RU2638137C2 - Твердые формы внутренней соли пиридопиримидиния - Google Patents

Твердые формы внутренней соли пиридопиримидиния Download PDF

Info

Publication number
RU2638137C2
RU2638137C2 RU2015101646A RU2015101646A RU2638137C2 RU 2638137 C2 RU2638137 C2 RU 2638137C2 RU 2015101646 A RU2015101646 A RU 2015101646A RU 2015101646 A RU2015101646 A RU 2015101646A RU 2638137 C2 RU2638137 C2 RU 2638137C2
Authority
RU
Russia
Prior art keywords
methyl
compound
polymorphic form
dichlorophenyl
thiazolyl
Prior art date
Application number
RU2015101646A
Other languages
English (en)
Russian (ru)
Other versions
RU2015101646A (ru
Inventor
Кристиан ХОФФМАНН
Вэньмин Чжан
Юйчжун ЧЭНЬ
Original Assignee
Е.И.Дюпон Де Немур Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Е.И.Дюпон Де Немур Энд Компани filed Critical Е.И.Дюпон Де Немур Энд Компани
Publication of RU2015101646A publication Critical patent/RU2015101646A/ru
Application granted granted Critical
Publication of RU2638137C2 publication Critical patent/RU2638137C2/ru

Links

Images

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
RU2015101646A 2012-06-21 2013-06-14 Твердые формы внутренней соли пиридопиримидиния RU2638137C2 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261662532P 2012-06-21 2012-06-21
US61/662,532 2012-06-21
PCT/US2013/045815 WO2013192035A1 (en) 2012-06-21 2013-06-14 Solid forms of a pyrido-pyrimidinium inner salt

Publications (2)

Publication Number Publication Date
RU2015101646A RU2015101646A (ru) 2016-08-10
RU2638137C2 true RU2638137C2 (ru) 2017-12-15

Family

ID=48692690

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2015101646A RU2638137C2 (ru) 2012-06-21 2013-06-14 Твердые формы внутренней соли пиридопиримидиния

Country Status (18)

Country Link
US (1) US9238650B2 (enrdf_load_stackoverflow)
EP (1) EP2864327B1 (enrdf_load_stackoverflow)
JP (1) JP6272843B2 (enrdf_load_stackoverflow)
KR (1) KR102047575B1 (enrdf_load_stackoverflow)
CN (1) CN104540824B (enrdf_load_stackoverflow)
AR (2) AR091521A1 (enrdf_load_stackoverflow)
AU (1) AU2013277462B2 (enrdf_load_stackoverflow)
BR (1) BR112014032385A2 (enrdf_load_stackoverflow)
CA (1) CA2876941C (enrdf_load_stackoverflow)
ES (1) ES2617554T3 (enrdf_load_stackoverflow)
IL (1) IL236106B (enrdf_load_stackoverflow)
IN (1) IN2015DN00375A (enrdf_load_stackoverflow)
MX (1) MX352976B (enrdf_load_stackoverflow)
MY (1) MY168088A (enrdf_load_stackoverflow)
RU (1) RU2638137C2 (enrdf_load_stackoverflow)
TW (1) TWI592412B (enrdf_load_stackoverflow)
WO (1) WO2013192035A1 (enrdf_load_stackoverflow)
ZA (1) ZA201409327B (enrdf_load_stackoverflow)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
JP2016522173A (ja) 2013-04-19 2016-07-28 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 有害動物を駆除するためのｎ−置換アシル−イミノ−ピリジン化合物および誘導体
BR112016008555A8 (pt) 2013-10-18 2020-03-10 Basf Agrochemical Products Bv usos do composto carboxamida ativo pesticida e método de proteção de material de propagação vegetal
WO2015104422A1 (en) 2014-01-13 2015-07-16 Basf Se Dihydrothiophene compounds for controlling invertebrate pests
CN118266473A (zh) * 2014-12-22 2024-07-02 日本农药株式会社 用于农业和园艺应用的有害生物防除剂组合物和应用该组合物的方法
CN110317200B (zh) * 2018-03-28 2020-09-11 东莞市东阳光农药研发有限公司 嘧啶鎓化合物及其用途
CN111096326A (zh) * 2018-10-26 2020-05-05 燕化永乐（乐亭）生物科技有限公司 一种杀虫组合物
CN111642510A (zh) * 2020-07-03 2020-09-11 浙江中山化工集团股份有限公司 一种含二氯噻吡嘧啶和蛇床子素的农药组合物
KR20250078983A (ko) * 2022-09-30 2025-06-04 아다마 마켓심 리미티드 효율적인 살충 방제를 위한 노발루론 혼합물
CN119096987B (zh) * 2024-09-02 2025-09-05 漯河市农业科学院 一种防治蛴螬的农药组合物

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5089501A (en) * 1989-09-01 1992-02-18 Ciba Geigy Corp Anthelmintics
WO2011017342A2 (en) * 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides
EA201070926A1 (ru) * 2008-02-06 2011-04-29 Е.И.Дюпон Де Немур Энд Компани Мезоионные пестициды

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2891855A (en) 1954-08-16 1959-06-23 Geigy Ag J R Compositions and methods for influencing the growth of plants
US3235361A (en) 1962-10-29 1966-02-15 Du Pont Method for the control of undesirable vegetation
US3060084A (en) 1961-06-09 1962-10-23 Du Pont Improved homogeneous, readily dispersed, pesticidal concentrate
US3299566A (en) 1964-06-01 1967-01-24 Olin Mathieson Water soluble film containing agricultural chemicals
US3309192A (en) 1964-12-02 1967-03-14 Du Pont Method of controlling seedling weed grasses
US4144050A (en) 1969-02-05 1979-03-13 Hoechst Aktiengesellschaft Micro granules for pesticides and process for their manufacture
US3920442A (en) 1972-09-18 1975-11-18 Du Pont Water-dispersible pesticide aggregates
US4172714A (en) 1976-12-20 1979-10-30 E. I. Du Pont De Nemours And Company Dry compactible, swellable herbicidal compositions and pellets produced therefrom
GB2095558B (en) 1981-03-30 1984-10-24 Avon Packers Ltd Formulation of agricultural chemicals
DE3246493A1 (de) 1982-12-16 1984-06-20 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von wasserdispergierbaren granulaten
US5180587A (en) 1988-06-28 1993-01-19 E. I. Du Pont De Nemours And Company Tablet formulations of pesticides
ZW13690A1 (en) 1989-08-30 1990-11-21 Aeci Ltd Active ingredient dosage device
EP0430885A3 (en) * 1989-12-01 1991-11-06 Ciba-Geigy Ag Anthelmintical compounds
PL167613B1 (pl) 1990-03-12 1995-09-30 Du Pont Granulowana kompozycja rozpuszczalna lub dyspergowalna w wodzie PL
ES2091878T3 (es) 1990-10-11 1996-11-16 Sumitomo Chemical Co Composicion plaguicida.
US6406690B1 (en) 1995-04-17 2002-06-18 Minrav Industries Ltd. Bacillus firmus CNCM I-1582 or Bacillus cereus CNCM I-1562 for controlling nematodes
TW200724033A (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI572587B (zh) 2011-12-15 2017-03-01 杜邦股份有限公司 丙二酸二鹽及用以製備丙二醯基二鹵化物之方法

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5089501A (en) * 1989-09-01 1992-02-18 Ciba Geigy Corp Anthelmintics
EA201070926A1 (ru) * 2008-02-06 2011-04-29 Е.И.Дюпон Де Немур Энд Компани Мезоионные пестициды
WO2011017342A2 (en) * 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides

Also Published As

Publication number Publication date
ES2617554T3 (es) 2017-06-19
ZA201409327B (en) 2016-09-28
EP2864327B1 (en) 2016-12-14
AR120841A2 (es) 2022-03-23
JP2015521620A (ja) 2015-07-30
KR102047575B1 (ko) 2019-11-21
AU2013277462B2 (en) 2017-06-29
IN2015DN00375A (enrdf_load_stackoverflow) 2015-06-12
BR112014032385A2 (pt) 2017-06-27
JP6272843B2 (ja) 2018-01-31
MX2014015663A (es) 2015-04-09
EP2864327A1 (en) 2015-04-29
TW201400483A (zh) 2014-01-01
WO2013192035A1 (en) 2013-12-27
AU2013277462A1 (en) 2015-01-22
RU2015101646A (ru) 2016-08-10
US9238650B2 (en) 2016-01-19
CN104540824A (zh) 2015-04-22
CA2876941A1 (en) 2013-12-27
IL236106A0 (en) 2015-02-01
MX352976B (es) 2017-12-15
KR20150021058A (ko) 2015-02-27
MY168088A (en) 2018-10-11
US20150252040A1 (en) 2015-09-10
AR091521A1 (es) 2015-02-11
CN104540824B (zh) 2017-03-29
CA2876941C (en) 2021-01-26
TWI592412B (zh) 2017-07-21
IL236106B (en) 2018-12-31

Similar Documents

Publication Publication Date Title
KR102336442B1 (ko) 복소환 치환된 이환식 아졸계 농약
RU2638137C2 (ru) Твердые формы внутренней соли пиридопиримидиния
RU2585616C2 (ru) МЕЗОИОННЫЕ ПИРИДО[1,2-a]ПИРИМИДИНОВЫЕ ПЕСТИЦИДЫ
JP7146005B2 (ja) 二環式ピラゾール殺有害生物剤
RU2758667C2 (ru) Замещенные по гетероциклу бициклические азол пестициды
KR102604099B1 (ko) 메소이온성 살곤충제
KR101951976B1 (ko) 1,3-다이아릴 치환된 복소환식 살충제
TWI812673B (zh) 用於防治無脊椎害蟲之萘異噁唑啉化合物
CN104302637A (zh) 1,3-二芳基取代的杂环杀虫剂
TW202005533A (zh) 包含吲唑之殺蟲混合物
KR20210033494A (ko) 무척추동물 해충을 방제하기 위한 이속사졸린 화합물
KR102389531B1 (ko) 1-아릴-3-알킬피라졸 살충제
KR102447284B1 (ko) 헤테로사이클-치환된 비시클릭 아졸 살충제
JP6937748B2 (ja) 複素環で置換した二環式アゾール有害生物防除剤
KR20250121575A (ko) 무척추동물 해충을 방제 및 퇴치하기 위한 아졸 화합물

Legal Events

Date Code Title Description
PD4A Correction of name of patent owner
PC41 Official registration of the transfer of exclusive right

Effective date: 20190111