RS51117B - Lekovi za alchajmerovu bolest - Google Patents
Lekovi za alchajmerovu bolestInfo
- Publication number
- RS51117B RS51117B RSP-2009/0363A RSP20090363A RS51117B RS 51117 B RS51117 B RS 51117B RS P20090363 A RSP20090363 A RS P20090363A RS 51117 B RS51117 B RS 51117B
- Authority
- RS
- Serbia
- Prior art keywords
- sub
- moiety
- group
- acid derivatives
- alzheimer
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Indole Compounds (AREA)
Abstract
Jedinjenje opšte formule-I:gde R predstavlja nesteroidni i antiinflamatorni deo molekula koji je odabran ili od:i) indometacina iliii) od derivata propionske kiseline koji je sadržan u naproksenu, ibuprofenu ili ketoprofenu gde A predstavlja CHOH grupu ili CH2 grupu ili (CH2)2 grupudok Y predstavlja:i) antioksidativni deo molekula koji je odabran od cistamina ili cistein etil estra iliii) neuroprotektivnog dela molekula 2-piridin-3-il-alkanol iliiii) NGF-indukujućeg dela molekula 2-metoksi-4-metilfenola.Prijava sadrži još 13 patentnih zahteva.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/GR2005/000005 WO2006090192A1 (en) | 2005-02-28 | 2005-02-28 | Medicaments for alzheimer |
Publications (1)
Publication Number | Publication Date |
---|---|
RS51117B true RS51117B (sr) | 2010-10-31 |
Family
ID=35044605
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RSP-2009/0363A RS51117B (sr) | 2005-02-28 | 2005-02-28 | Lekovi za alchajmerovu bolest |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP1856102B1 (sr) |
AT (1) | ATE433970T1 (sr) |
CY (1) | CY1109317T1 (sr) |
DE (1) | DE602005015033D1 (sr) |
DK (1) | DK1856102T3 (sr) |
ES (1) | ES2328938T3 (sr) |
HR (1) | HRP20090448T1 (sr) |
PL (1) | PL1856102T3 (sr) |
PT (1) | PT1856102E (sr) |
RS (1) | RS51117B (sr) |
SI (1) | SI1856102T1 (sr) |
WO (1) | WO2006090192A1 (sr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2008067451A1 (en) * | 2006-11-30 | 2008-06-05 | Itherx Pharmaceuticals, Inc. | Novel 3-benzylidine and 3-benzyl substituted chromanones |
US9085555B2 (en) | 2011-01-04 | 2015-07-21 | Novartis Ag | Complement pathway modulators and uses thereof |
CN105121429B (zh) | 2012-06-28 | 2017-12-12 | 诺华股份有限公司 | 补体途径调节剂和其用途 |
US9388199B2 (en) | 2012-06-28 | 2016-07-12 | Novartis Ag | Pyrrolidine derivatives and their use as complement pathway modulators |
EP2867227B1 (en) | 2012-06-28 | 2018-11-21 | Novartis AG | Complement pathway modulators and uses thereof |
EP2867229B1 (en) | 2012-06-28 | 2017-07-26 | Novartis AG | Pyrrolidine derivatives and their use as complement pathway modulators |
CN104619698B (zh) | 2012-06-28 | 2016-08-31 | 诺华股份有限公司 | 吡咯烷衍生物及其作为补体途径调节剂的用途 |
EP2872503B1 (en) | 2012-07-12 | 2018-06-20 | Novartis AG | Complement pathway modulators and uses thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4123544A (en) * | 1977-03-02 | 1978-10-31 | Merrell Toraude S. A. | Acetylsalicylic acid derivatives |
NZ228329A (en) * | 1988-03-18 | 1991-12-23 | Mitsui Toatsu Chemicals | Catechol derivatives and pharmaceutical compositions thereof |
FR2669029B1 (fr) * | 1990-11-14 | 1994-09-02 | Adir | Nouveaux derives de la n-benzoyl proline, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
-
2005
- 2005-02-28 RS RSP-2009/0363A patent/RS51117B/sr unknown
- 2005-02-28 AT AT05708486T patent/ATE433970T1/de active
- 2005-02-28 PT PT05708486T patent/PT1856102E/pt unknown
- 2005-02-28 SI SI200530782T patent/SI1856102T1/sl unknown
- 2005-02-28 DE DE602005015033T patent/DE602005015033D1/de active Active
- 2005-02-28 ES ES05708486T patent/ES2328938T3/es active Active
- 2005-02-28 WO PCT/GR2005/000005 patent/WO2006090192A1/en active Application Filing
- 2005-02-28 PL PL05708486T patent/PL1856102T3/pl unknown
- 2005-02-28 DK DK05708486T patent/DK1856102T3/da active
- 2005-02-28 EP EP05708486A patent/EP1856102B1/en active Active
-
2009
- 2009-08-14 CY CY20091100875T patent/CY1109317T1/el unknown
- 2009-08-21 HR HR20090448T patent/HRP20090448T1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
DK1856102T3 (da) | 2009-08-31 |
WO2006090192A1 (en) | 2006-08-31 |
PL1856102T3 (pl) | 2009-11-30 |
HRP20090448T1 (en) | 2009-09-30 |
SI1856102T1 (sl) | 2009-12-31 |
DE602005015033D1 (de) | 2009-07-30 |
EP1856102B1 (en) | 2009-06-17 |
EP1856102A1 (en) | 2007-11-21 |
PT1856102E (pt) | 2009-08-24 |
ES2328938T3 (es) | 2009-11-19 |
CY1109317T1 (el) | 2014-07-02 |
ATE433970T1 (de) | 2009-07-15 |
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