RU2679407C1 - Аналоги гамма-аминомасляной кислоты (гамк) для лечения боли и других заболеваний - Google Patents
Аналоги гамма-аминомасляной кислоты (гамк) для лечения боли и других заболеваний Download PDFInfo
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- RU2679407C1 RU2679407C1 RU2016128012A RU2016128012A RU2679407C1 RU 2679407 C1 RU2679407 C1 RU 2679407C1 RU 2016128012 A RU2016128012 A RU 2016128012A RU 2016128012 A RU2016128012 A RU 2016128012A RU 2679407 C1 RU2679407 C1 RU 2679407C1
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Classifications
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- C07C259/14—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. N-hydroxyamidines having carbon atoms of hydroxamidine groups bound to hydrogen atoms or to acyclic carbon atoms
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| US201361917623P | 2013-12-18 | 2013-12-18 | |
| US61/917,623 | 2013-12-18 | ||
| PCT/EP2014/077937 WO2015091463A1 (en) | 2013-12-18 | 2014-12-16 | Gamma-aminobutyric acid (gaba) analogues for the treatment of pain and other disorders |
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| RU2679407C1 true RU2679407C1 (ru) | 2019-02-08 |
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| JP6491213B2 (ja) * | 2013-12-18 | 2019-03-27 | ノヴァッセイ エスエー | 疼痛および他の障害の治療のためのガンマ−アミノ酪酸（ｇａｂａ）類似体 |
| CN107667097B (zh) * | 2015-05-27 | 2021-02-12 | 诺瓦色生物公司 | 3-乙基双环[3.2.0]庚-3-烯-6-酮的对映体的分离 |
| CN110818582B (zh) * | 2019-11-20 | 2023-06-09 | 合肥拓锐生物科技有限公司 | 一种gaba类似物及其盐，及其合成方法、应用、药物 |
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| RU2115655C1 (ru) * | 1995-03-09 | 1998-07-20 | Вакер-Хеми ГмбХ | Способ получения ди- и триалкилсиланов |
| EP1199072A2 (en) * | 2000-10-17 | 2002-04-24 | Warner-Lambert Company | Method of treating cartilage damage |
| RU2446148C2 (ru) * | 2007-09-28 | 2012-03-27 | Дайити Санкио Компани, Лимитед | Бициклическое производное гамма-аминокислоты |
| WO2015005298A1 (ja) * | 2013-07-08 | 2015-01-15 | 第一三共株式会社 | 光学活性な二環性γ－アミノ酸誘導体の製造方法 |
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| CN1131855C (zh) * | 1997-12-16 | 2003-12-24 | 沃尼尔·朗伯公司 | 1－取代－1－氨基甲基－环烷衍生物(=加巴喷丁类似物)、其制备及其在治疗神经病方面的用途 |
| NZ545494A (en) * | 2003-09-12 | 2009-10-30 | Pfizer | Combinations comprising alpha-2-delta ligands and serotonin / noradrenaline re-uptake inhibitors |
| WO2010079668A1 (ja) | 2009-01-08 | 2010-07-15 | 第一三共株式会社 | オレフィン化合物 |
| JP5557292B2 (ja) | 2009-03-26 | 2014-07-23 | 第一三共株式会社 | 二環性γ−アミノ酸誘導体の製造方法 |
| CN104755465A (zh) * | 2012-08-24 | 2015-07-01 | 武田药品工业株式会社 | 杂环化合物 |
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- 2014-12-16 RU RU2016128012A patent/RU2679407C1/ru active
- 2014-12-16 CA CA2932050A patent/CA2932050C/en active Active
- 2014-12-16 WO PCT/EP2014/077937 patent/WO2015091463A1/en not_active Ceased
- 2014-12-16 CN CN201910061968.8A patent/CN109721562A/zh active Pending
- 2014-12-16 EP EP14821571.8A patent/EP3083572B1/en active Active
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2016
- 2016-11-22 US US15/359,120 patent/US9750720B2/en active Active
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2115655C1 (ru) * | 1995-03-09 | 1998-07-20 | Вакер-Хеми ГмбХ | Способ получения ди- и триалкилсиланов |
| EP1199072A2 (en) * | 2000-10-17 | 2002-04-24 | Warner-Lambert Company | Method of treating cartilage damage |
| RU2446148C2 (ru) * | 2007-09-28 | 2012-03-27 | Дайити Санкио Компани, Лимитед | Бициклическое производное гамма-аминокислоты |
| EP2192109B1 (en) * | 2007-09-28 | 2013-09-04 | Daiichi Sankyo Company, Limited | Bicyclic -amino acid derivative |
| WO2015005298A1 (ja) * | 2013-07-08 | 2015-01-15 | 第一三共株式会社 | 光学活性な二環性γ－アミノ酸誘導体の製造方法 |
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| CA2932050A1 (en) | 2015-06-25 |
| CA2932050C (en) | 2023-09-26 |
| CN105899495B (zh) | 2019-02-19 |
| WO2015091463A1 (en) | 2015-06-25 |
| EP3083572B1 (en) | 2019-02-13 |
| KR102031334B1 (ko) | 2019-10-11 |
| US9750720B2 (en) | 2017-09-05 |
| US9663479B2 (en) | 2017-05-30 |
| JP2017502020A (ja) | 2017-01-19 |
| KR20160095166A (ko) | 2016-08-10 |
| EP3083572A1 (en) | 2016-10-26 |
| US20160318885A1 (en) | 2016-11-03 |
| US20170071909A1 (en) | 2017-03-16 |
| CN109721562A (zh) | 2019-05-07 |
| AU2014364693A1 (en) | 2016-07-28 |
| AU2014364693B2 (en) | 2018-12-06 |
| CN105899495A (zh) | 2016-08-24 |
| JP6491213B2 (ja) | 2019-03-27 |
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