RU2012104247A - Новые нанокристаллы на основе золота для терапевтического лечения и процессы их электрохимического производства - Google Patents
Новые нанокристаллы на основе золота для терапевтического лечения и процессы их электрохимического производства Download PDFInfo
- Publication number
- RU2012104247A RU2012104247A RU2012104247/15A RU2012104247A RU2012104247A RU 2012104247 A RU2012104247 A RU 2012104247A RU 2012104247/15 A RU2012104247/15 A RU 2012104247/15A RU 2012104247 A RU2012104247 A RU 2012104247A RU 2012104247 A RU2012104247 A RU 2012104247A
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- Prior art keywords
- suspension
- water
- specified
- electrokinetic potential
- nanocrystals
- Prior art date
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- 239000002159 nanocrystal Substances 0.000 title claims abstract 13
- 238000000034 method Methods 0.000 title claims 11
- 230000001225 therapeutic effect Effects 0.000 title 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims abstract 25
- 239000000725 suspension Substances 0.000 claims abstract 23
- 239000000203 mixture Substances 0.000 claims abstract 13
- PCHJSUWPFVWCPO-UHFFFAOYSA-N gold Chemical compound [Au] PCHJSUWPFVWCPO-UHFFFAOYSA-N 0.000 claims abstract 11
- 239000010931 gold Substances 0.000 claims abstract 11
- 229910052737 gold Inorganic materials 0.000 claims abstract 11
- 239000003623 enhancer Substances 0.000 claims abstract 10
- 239000000126 substance Substances 0.000 claims abstract 8
- UIIMBOGNXHQVGW-UHFFFAOYSA-M Sodium bicarbonate Chemical compound [Na+].OC([O-])=O UIIMBOGNXHQVGW-UHFFFAOYSA-M 0.000 claims abstract 4
- 239000002245 particle Substances 0.000 claims abstract 4
- 150000001805 chlorine compounds Chemical class 0.000 claims abstract 2
- 239000007971 pharmaceutical suspension Substances 0.000 claims abstract 2
- 229910000030 sodium bicarbonate Inorganic materials 0.000 claims abstract 2
- 235000017557 sodium bicarbonate Nutrition 0.000 claims abstract 2
- 239000002184 metal Substances 0.000 claims 4
- 229910052751 metal Inorganic materials 0.000 claims 4
- 230000002917 arthritic effect Effects 0.000 claims 2
- 239000002105 nanoparticle Substances 0.000 claims 2
- 208000023275 Autoimmune disease Diseases 0.000 claims 1
- 208000011231 Crohn disease Diseases 0.000 claims 1
- 230000015572 biosynthetic process Effects 0.000 claims 1
- 230000004968 inflammatory condition Effects 0.000 claims 1
- 206010039073 rheumatoid arthritis Diseases 0.000 claims 1
- 238000002560 therapeutic procedure Methods 0.000 claims 1
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Abstract
1. Фармацевтически приемлемая суспензия, содержащаяa. воду фармацевтической степени чистоты;b. по меньшей мере один усилитель обработки иc. нанокристаллы золота, суспендированные в указанной воде, формирующие суспензию, где указанные нанокристаллы золотаi. имеют поверхности, которые содержат по меньшей мере одну характеристику, выбранную из группы характеристик, состоящей из (1) органических химических составляющих, не прилипших или не прикрепленных к указанным поверхностям, и/или (2) являющихся по существу чистыми и не имеющих химических составляющих, прилипших или прикрепленных к поверхностям, отличных от воды или указанного усилителя обработки, которые изменяют функционирование указанных нанокристаллов;ii. имеют моду размера частицы менее приблизительно 50 нм;iii. присутствуют в указанной суспензии в концентрации приблизительно 2-200 м.д.; иd. указанную суспензию, имеющую pH между приблизительно 5 и приблизительно 9,5, электрокинетический потенциал по меньшей мере приблизительно -20 мВ, и суспензия не содержит хлориды.2. Композиция по п.1, где указанный усилитель обработки содержит бикарбонат натрия.3. Композиция по п.1, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -30 мВ.4. Композиция по п.1, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -40 мВ.5. Композиция по п.1, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -50 мВ.6. Фармацевтическая суспензия, содержащаяa. воду фармацевтической степени чистоты, содержащую по меньшей мере один усилитель обработки, имеющую pH между приблизительно 5 и п
Claims (19)
1. Фармацевтически приемлемая суспензия, содержащая
a. воду фармацевтической степени чистоты;
b. по меньшей мере один усилитель обработки и
c. нанокристаллы золота, суспендированные в указанной воде, формирующие суспензию, где указанные нанокристаллы золота
i. имеют поверхности, которые содержат по меньшей мере одну характеристику, выбранную из группы характеристик, состоящей из (1) органических химических составляющих, не прилипших или не прикрепленных к указанным поверхностям, и/или (2) являющихся по существу чистыми и не имеющих химических составляющих, прилипших или прикрепленных к поверхностям, отличных от воды или указанного усилителя обработки, которые изменяют функционирование указанных нанокристаллов;
ii. имеют моду размера частицы менее приблизительно 50 нм;
iii. присутствуют в указанной суспензии в концентрации приблизительно 2-200 м.д.; и
d. указанную суспензию, имеющую pH между приблизительно 5 и приблизительно 9,5, электрокинетический потенциал по меньшей мере приблизительно -20 мВ, и суспензия не содержит хлориды.
2. Композиция по п.1, где указанный усилитель обработки содержит бикарбонат натрия.
3. Композиция по п.1, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -30 мВ.
4. Композиция по п.1, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -40 мВ.
5. Композиция по п.1, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -50 мВ.
6. Фармацевтическая суспензия, содержащая
a. воду фармацевтической степени чистоты, содержащую по меньшей мере один усилитель обработки, имеющую pH между приблизительно 5 и приблизительно 9,5;
b. нанокристаллы золота определенной формы в указанной воде, формирующие указанную суспензию, имеющую электрокинетический потенциал по меньшей мере приблизительно -20 мВ, и где указанные нанокристаллы золота
i. имеют поверхности, которые содержат по меньшей мере одну характеристику, выбранную из группы характеристик, состоящей из (1) органических химических составляющих, не прилипших или не прикрепленных к указанным поверхностям, и/или (2) являющихся по существу чистыми и не имеющих химических составляющих, прилипших или прикрепленных к поверхностям, отличным от воды или указанного усилителя обработки, которые изменяют функционирование указанных нанокристаллов;
ii. имеют моду размера частицы менее приблизительно 50 нм;
iii. присутствуют в указанной суспензии в концентрации приблизительно 2-200 м.д.; и
iv. имеют формы, содержащие пентагональные бипирамиды и тетраэдры в диапазоне приблизительно 15-50%.
7. Композиция по п.6, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -40 мВ.
8. Суспензия, содержащая
a. воду фармацевтической степени чистоты, содержащую по меньшей мере один усилитель обработки, имеющую pH между приблизительно 5 и приблизительно 9,5;
b. нанокристаллы золота в указанной воде, формирующие указанную суспензию, имеющую электрокинетический потенциал по меньшей мере приблизительно -20 мВ, и где указанные нанокристаллы золота
i. имеют поверхности, которые содержат по меньшей мере одну характеристику, выбранную из группы характеристик, состоящей из (1) органических химических составляющих, не прилипших или не прикрепленных к указанным поверхностям, и/или (2) являющихся по существу чистыми и не имеющих химических составляющих, прилипших или прикрепленных к поверхностям, отличных от воды или указанного усилителя обработки, которые изменяют функционирование указанных нанокристаллов;
ii. имеют моду размера частицы менее приблизительно 50 нм;
iii. присутствуют в указанной суспензии в концентрации приблизительно 2-200 м.д.
9. Композиция по п.8, где указанная суспензия имеет электрокинетический потенциал по меньшей мере приблизительно -40 мВ.
10. Способ лечения пациента с артритическим состоянием, включающий введение нуждающемуся в этом пациенту эффективного количества композиции по п.1.
11. Способ по п.10, где артритическим состоянием является ревматоидный артрит.
12. Способ лечения пациента с состоянием, восприимчивым к терапии золотом, включающий введение нуждающемуся в этом пациенту эффективного количества композиции по п.1.
13. Способ по п.12, где состоянием является болезнь Крона.
14. Способ по п.12, где состоянием является боль.
15. Способ по п.12, где состоянием является аутоиммунное заболевание.
16. Способ по п.12, где состоянием является воспалительное состояние.
17. Способ по п.11, где композицию вводят перорально.
18. Способ формирования наночастиц золота, суспендированных в воде:
предоставление по меньшей мере одного усилителя обработки в указанной воде;
предоставление по меньшей мере одного лоткового элемента;
создание направления потока указанной воды через указанный по меньшей мере один лотковый элемент;
предоставление по меньшей мере одного формирующего плазму электрода на основе металла, удаленного от поверхности указанной воды, тем самым формируя пространство между указанным по меньшей мере одним формирующим плазму электродом на основе металла и указанной поверхностью указанной воды;
формирование по меньшей мере одной плазмы в указанном пространстве между указанным по меньшей мере одним формирующим плазму электродом на основе металла и указанной поверхностью указанной воды;
предоставление по меньшей мере одного комплекта электродов, контактирующего с указанной водой, указанный по меньшей мере один комплект электродов контактирует с указанной водой после того, как указанная вода обтекла указанный по меньшей мере один формирующий плазму электрод на основе металла; и
обеспечение реакции указанного по меньшей мере одного комплекта электродов с указанной водой, когда указанная вода контактирует с указанным по меньшей мере одним комплектом электродов, посредством чего в указанной воде формируют указанные наночастицы золота.
19. Продукт, изготовленный способом по п.18.
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