RU2302240C2 - Производные карбаматов для предотвращения или лечения психотических нарушений - Google Patents

Производные карбаматов для предотвращения или лечения психотических нарушений Download PDF

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Publication number
RU2302240C2
RU2302240C2 RU2003128983/14A RU2003128983A RU2302240C2 RU 2302240 C2 RU2302240 C2 RU 2302240C2 RU 2003128983/14 A RU2003128983/14 A RU 2003128983/14A RU 2003128983 A RU2003128983 A RU 2003128983A RU 2302240 C2 RU2302240 C2 RU 2302240C2
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RU
Russia
Prior art keywords
formula
group
disorder
enantiomer
psychotic
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RU2003128983/14A
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English (en)
Russian (ru)
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RU2003128983A (ru
Inventor
Карлос Р. ПЛАТА-САЛАМАН (US)
Карлос Р. Плата-Саламан
Бою ЗАО (US)
Бою ЗАО
Рой Э. ТУАЙМЭН (US)
Рой Э. ТУАЙМЭН
Original Assignee
Орто-Макнейл Фармасьютикал, Инк.
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Publication of RU2003128983A publication Critical patent/RU2003128983A/ru
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Publication of RU2302240C2 publication Critical patent/RU2302240C2/ru

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/325Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RU2003128983/14A 2001-02-27 2002-02-21 Производные карбаматов для предотвращения или лечения психотических нарушений RU2302240C2 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US27188901P 2001-02-27 2001-02-27
US60/271,889 2001-02-27
US10/081,761 2002-02-21
US10/081,761 US6541513B2 (en) 2001-02-27 2002-02-21 Carbamate compounds for use in preventing or treating psychotic disorders

Publications (2)

Publication Number Publication Date
RU2003128983A RU2003128983A (ru) 2005-03-10
RU2302240C2 true RU2302240C2 (ru) 2007-07-10

Family

ID=26765939

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2003128983/14A RU2302240C2 (ru) 2001-02-27 2002-02-21 Производные карбаматов для предотвращения или лечения психотических нарушений

Country Status (25)

Country Link
US (1) US6541513B2 (https=)
EP (1) EP1401424B1 (https=)
JP (1) JP4276841B2 (https=)
KR (1) KR100886578B1 (https=)
CN (1) CN1262271C (https=)
AR (1) AR032876A1 (https=)
AT (1) ATE346597T1 (https=)
AU (1) AU2002242296B2 (https=)
BR (1) BR0207829A (https=)
CA (1) CA2439480C (https=)
CZ (1) CZ302412B6 (https=)
DE (1) DE60216457T2 (https=)
DK (1) DK1401424T3 (https=)
ES (1) ES2275844T3 (https=)
HU (1) HUP0303342A3 (https=)
IL (2) IL157588A0 (https=)
MX (1) MXPA03007722A (https=)
NO (1) NO20033801L (https=)
NZ (1) NZ527991A (https=)
PL (1) PL365021A1 (https=)
PT (1) PT1401424E (https=)
RS (1) RS51056B (https=)
RU (1) RU2302240C2 (https=)
TW (1) TWI251486B (https=)
WO (1) WO2002067927A1 (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE267629T1 (de) * 2000-07-21 2004-06-15 Ortho Mcneil Pharm Inc Verwendung von carbamat verbindungen zur vorbeugung oder behandlung von neuropathischen- , cluster- und migräneartigen kopfschmerzen
EP1383489B1 (en) * 2001-02-27 2007-05-09 Ortho-Mcneil Pharmaceutical, Inc. Carbamate compounds for use in preventing or treating neurodegenerative disorders
IL157594A0 (en) 2001-02-27 2004-03-28 Ortho Mcneil Pharm Inc Carbamate compounds for use in preventing or treating anxiety disorders
ATE435014T1 (de) 2001-07-16 2009-07-15 Ortho Mcneil Pharm Inc Carbamate verbindungen zur vorbeugung oder behandlung von neuropathischen schmerzen
EP1744750A2 (en) * 2004-05-06 2007-01-24 Sandoz AG Pharmaceutical composition comprising hydrophobic drug having improved solubility
ES2385087T3 (es) * 2005-07-26 2012-07-18 Sk Biopharmaceuticals Co., Ltd Procedimientos para tratar trastornos relacionados con sustancias
EP2081648A2 (en) * 2006-10-30 2009-07-29 Janssen Pharmaceutica, N.V. Carbamate compounds for use in treating depression
BRPI0718323A2 (pt) * 2006-10-31 2013-11-26 Janssen Pharmaceutica Nv Tratamento de transtornos invasivos do desenvolvimento.
US8609849B1 (en) 2010-11-30 2013-12-17 Fox Chase Chemical Diversity Center, Inc. Hydroxylated sulfamides exhibiting neuroprotective action and their method of use
CN105189451A (zh) * 2013-03-12 2015-12-23 比皮艾思药物研发有限公司 氨基甲酸苯酯化合物和包含该化合物的用于预防或治疗神经性毒气引起的疾病的组合物
CN109939092B (zh) 2013-03-12 2022-03-22 比皮艾思药物研发有限公司 用于预防或治疗小儿癫痫和癫痫相关综合征的苯基氨基甲酸酯化合物
KR102900173B1 (ko) * 2016-12-14 2025-12-12 에스케이바이오팜 주식회사 조현병, 강박장애 및 투렛증후군으로부터 선택되는 정신증 장애의 예방, 경감 또는 치료에 있어서의 카바메이트 화합물의 용도

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US278380A (en) * 1883-05-29 Thermometer
US3265728A (en) * 1962-07-18 1966-08-09 Armour Pharma Substituted phenethyl carbamates
RU2023712C1 (ru) * 1989-06-09 1994-11-30 Дзе Апджон Компани Трициклические азотсодержащие соединения и производные тетрагидрохинолина или их фармацевтически приемлемые соли
US5492930A (en) * 1994-04-25 1996-02-20 Schering Corporation Method and formulation for treating CNS disorders
US6103759A (en) * 1996-01-16 2000-08-15 Sk Corporation Halogen substituted carbamate compounds from 2-phenyl-1, 2-ethanediol

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3313692A (en) * 1958-04-21 1967-04-11 Armour Pharma Method of inducing calming and muscle relaxation with carbamates

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US278380A (en) * 1883-05-29 Thermometer
US3265728A (en) * 1962-07-18 1966-08-09 Armour Pharma Substituted phenethyl carbamates
RU2023712C1 (ru) * 1989-06-09 1994-11-30 Дзе Апджон Компани Трициклические азотсодержащие соединения и производные тетрагидрохинолина или их фармацевтически приемлемые соли
US5492930A (en) * 1994-04-25 1996-02-20 Schering Corporation Method and formulation for treating CNS disorders
US6103759A (en) * 1996-01-16 2000-08-15 Sk Corporation Halogen substituted carbamate compounds from 2-phenyl-1, 2-ethanediol

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
КАПЛАН Г. и др. Клиническая психиатрия. - М.: ГЭОТАР МЕДИЦИНА, 1994, с.124. VOVIN R.Ia. et al. Effectiveness of finlepsin in the prophylactic therapy of phasic affective psychoses. Zh Nevropatol Psikhiatr Im S S Korsakova. 1987; 87(9):1396-400. *
Психиатрия. / Под ред. Р.Шейдера. - М.: Практика, 1998, с.420. *

Also Published As

Publication number Publication date
TWI251486B (en) 2006-03-21
NZ527991A (en) 2005-04-29
HUP0303342A2 (hu) 2004-01-28
EP1401424A1 (en) 2004-03-31
ATE346597T1 (de) 2006-12-15
DE60216457D1 (de) 2007-01-11
KR100886578B1 (ko) 2009-03-05
DE60216457T2 (de) 2007-09-20
NO20033801L (no) 2003-10-22
EP1401424B1 (en) 2006-11-29
RS67503A (sr) 2006-12-15
CA2439480A1 (en) 2002-09-06
PT1401424E (pt) 2007-02-28
IL157588A0 (en) 2004-03-28
US20020165272A1 (en) 2002-11-07
CZ20032297A3 (cs) 2004-06-16
CN1262271C (zh) 2006-07-05
MXPA03007722A (es) 2004-11-12
CA2439480C (en) 2011-04-26
KR20030076713A (ko) 2003-09-26
DK1401424T3 (da) 2007-02-26
BR0207829A (pt) 2004-06-22
WO2002067927A1 (en) 2002-09-06
PL365021A1 (en) 2004-12-27
JP4276841B2 (ja) 2009-06-10
ES2275844T3 (es) 2007-06-16
IL157588A (en) 2009-12-24
US6541513B2 (en) 2003-04-01
AR032876A1 (es) 2003-11-26
RS51056B (sr) 2010-10-31
NO20033801D0 (no) 2003-08-26
JP2004523556A (ja) 2004-08-05
RU2003128983A (ru) 2005-03-10
CN1505507A (zh) 2004-06-16
AU2002242296B2 (en) 2006-06-29
CZ302412B6 (cs) 2011-05-04
HUP0303342A3 (en) 2012-07-30

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PC43 Official registration of the transfer of the exclusive right without contract for inventions

Effective date: 20190207

PD4A Correction of name of patent owner
PC41 Official registration of the transfer of exclusive right

Effective date: 20190506