RU2016103088A - Фармацевтическое водорастворимое противогрибковое макромолекулярное соединение - Google Patents

Фармацевтическое водорастворимое противогрибковое макромолекулярное соединение Download PDF

Info

Publication number
RU2016103088A
RU2016103088A RU2016103088A RU2016103088A RU2016103088A RU 2016103088 A RU2016103088 A RU 2016103088A RU 2016103088 A RU2016103088 A RU 2016103088A RU 2016103088 A RU2016103088 A RU 2016103088A RU 2016103088 A RU2016103088 A RU 2016103088A
Authority
RU
Russia
Prior art keywords
polyconjugate
amino acid
drug substance
active drug
macromolecular polymer
Prior art date
Application number
RU2016103088A
Other languages
English (en)
Russian (ru)
Inventor
Гуангуи ВЭНЬ
Люйи ВАНЬ
Дунфан ЮЙ
Цзинвэнь ЯН
Хаоцзюнь ВАН
Original Assignee
Бейджин Лэбуорлд Био-Медисин Текнолоджи Корп. Лтд
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Бейджин Лэбуорлд Био-Медисин Текнолоджи Корп. Лтд filed Critical Бейджин Лэбуорлд Био-Медисин Текнолоджи Корп. Лтд
Publication of RU2016103088A publication Critical patent/RU2016103088A/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/61Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule the organic macromolecular compound being a polysaccharide or a derivative thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/62Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
    • A61K47/64Drug-peptide, drug-protein or drug-polyamino acid conjugates, i.e. the modifying agent being a peptide, protein or polyamino acid which is covalently bonded or complexed to a therapeutically active agent
    • A61K47/645Polycationic or polyanionic oligopeptides, polypeptides or polyamino acids, e.g. polylysine, polyarginine, polyglutamic acid or peptide TAT
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
RU2016103088A 2013-07-25 2014-02-08 Фармацевтическое водорастворимое противогрибковое макромолекулярное соединение RU2016103088A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201310315504 2013-07-25
CN201310315504.8 2013-07-25
PCT/CN2014/000146 WO2015010439A1 (zh) 2013-07-25 2014-02-08 药用水溶性抗真菌大分子化合物

Publications (1)

Publication Number Publication Date
RU2016103088A true RU2016103088A (ru) 2017-08-30

Family

ID=51543906

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2016103088A RU2016103088A (ru) 2013-07-25 2014-02-08 Фармацевтическое водорастворимое противогрибковое макромолекулярное соединение

Country Status (10)

Country Link
US (1) US20160158376A1 (enExample)
EP (1) EP3025733A4 (enExample)
JP (1) JP2016525129A (enExample)
KR (1) KR101749004B1 (enExample)
CN (1) CN104055787B (enExample)
AU (1) AU2014295747B2 (enExample)
CA (1) CA2919145A1 (enExample)
HK (1) HK1220629A1 (enExample)
RU (1) RU2016103088A (enExample)
WO (1) WO2015010439A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110669087B (zh) * 2018-07-02 2023-03-31 上海医药工业研究院 两性霉素b肽衍生物及其制备方法
CN110343650B (zh) * 2019-05-28 2020-12-29 浙江工业大学 一种产两性霉素b的重组结节链霉菌及其应用
CN110577921B (zh) * 2019-05-28 2021-04-02 浙江工业大学 产两性霉素b的重组结节链霉菌及其应用
CN112094362B (zh) * 2020-09-29 2022-04-12 四川大学华西医院 烟酰胺核糖或单核苷酸类似物-大分子载体轭合物及制法和应用

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1359473A (en) 1970-11-03 1974-07-10 Prodotti Antibiotici Spa Polyenic antibiotic
AU5858690A (en) * 1989-06-14 1991-01-08 Cetus Corporation Polymer/antibiotic conjugate
US5610264A (en) 1995-11-16 1997-03-11 Calwood Chemical Industries, Inc. Continuous process for polyaspartic acid synthesis
DE10129369C1 (de) * 2001-06-21 2003-03-06 Fresenius Kabi De Gmbh Wasserlösliches, einen Aminozucker aufweisendes Antibiotikum in Form eines Pol ysaccharid-Konjugats
DE10155098A1 (de) * 2001-11-09 2003-05-22 Supramol Parenteral Colloids Mittel zur Prävention von mykotischen Kontaminationen bei der Zell- und Gewebekultur bakteriellen, pflanzlichen, animalischen und humanen Ursprungs, bestehend aus Polyen-Makrolid-Konjugaten mit Polysacchariden
US7261875B2 (en) * 2001-12-21 2007-08-28 Board Of Regents, The University Of Texas System Dendritic poly (amino acid) carriers and methods of use
CA2625426A1 (en) * 2005-09-22 2007-03-29 Hadasit Medical Research Services & Development Limited Dextran and arabinogalactan conjugates of therapeutically active compounds
US20080181852A1 (en) * 2007-01-29 2008-07-31 Nitto Denko Corporation Multi-functional Drug Carriers
CN101333044A (zh) * 2008-05-20 2008-12-31 北京能拓高科技有限公司 箱式组合式污水处理系统
EP2277547A1 (de) * 2009-07-20 2011-01-26 Merck Patent GmbH Epsilon-Polylysin-Konjugate und deren Verwendung
CN101935336B (zh) * 2010-09-01 2014-04-09 北京大学 一类水溶性紫杉烷类药物的制备方法和应用
CA2809934C (en) * 2010-09-02 2018-09-04 Nippon Kayaku Kabushiki Kaisha Process for producing drug-block copolymer composite and pharmaceutical preparation containing same
US8785569B2 (en) * 2011-11-22 2014-07-22 Original Biomedicals Co., Ltd. Drug carrier with chelating complex micelles and the application thereof

Also Published As

Publication number Publication date
KR101749004B1 (ko) 2017-06-19
CN104055787A (zh) 2014-09-24
CN104055787B (zh) 2017-04-26
JP2016525129A (ja) 2016-08-22
CA2919145A1 (en) 2015-01-29
US20160158376A1 (en) 2016-06-09
EP3025733A4 (en) 2017-09-20
EP3025733A1 (en) 2016-06-01
AU2014295747A1 (en) 2016-02-11
HK1220629A1 (en) 2017-05-12
AU2014295747B2 (en) 2016-08-25
WO2015010439A1 (zh) 2015-01-29
KR20160022915A (ko) 2016-03-02

Similar Documents

Publication Publication Date Title
Zhang et al. Pharmacokinetics, biodistribution, efficacy and safety of N-octyl-O-sulfate chitosan micelles loaded with paclitaxel
Van de Ven et al. PLGA nanoparticles and nanosuspensions with amphotericin B: potent in vitro and in vivo alternatives to Fungizone and AmBisome
CN101791411B (zh) 两亲性多糖偶联物及其药物组合物的制备和应用
RU2016103088A (ru) Фармацевтическое водорастворимое противогрибковое макромолекулярное соединение
EP2431403B1 (en) Polymer conjugate of bioactive substance having hydroxy group
Mei et al. Effect of chitosan structure properties and molecular weight on the intranasal absorption of tetramethylpyrazine phosphate in rats
JP2011144207A5 (enExample)
NZ596610A (en) A poorly soluble drug containing microsphere with improved bioavailability and method of preparing the same
WO2010039496A3 (en) Nanocarriers for drug delivery
CN104758255A (zh) 一种姜黄素胶束载药系统及其制备方法
RU2013114993A (ru) Композиция каспофунгина
CN102634033A (zh) 葡聚糖基两亲性嵌段共聚物制备方法
KR20140024833A (ko) 신규한 시티딘계 대사길항제의 고분자 유도체
JP2013537212A5 (enExample)
US9925275B2 (en) Amphotericin B derivatives
CN102908316B (zh) 伊维菌素水溶性固体分散体及其制备方法
Han et al. Synthesis of a new amphiphilic glycodendrimer with antiviral functionality
Chen et al. In vitro and in vivo evaluation of PEG-conjugated ketal-based chitosan micelles as pH-sensitive carriers
WO2009066956A3 (en) Lyophilized pharmaceutical composition with improved reconstitution time containing taxane derivatives and method of manufacturing the same
JP2016525129A5 (enExample)
US20170080098A1 (en) Methods of folding a graft copolymer with dual anticancer drugs and related applications
KR101726728B1 (ko) 고분자 담체 함유 약학 조성물의 유연물질 분석 방법
Dong et al. Assessment of the safety, targeting, and distribution characteristics of a novel pH-sensitive hydrogel
RU2011128540A (ru) Композиции наночастиц
CN103656669A (zh) 基于复合胶束的纳米载体、其制备方法及应用