IN2015DN00375A - - Google Patents

Info

Publication number
IN2015DN00375A
IN2015DN00375A IN375DEN2015A IN2015DN00375A IN 2015DN00375 A IN2015DN00375 A IN 2015DN00375A IN 375DEN2015 A IN375DEN2015 A IN 375DEN2015A IN 2015DN00375 A IN2015DN00375 A IN 2015DN00375A
Authority
IN
India
Prior art keywords
compound
disclosed
solid form
solid
seed
Prior art date
Application number
Inventor
Christian Hoffmann
Wenming Zhang
Yuzhong Chen
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Publication of IN2015DN00375A publication Critical patent/IN2015DN00375A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/781,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Disclosed are solid forms of 1-[(2-chloro-5-thiazolyl)methyl]-3-(3,5-dichlorophenyl)- 2-hydroxy-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidinium inner salt (Compound 15 ). Methods for the preparation of solid forms of Compound 1 and for the conversion of one solid form of Compound 1 into another are disclosed. Disclosed are compositions for controlling an invertebrate pest comprising a biologically effective amount of a solid form of Compound 1 and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid carriers. Compositions comprising a mixture of a solid form of Compound 1 and at least one other nematocide, insecticide and/or fungicide are also disclosed. Also disclosed are methods for controlling invertebrate pests comprising applying to a plant or seed, or to the environment of the plant or seed, a biologically effective amount of a solid form of Compound 1.
IN375DEN2015 2012-06-21 2013-06-14 IN2015DN00375A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261662532P 2012-06-21 2012-06-21
PCT/US2013/045815 WO2013192035A1 (en) 2012-06-21 2013-06-14 Solid forms of a pyrido-pyrimidinium inner salt

Publications (1)

Publication Number Publication Date
IN2015DN00375A true IN2015DN00375A (en) 2015-06-12

Family

ID=48692690

Family Applications (1)

Application Number Title Priority Date Filing Date
IN375DEN2015 IN2015DN00375A (en) 2012-06-21 2013-06-14

Country Status (18)

Country Link
US (1) US9238650B2 (en)
EP (1) EP2864327B1 (en)
JP (1) JP6272843B2 (en)
KR (1) KR102047575B1 (en)
CN (1) CN104540824B (en)
AR (2) AR091521A1 (en)
AU (1) AU2013277462B2 (en)
BR (1) BR112014032385A2 (en)
CA (1) CA2876941C (en)
ES (1) ES2617554T3 (en)
IL (1) IL236106B (en)
IN (1) IN2015DN00375A (en)
MX (1) MX352976B (en)
MY (1) MY168088A (en)
RU (1) RU2638137C2 (en)
TW (1) TWI592412B (en)
WO (1) WO2013192035A1 (en)
ZA (1) ZA201409327B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA110924C2 (en) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Mesoionic pesticides
US20160050923A1 (en) 2013-04-19 2016-02-25 Basf Se N-substituted acyl-imino-pyridine compounds and derivatives for combating animal pests
WO2015055757A1 (en) 2013-10-18 2015-04-23 Basf Se Use of pesticidal active carboxamide derivative in soil and seed application and treatment methods
WO2015104422A1 (en) 2014-01-13 2015-07-16 Basf Se Dihydrothiophene compounds for controlling invertebrate pests
JP6731351B2 (en) * 2014-12-22 2020-07-29 日本農薬株式会社 Agro-horticultural pest control composition and method of using the same
CN110317200B (en) * 2018-03-28 2020-09-11 东莞市东阳光农药研发有限公司 Pyrimidinium compounds and uses thereof
CN111096326A (en) * 2018-10-26 2020-05-05 燕化永乐(乐亭)生物科技有限公司 Insecticidal composition
CN111642510A (en) * 2020-07-03 2020-09-11 浙江中山化工集团股份有限公司 Pesticide composition containing imidaclothizine and osthole
WO2024069632A2 (en) * 2022-09-30 2024-04-04 Adama Makhteshim Ltd. Novaluron mixtures for efficient insecticidal controls

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2891855A (en) 1954-08-16 1959-06-23 Geigy Ag J R Compositions and methods for influencing the growth of plants
US3235361A (en) 1962-10-29 1966-02-15 Du Pont Method for the control of undesirable vegetation
US3060084A (en) 1961-06-09 1962-10-23 Du Pont Improved homogeneous, readily dispersed, pesticidal concentrate
US3299566A (en) 1964-06-01 1967-01-24 Olin Mathieson Water soluble film containing agricultural chemicals
US3309192A (en) 1964-12-02 1967-03-14 Du Pont Method of controlling seedling weed grasses
US4144050A (en) 1969-02-05 1979-03-13 Hoechst Aktiengesellschaft Micro granules for pesticides and process for their manufacture
US3920442A (en) 1972-09-18 1975-11-18 Du Pont Water-dispersible pesticide aggregates
US4172714A (en) 1976-12-20 1979-10-30 E. I. Du Pont De Nemours And Company Dry compactible, swellable herbicidal compositions and pellets produced therefrom
GB2095558B (en) 1981-03-30 1984-10-24 Avon Packers Ltd Formulation of agricultural chemicals
DE3246493A1 (en) 1982-12-16 1984-06-20 Bayer Ag, 5090 Leverkusen METHOD FOR PRODUCING WATER-DISPERSIBLE GRANULES
US5180587A (en) 1988-06-28 1993-01-19 E. I. Du Pont De Nemours And Company Tablet formulations of pesticides
ES2166919T3 (en) 1989-08-30 2002-05-01 Kynoch Agrochemicals Proprieta PREPARATION OF A DOSING DEVICE.
EP0415889A3 (en) * 1989-09-01 1991-08-28 Ciba-Geigy Ag Anthelmintic agent
EP0430885A3 (en) * 1989-12-01 1991-11-06 Ciba-Geigy Ag Anthelmintical compounds
CA2083185A1 (en) 1990-03-12 1991-09-13 William Lawrence Geigle Water-dispersible or water-soluble pesticide granules from heat-activated binders
DE69122201T2 (en) 1990-10-11 1997-02-06 Sumitomo Chemical Co Pesticides composition
US6406690B1 (en) 1995-04-17 2002-06-18 Minrav Industries Ltd. Bacillus firmus CNCM I-1582 or Bacillus cereus CNCM I-1562 for controlling nematodes
TW200724033A (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI468407B (en) * 2008-02-06 2015-01-11 Du Pont Mesoionic pesticides
UA110924C2 (en) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Mesoionic pesticides
TWI572587B (en) 2011-12-15 2017-03-01 杜邦股份有限公司 Malonic acid di-salts and a method for preparing malonyl dihalides

Also Published As

Publication number Publication date
JP6272843B2 (en) 2018-01-31
IL236106A0 (en) 2015-02-01
CN104540824B (en) 2017-03-29
RU2638137C2 (en) 2017-12-15
AU2013277462A1 (en) 2015-01-22
MY168088A (en) 2018-10-11
KR102047575B1 (en) 2019-11-21
IL236106B (en) 2018-12-31
CA2876941A1 (en) 2013-12-27
AU2013277462B2 (en) 2017-06-29
BR112014032385A2 (en) 2017-06-27
CA2876941C (en) 2021-01-26
KR20150021058A (en) 2015-02-27
EP2864327A1 (en) 2015-04-29
TW201400483A (en) 2014-01-01
TWI592412B (en) 2017-07-21
US20150252040A1 (en) 2015-09-10
MX2014015663A (en) 2015-04-09
AR120841A2 (en) 2022-03-23
JP2015521620A (en) 2015-07-30
CN104540824A (en) 2015-04-22
US9238650B2 (en) 2016-01-19
EP2864327B1 (en) 2016-12-14
RU2015101646A (en) 2016-08-10
WO2013192035A1 (en) 2013-12-27
ES2617554T3 (en) 2017-06-19
AR091521A1 (en) 2015-02-11
MX352976B (en) 2017-12-15
ZA201409327B (en) 2016-09-28

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