BR0207829A - Composto de carbamato para uso na prevenção ou tratamento de distúrbios psicóticos - Google Patents
Composto de carbamato para uso na prevenção ou tratamento de distúrbios psicóticosInfo
- Publication number
- BR0207829A BR0207829A BR0207829-5A BR0207829A BR0207829A BR 0207829 A BR0207829 A BR 0207829A BR 0207829 A BR0207829 A BR 0207829A BR 0207829 A BR0207829 A BR 0207829A
- Authority
- BR
- Brazil
- Prior art keywords
- group
- psychotic disorders
- prevention
- treatment
- phenyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pain & Pain Management (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
"COMPOSTOS DE CARBAMATO PARA USO NA PREVENçãO OU TRATAMENTO DE DISTúRBIOS PSICóTICOS". A presente invenção refere-se a um método para prevenir ou tratar distúrbios psicóticos compreendendo administrar a um indivíduo em necessidade deste uma quantidade terapeuticamente eficaz de um composto selecionado do grupo que consiste na Fórmula (I) e Fórmula (II): onde fenila é substituída em X com um a cinco átomos de halogênio selecionados do grupo que consiste em flúor, cloro, bromo e iodo; e, R~ 1~, R~ 2~, R~ 3~, R~ 4~, R~ 5~ e R~ 6~ são independentemente selecionados do grupo que consiste em hidrogênio e C~ 1~-C~ 4~ alquila; onde C~ 1~-C~ 4~ alquila é opcionalmente substituída por fenila (onde fenila é opcionalmente substituída por substituintes independentemente selecionados do grupo que consiste em halogênio, C~ 1~-C~ 4~ alquila, C~ 1~-C~ 4~ alcóxi, amino, nitro e ciano).
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US27188901P | 2001-02-27 | 2001-02-27 | |
PCT/US2002/006119 WO2002067927A1 (en) | 2001-02-27 | 2002-02-21 | Carbamate compounds for use in preventing or treating psychotic disorders |
US10/081,761 US6541513B2 (en) | 2001-02-27 | 2002-02-21 | Carbamate compounds for use in preventing or treating psychotic disorders |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0207829A true BR0207829A (pt) | 2004-06-22 |
Family
ID=26765939
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0207829-5A BR0207829A (pt) | 2001-02-27 | 2002-02-21 | Composto de carbamato para uso na prevenção ou tratamento de distúrbios psicóticos |
Country Status (25)
Country | Link |
---|---|
US (1) | US6541513B2 (pt) |
EP (1) | EP1401424B1 (pt) |
JP (1) | JP4276841B2 (pt) |
KR (1) | KR100886578B1 (pt) |
CN (1) | CN1262271C (pt) |
AR (1) | AR032876A1 (pt) |
AT (1) | ATE346597T1 (pt) |
AU (1) | AU2002242296B2 (pt) |
BR (1) | BR0207829A (pt) |
CA (1) | CA2439480C (pt) |
CZ (1) | CZ302412B6 (pt) |
DE (1) | DE60216457T2 (pt) |
DK (1) | DK1401424T3 (pt) |
ES (1) | ES2275844T3 (pt) |
HU (1) | HUP0303342A3 (pt) |
IL (2) | IL157588A0 (pt) |
MX (1) | MXPA03007722A (pt) |
NO (1) | NO20033801L (pt) |
NZ (1) | NZ527991A (pt) |
PL (1) | PL365021A1 (pt) |
PT (1) | PT1401424E (pt) |
RS (1) | RS51056B (pt) |
RU (1) | RU2302240C2 (pt) |
TW (1) | TWI251486B (pt) |
WO (1) | WO2002067927A1 (pt) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU7349301A (en) * | 2000-07-21 | 2002-02-05 | Ortho Mcneil Pharm Inc | Carbamate compounds for use in preventing or treating neuropathic pain and cluster and migraine headache-associated pain |
ATE324107T1 (de) * | 2001-02-27 | 2006-05-15 | Ortho Mcneil Pharm Inc | Carbamat-verbindungen zur prävention oder behandlung von angstzuständen |
PL364680A1 (en) * | 2001-02-27 | 2004-12-13 | Ortho-Mcneil Pharmaceutical, Inc. | Carbamate compounds for use in preventing or treating neurodegenerative disorders |
HUP0401367A2 (hu) | 2001-07-16 | 2004-12-28 | Ortho-Mcneil Pharmaceutical, Inc. | Karbamátvegyületek alkalmazása neuropátiás fájdalom, valamint cluster és migrénes fejfájással társuló fájdalom megelőzésére vagy kezelésére |
WO2005107719A2 (en) * | 2004-05-06 | 2005-11-17 | Sandoz Ag | Pharmaceutical composition comprising hydrophobic drug having improved solubility |
WO2007018496A1 (en) * | 2005-07-26 | 2007-02-15 | Janssen Pharmaceutica, N.V. | Methods for treating substance-related disorders |
EA200970436A1 (ru) * | 2006-10-30 | 2009-12-30 | Янссен Фармацевтика, Н.В. | Соединения карбамата для лечения депрессии |
US20080103199A1 (en) * | 2006-10-31 | 2008-05-01 | Haas Magali | Treatment of pervasive developmental disorders |
US8609849B1 (en) | 2010-11-30 | 2013-12-17 | Fox Chase Chemical Diversity Center, Inc. | Hydroxylated sulfamides exhibiting neuroprotective action and their method of use |
WO2014142477A1 (en) | 2013-03-12 | 2014-09-18 | Bio-Pharm Solutions Co., Ltd. | Phenyl carbamate compounds for use in preventing or treating pediatric epilesy and epilesy-related syndromes |
CN105189451A (zh) * | 2013-03-12 | 2015-12-23 | 比皮艾思药物研发有限公司 | 氨基甲酸苯酯化合物和包含该化合物的用于预防或治疗神经性毒气引起的疾病的组合物 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3313692A (en) * | 1958-04-21 | 1967-04-11 | Armour Pharma | Method of inducing calming and muscle relaxation with carbamates |
US3265728A (en) * | 1962-07-18 | 1966-08-09 | Armour Pharma | Substituted phenethyl carbamates |
US5492930A (en) * | 1994-04-25 | 1996-02-20 | Schering Corporation | Method and formulation for treating CNS disorders |
US5698588A (en) * | 1996-01-16 | 1997-12-16 | Yukong Limited | Halogen substituted carbamate compounds from 2-phenyl-1,2-ethanediol |
-
2002
- 2002-02-21 RU RU2003128983/14A patent/RU2302240C2/ru active
- 2002-02-21 AT AT02707927T patent/ATE346597T1/de active
- 2002-02-21 KR KR1020037011292A patent/KR100886578B1/ko active IP Right Grant
- 2002-02-21 JP JP2002567294A patent/JP4276841B2/ja not_active Expired - Lifetime
- 2002-02-21 DE DE60216457T patent/DE60216457T2/de not_active Expired - Lifetime
- 2002-02-21 WO PCT/US2002/006119 patent/WO2002067927A1/en active IP Right Grant
- 2002-02-21 US US10/081,761 patent/US6541513B2/en not_active Expired - Lifetime
- 2002-02-21 BR BR0207829-5A patent/BR0207829A/pt not_active Application Discontinuation
- 2002-02-21 AU AU2002242296A patent/AU2002242296B2/en not_active Ceased
- 2002-02-21 MX MXPA03007722A patent/MXPA03007722A/es active IP Right Grant
- 2002-02-21 NZ NZ527991A patent/NZ527991A/en unknown
- 2002-02-21 EP EP02707927A patent/EP1401424B1/en not_active Expired - Lifetime
- 2002-02-21 RS YUP-675/03A patent/RS51056B/sr unknown
- 2002-02-21 CN CNB028089235A patent/CN1262271C/zh not_active Expired - Fee Related
- 2002-02-21 HU HU0303342A patent/HUP0303342A3/hu unknown
- 2002-02-21 IL IL15758802A patent/IL157588A0/xx unknown
- 2002-02-21 CZ CZ20032297A patent/CZ302412B6/cs not_active IP Right Cessation
- 2002-02-21 PL PL02365021A patent/PL365021A1/xx unknown
- 2002-02-21 DK DK02707927T patent/DK1401424T3/da active
- 2002-02-21 CA CA2439480A patent/CA2439480C/en not_active Expired - Fee Related
- 2002-02-21 PT PT02707927T patent/PT1401424E/pt unknown
- 2002-02-21 ES ES02707927T patent/ES2275844T3/es not_active Expired - Lifetime
- 2002-02-27 AR ARP020100702A patent/AR032876A1/es unknown
- 2002-03-05 TW TW091103972A patent/TWI251486B/zh not_active IP Right Cessation
-
2003
- 2003-08-26 IL IL157588A patent/IL157588A/en not_active IP Right Cessation
- 2003-08-26 NO NO20033801A patent/NO20033801L/no not_active Application Discontinuation
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B25A | Requested transfer of rights approved |
Free format text: JOHNSON & JOHNSON (US) |
|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |