RU2278112C2 - Производные аминохинолина и аминопиридина и их применение в качестве лигандов аденозина a3 - Google Patents

Производные аминохинолина и аминопиридина и их применение в качестве лигандов аденозина a3 Download PDF

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RU2278112C2
RU2278112C2 RU2003137836/04A RU2003137836A RU2278112C2 RU 2278112 C2 RU2278112 C2 RU 2278112C2 RU 2003137836/04 A RU2003137836/04 A RU 2003137836/04A RU 2003137836 A RU2003137836 A RU 2003137836A RU 2278112 C2 RU2278112 C2 RU 2278112C2
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group
branched
straight
compounds
hydrogen atom
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RU2003137836/04A
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RU2003137836A (ru
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Петер АРАНЬИ (HU)
Петер Араньи
Ласло БАЛАЖ (HU)
Ласло Балаж
Мари БАЛОГ (HU)
Мария Балог
Имре БАТА (HU)
Имре Бата
Шандор БАТОРИ (HU)
Шандор Батори
НАДЬ Лайош Т. (HU)
Надь Лайош Т.
Геза ТИМАРИ (HU)
Геза Тимари
Кинга БОЭР (HU)
Кинга Боэр
Оливье ФИНАНС (FR)
Оливье Финанс
Зольтан КАПУИ (HU)
Зольтан Капуи
Эндре МИКУШ (HU)
Эндре Микуш
Жужанна САМОСВЕЛЬДЬИ (HU)
Жужанна Самосвельдьи
Габор СЕЛЕЦКИ (HU)
Габор Селецки
Каталин УРБАН-САБО (HU)
Каталин Урбан-Сабо
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Санофи-Авентис
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Priority claimed from HU0102279A external-priority patent/HUP0102279A3/hu
Priority claimed from HU0200774A external-priority patent/HUP0200774A2/hu
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Chemical & Material Sciences (AREA)
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  • Pulmonology (AREA)
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
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  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Psychology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
RU2003137836/04A 2001-05-31 2002-05-29 Производные аминохинолина и аминопиридина и их применение в качестве лигандов аденозина a3 RU2278112C2 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
HU0102279A HUP0102279A3 (en) 2001-05-31 2001-05-31 A3 antagonist amino-quinoline-derivatives, process for their preparation, pharmaceutical compositions containing them and their use
HUP0102279 2001-05-31
HUP0200774 2002-03-01
HU0200774A HUP0200774A2 (hu) 2002-03-01 2002-03-01 Amino-piridin és amino-kinolin származékok, eljárás előállításukra, ezeket tartalmazó gyógyszerkészítmények és intermedierjeik

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Publication Number Publication Date
RU2003137836A RU2003137836A (ru) 2005-05-27
RU2278112C2 true RU2278112C2 (ru) 2006-06-20

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US (1) US6969723B2 (enExample)
EP (1) EP1390349B1 (enExample)
JP (1) JP4409935B2 (enExample)
KR (1) KR100745307B1 (enExample)
CN (1) CN1257160C (enExample)
AR (1) AR036074A1 (enExample)
AU (1) AU2002304358B2 (enExample)
BG (1) BG108477A (enExample)
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NZ (1) NZ529966A (enExample)
PL (1) PL366516A1 (enExample)
RS (1) RS95003A (enExample)
RU (1) RU2278112C2 (enExample)
SK (1) SK14142003A3 (enExample)
TN (1) TNSN03117A1 (enExample)
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2489432C2 (ru) * 2007-06-07 2013-08-10 Санофи-Авентис ТРИАЗОЛО[1,5-a]ХИНОЛИНЫ В КАЧЕСТВЕ ЛИГАНДОВ РЕЦЕПТОРА АДЕНОЗИНА А3

Families Citing this family (15)

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HUP0203976A3 (en) * 2002-11-15 2004-08-30 Sanofi Aventis Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them
US8729107B2 (en) * 2002-12-06 2014-05-20 Purdue Research Foundation Pyridines for treating injured mammalian nerve tissue
WO2004052291A2 (en) 2002-12-06 2004-06-24 Purdue Research Foundation Pyridines for treating injured mammalian nerve tissue
RU2317290C2 (ru) * 2003-07-31 2008-02-20 Санофи-Авентис Производные аминохинолина и их применение в качестве лигандов аденозина а3
PL1663982T3 (pl) * 2003-07-31 2008-03-31 Sanofi Aventis Pochodne aminochinoliny i ich zastosowanie jako ligandów adenozyny A3
HUP0400812A2 (en) * 2004-04-19 2006-02-28 Sanofi Aventis Crystalline forms of 2-amino-3-cyano-quinoline derivatives, process for their preparation and pharmaceutical compositions containing them
WO2006040645A1 (en) * 2004-10-11 2006-04-20 Ranbaxy Laboratories Limited N-(3,5-dichloropyridin-4-yl)-2,4,5-alkoxy and 2,3,4-alkoxy benzamide derivatives as pde-iv (phophodiesterase type-iv) inhibitors for the treatment of inflammatory diseases such as asthma
HUP0402371A2 (en) * 2004-11-15 2006-09-28 Sanofi Aventis Novel 125-i-labeled amino-quinoline derivatives
KR100788161B1 (ko) * 2006-01-06 2007-12-21 (주)아모레퍼시픽 벤즈이미다졸 아민 유도체 또는 아미노퀴놀린 유도체를 함유하는 피부 미백용 조성물
KR101106050B1 (ko) * 2009-03-25 2012-01-18 한국과학기술연구원 아미노퀴놀린 화합물, 이의 제조 방법 및 이를 함유하는 의약 조성물
WO2012030918A1 (en) * 2010-09-01 2012-03-08 Ambit Biosciences Corporation Adenosine a3 receptor modulating compounds and methods of use thereof
WO2012166654A1 (en) * 2011-05-27 2012-12-06 The Regents Of The University Of California Cyanoquinoline compounds having activity in correcting mutant-cftr processing and increasing ion transport and uses thereof
CA2754237A1 (en) 2011-05-27 2012-11-27 The Regents Of The University Of California Cyanoquinoline compounds having activity in correcting mutant-cftr processing and increasing ion transport and uses thereof
ES2578363B1 (es) 2015-01-22 2017-01-31 Palobiofarma, S.L. Moduladores de los receptores A3 de adenosina
CN108137547B (zh) 2015-08-03 2021-11-12 百时美施贵宝公司 可用作TNFα调节剂的杂环化合物

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SU1470183A3 (ru) * 1985-05-30 1989-03-30 Рон-Пуленк Санте (Фирма) Способ получени амидных производных хинолина или их солей присоединени кислоты
WO1995011244A1 (en) * 1993-10-22 1995-04-27 Zeneca Limited Pyridazino quinoline compounds
EP1180518A1 (en) * 1999-04-23 2002-02-20 Takeda Chemical Industries, Ltd. 5-pyridyl-1,3-azole compounds, process for producing the same and use thereof

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Patent Citations (3)

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SU1470183A3 (ru) * 1985-05-30 1989-03-30 Рон-Пуленк Санте (Фирма) Способ получени амидных производных хинолина или их солей присоединени кислоты
WO1995011244A1 (en) * 1993-10-22 1995-04-27 Zeneca Limited Pyridazino quinoline compounds
EP1180518A1 (en) * 1999-04-23 2002-02-20 Takeda Chemical Industries, Ltd. 5-pyridyl-1,3-azole compounds, process for producing the same and use thereof

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CHEMICAL ABSTRACTS, vol.116, no.25, 22.06.1992, abstract no.255453f. *

Cited By (1)

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RU2489432C2 (ru) * 2007-06-07 2013-08-10 Санофи-Авентис ТРИАЗОЛО[1,5-a]ХИНОЛИНЫ В КАЧЕСТВЕ ЛИГАНДОВ РЕЦЕПТОРА АДЕНОЗИНА А3

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