04-13
CH1129/93-6 1993-04-13

Publications (1)

Publication Number Publication Date
RU95110939A true RU95110939A (ru) 1996-10-27

Family

ID=4203174

Family Applications (1)

Application Number Title Priority Date Filing Date
RU95110939/04A RU95110939A (ru) 1993-04-13 1994-04-02 Ингибирующие орнитиндекарбоксилазу разветвленные аминооксиаминоалкан производные

Country Status (18)

Country Link
US (1) US5610195A (ru)
EP (1) EP0644873B1 (ru)
JP (1) JPH07508046A (ru)
CN (1) CN1034930C (ru)
AT (1) ATE150009T1 (ru)
AU (1) AU673073B2 (ru)
CA (1) CA2135781A1 (ru)
CZ (1) CZ7995A3 (ru)
DE (1) DE69402021T2 (ru)
DK (1) DK0644873T3 (ru)
ES (1) ES2102221T3 (ru)
GR (1) GR3023429T3 (ru)
HU (1) HUT72751A (ru)
NZ (1) NZ265253A (ru)
PL (1) PL306765A1 (ru)
RU (1) RU95110939A (ru)
SK (1) SK3795A3 (ru)
WO (1) WO1994024094A1 (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT70522A (en) * 1993-04-13 1995-10-30 Ciba Geigy Ag Ornithine decarboxylase inhibiting cyclic aminooxy compounds, process to prepare them and pharmaceutical compns. contg them
US20030185754A1 (en) * 2001-01-16 2003-10-02 Genset, S.A. Treatment of CNS disorders using D-amino acid oxidase and D-aspartate oxidase antagonists
US20030166554A1 (en) * 2001-01-16 2003-09-04 Genset, S.A. Treatment of CNS disorders using D-amino acid oxidase and D-aspartate oxidase antagonists

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB974163A (en) * 1960-04-08 1964-11-04 Ciba Ltd Manufacture of 1-amino-ªÏ-hydroxylamino-alkanes
US3137705A (en) * 1960-04-08 1964-06-16 Ciba Geigy Corp Hydroxylamino compounds
US3869278A (en) * 1972-07-27 1975-03-04 Merrill Wilcox Hydroxylamines and derivatives thereof as abscission agents
US4390534A (en) * 1978-12-29 1983-06-28 Fujisawa Pharmaceutical Co., Ltd. Cephem and cepham compounds
DE3501616A1 (de) * 1985-01-17 1986-07-17 Schering AG, 1000 Berlin und 4709 Bergkamen Verfahren zur herstellung von hydroxylamin-derivaten
US4853467A (en) * 1987-05-19 1989-08-01 Bristol-Myers Company Nitrogen containing derivatives of epipodophyllotoxin glucosides
GB8729521D0 (en) * 1987-12-18 1988-02-03 May & Baker Ltd New compositions of matter
EP0369944A1 (de) * 1988-11-18 1990-05-23 Ciba-Geigy Ag Substituierte Oxadiaminobutane
CA2014880A1 (en) * 1989-04-27 1990-10-27 Indu Sawhney Thiazole derivatives
NO903360L (no) * 1989-08-11 1991-02-12 Ici Pharma Antibiotiske forbindelser.
EP0483427A1 (en) * 1990-11-01 1992-05-06 The Procter & Gamble Company Amine deodorant composition and method of deodorization
HUT70522A (en) * 1993-04-13 1995-10-30 Ciba Geigy Ag Ornithine decarboxylase inhibiting cyclic aminooxy compounds, process to prepare them and pharmaceutical compns. contg them

Also Published As

Publication number Publication date
ES2102221T3 (es) 1997-07-16
SK3795A3 (en) 1995-05-10
ATE150009T1 (de) 1997-03-15
CN1034930C (zh) 1997-05-21
CA2135781A1 (en) 1994-10-27
HUT72751A (en) 1996-05-28
DK0644873T3 (da) 1997-04-07
NZ265253A (en) 1996-10-28
PL306765A1 (en) 1995-04-18
DE69402021D1 (en) 1997-04-17
CZ7995A3 (en) 1995-10-18
HU9500095D0 (en) 1995-03-28
US5610195A (en) 1997-03-11
WO1994024094A1 (en) 1994-10-27
EP0644873A1 (en) 1995-03-29
AU673073B2 (en) 1996-10-24
CN1104831A (zh) 1995-07-05
AU6564694A (en) 1994-11-08
GR3023429T3 (en) 1997-08-29
EP0644873B1 (en) 1997-03-12
JPH07508046A (ja) 1995-09-07
DE69402021T2 (de) 1997-10-30

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