RU2005138915A - Сульфонамид замещенные имидазохинолины - Google Patents

Сульфонамид замещенные имидазохинолины Download PDF

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Publication number
RU2005138915A
RU2005138915A RU2005138915/04A RU2005138915A RU2005138915A RU 2005138915 A RU2005138915 A RU 2005138915A RU 2005138915/04 A RU2005138915/04 A RU 2005138915/04A RU 2005138915 A RU2005138915 A RU 2005138915A RU 2005138915 A RU2005138915 A RU 2005138915A
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RU
Russia
Prior art keywords
animal
substance
effective amount
salt according
imidazochinolins
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RU2005138915/04A
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English (en)
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RU2374246C2 (ru
Inventor
Джордж В. ГРИЕСГРАБЕР (US)
Джордж В. ГРИЕСГРАБЕР
Original Assignee
3М Инновейтив Пропертиз Компани (US)
3М Инновейтив Пропертиз Компани
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Publication of RU2005138915A publication Critical patent/RU2005138915A/ru
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Publication of RU2374246C2 publication Critical patent/RU2374246C2/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Claims (5)

1. N-{2-[4-амино-2-(этоксиметил)-1H-имидазо-[4,5-c]-хинолин-1-ил]-1,1-диметилэтил}-метансульфонамид или фармацевтически приемлемая соль этого вещества.
2. Фармацевтическая композиция, содержащая терапевтически эффективное количество вещества или его соль по п.1 и фармацевтически приемлемый носитель.
3. Способ индукции биосинтеза цитокинов в организме животного, включающий введение эффективного количества вещества или его соли по п.1 в организм животного.
4. Способ лечения вирусного заболевания у животного, включающий введение эффективного количества вещества или его соли по п.1 в организм животного.
5. Способ лечения онкологического заболевания у животного, включающий введение эффективного количества вещества или его соли по п.1 в организм животного.
RU2005138915/04A 2003-06-27 2004-06-25 N-{2-[4-АМИНО-2-(ЭТОКСИМЕТИЛ)-1Н-ИМИДАЗО-[4,5-с]-ХИНОЛИН-1-ИЛ]-1,1-ДИМЕТИЛЭТИЛ}-МЕТАНСУЛЬФОНАМИД И ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ НА ЕГО ОСНОВЕ RU2374246C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48320003P 2003-06-27 2003-06-27
US60/483,200 2003-06-27

Publications (2)

Publication Number Publication Date
RU2005138915A true RU2005138915A (ru) 2006-06-27
RU2374246C2 RU2374246C2 (ru) 2009-11-27

Family

ID=33563911

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2005138915/04A RU2374246C2 (ru) 2003-06-27 2004-06-25 N-{2-[4-АМИНО-2-(ЭТОКСИМЕТИЛ)-1Н-ИМИДАЗО-[4,5-с]-ХИНОЛИН-1-ИЛ]-1,1-ДИМЕТИЛЭТИЛ}-МЕТАНСУЛЬФОНАМИД И ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ НА ЕГО ОСНОВЕ

Country Status (16)

Country Link
EP (1) EP1638566A4 (ru)
JP (1) JP2007521280A (ru)
KR (1) KR20060035637A (ru)
CN (1) CN1812789B (ru)
AR (2) AR044923A1 (ru)
AU (1) AU2004253929A1 (ru)
BR (1) BRPI0411916A (ru)
CA (1) CA2529322A1 (ru)
IL (1) IL172427A0 (ru)
MX (1) MXPA06000144A (ru)
MY (1) MY157827A (ru)
NZ (1) NZ544330A (ru)
RU (1) RU2374246C2 (ru)
TW (2) TW200511992A (ru)
WO (2) WO2005003064A2 (ru)
ZA (1) ZA200600769B (ru)

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KR101154101B1 (ko) 2003-10-03 2012-06-11 쓰리엠 이노베이티브 프로퍼티즈 컴파니 알콕시 치환된 이미다조퀴놀린
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Also Published As

Publication number Publication date
CN1812789A (zh) 2006-08-02
CN1812789B (zh) 2010-07-14
JP2007521280A (ja) 2007-08-02
AU2004253929A1 (en) 2005-01-13
EP1638566A4 (en) 2009-03-25
CA2529322A1 (en) 2005-01-13
WO2005003065A3 (en) 2005-03-10
RU2374246C2 (ru) 2009-11-27
WO2005003064A2 (en) 2005-01-13
WO2005003065A2 (en) 2005-01-13
AR044922A1 (es) 2005-10-12
ZA200600769B (en) 2007-05-30
AR044923A1 (es) 2005-10-12
MXPA06000144A (es) 2006-04-07
KR20060035637A (ko) 2006-04-26
MY157827A (en) 2016-07-29
TW200514784A (en) 2005-05-01
BRPI0411916A (pt) 2006-08-15
NZ544330A (en) 2009-06-26
IL172427A0 (en) 2006-04-10
WO2005003064A3 (en) 2005-03-31
TW200511992A (en) 2005-04-01
EP1638566A2 (en) 2006-03-29

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