RU2007121705A - Антиинфекционные липопептиды - Google Patents

Антиинфекционные липопептиды Download PDF

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Publication number
RU2007121705A
RU2007121705A RU2007121705/04A RU2007121705A RU2007121705A RU 2007121705 A RU2007121705 A RU 2007121705A RU 2007121705/04 A RU2007121705/04 A RU 2007121705/04A RU 2007121705 A RU2007121705 A RU 2007121705A RU 2007121705 A RU2007121705 A RU 2007121705A
Authority
RU
Russia
Prior art keywords
amino
composition
composition according
compound
protecting group
Prior art date
Application number
RU2007121705/04A
Other languages
English (en)
Russian (ru)
Inventor
Дилан Кристофер АЛЕКСАНДЕР (US)
Дилан Кристофер АЛЕКСАНДЕР
Ричард Х. БАЛЬТЦ (US)
Ричард Х. БАЛЬТЦ
Пол БРАЙАН (US)
Пол БРАЙАН
ГАЛЬ Мари-Франсуаз КЕФФЕ-ЛЕ (US)
ГАЛЬ Мари-Франсуаз КЕФФЕ-ЛЕ
Саша ДЕКЕЛЬ (US)
Саша ДЕКЕЛЬ
Сяовэй ХЭ (US)
Сяовэй ХЭ
Видья КУЛКАРНИ (US)
Видья КУЛКАРНИ
Кристофер ЛЕЙТЕЙЗЕР (US)
Кристофер ЛЕЙТЕЙЗЕР
Вивиан Пак Воон МИАО (CA)
Вивиан Пак Воон МИАО
Киен Трунг НГУЙЕН (US)
Киен Трунг НГУЙЕН
Ян Бэрри ПАРР (US)
Ян Бэрри ПАРР
Дэниел РИТЦ (CH)
Дэниел РИТЦ
Янчжи ЧЖАН (US)
Янчжи ЧЖАН
Original Assignee
Кьюбист Фармасьютикалз
Кьюбист Фармасьютикалз, Инк
Инк (Us)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Кьюбист Фармасьютикалз, Кьюбист Фармасьютикалз, Инк, Инк (Us) filed Critical Кьюбист Фармасьютикалз
Publication of RU2007121705A publication Critical patent/RU2007121705A/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
RU2007121705/04A 2004-11-12 2005-11-11 Антиинфекционные липопептиды RU2007121705A (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US62705604P 2004-11-12 2004-11-12
US60/627,056 2004-11-12
US71070505P 2005-08-23 2005-08-23
US60/710,705 2005-08-23
PCT/US2005/040919 WO2006110185A2 (en) 2004-11-12 2005-11-11 Antiinfective lipopeptides

Publications (1)

Publication Number Publication Date
RU2007121705A true RU2007121705A (ru) 2008-12-20

Family

ID=37087468

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2007121705/04A RU2007121705A (ru) 2004-11-12 2005-11-11 Антиинфекционные липопептиды

Country Status (10)

Country Link
EP (1) EP1814588A2 (pt)
JP (1) JP2008519848A (pt)
KR (1) KR20070086038A (pt)
AU (1) AU2005330517A1 (pt)
BR (1) BRPI0517830A (pt)
CA (1) CA2587848A1 (pt)
IL (1) IL183109A0 (pt)
NO (1) NO20072634L (pt)
RU (1) RU2007121705A (pt)
WO (1) WO2006110185A2 (pt)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2512396C2 (ru) * 2008-12-22 2014-04-10 Кьюбист Фармасьютикалз, Инк. Новые противобактериальные средства для лечения грамположительных инфекций

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2013157188A (ru) * 2011-05-26 2015-07-10 Кьюбист Фармасьютикалз, Инк. Композиции св-183,315 и относящиеся к ним способы
KR101723649B1 (ko) * 2014-10-23 2017-04-06 서울대학교산학협력단 신규한 펩티드 화합물, 이의 생산 방법, 및 이의 용도
CN113061164B (zh) * 2021-03-29 2023-01-10 四川大学 环脂肽类化合物及其在抗类风湿关节炎药物中的应用
WO2023152229A1 (en) * 2022-02-09 2023-08-17 Teitur Trophics Aps Novel peptides

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7408025B2 (en) * 1999-12-15 2008-08-05 Cubist Pharmaceuticals, Inc. Lipopeptides as antibacterial agents
EP1240181A2 (en) * 1999-12-15 2002-09-18 Cubist Pharmaceuticals, Inc. Daptomycin analogs as antibacterial agents
KR20020063230A (ko) * 1999-12-15 2002-08-01 큐비스트 파마슈티컬즈 인코포레이티드 항균제로서의 신규한 리포펩티드
EP1421097A4 (en) * 2001-08-06 2005-07-06 Cubist Pharm Inc COMPOSITIONS AND METHODS RELATING TO THE BIOSYNTHETIC MULTIGENIC FAMILY OF DAPTOMYCIN
NZ531493A (en) * 2001-08-06 2006-03-31 Cubist Pharm Inc Novel depsipeptides and process for preparing same, useful in the treatment of bacterial infection

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2512396C2 (ru) * 2008-12-22 2014-04-10 Кьюбист Фармасьютикалз, Инк. Новые противобактериальные средства для лечения грамположительных инфекций

Also Published As

Publication number Publication date
WO2006110185A2 (en) 2006-10-19
WO2006110185A3 (en) 2007-10-25
IL183109A0 (en) 2008-04-13
JP2008519848A (ja) 2008-06-12
EP1814588A2 (en) 2007-08-08
KR20070086038A (ko) 2007-08-27
CA2587848A1 (en) 2006-10-19
AU2005330517A1 (en) 2006-10-19
BRPI0517830A (pt) 2008-10-21
AU2005330517A2 (en) 2006-10-19
NO20072634L (no) 2007-08-09

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Legal Events

Date Code Title Description
FA92 Acknowledgement of application withdrawn (lack of supplementary materials submitted)

Effective date: 20100310