RO117375B1 - Derivaţi amidici n-sulfonil şi n-sulfinil de a-aminoacizi, procedee pentru prepararea acestora, compoziţie microbicidă şi metodă de control şi prevenire a infestării plantelor - Google Patents

Derivaţi amidici n-sulfonil şi n-sulfinil de a-aminoacizi, procedee pentru prepararea acestora, compoziţie microbicidă şi metodă de control şi prevenire a infestării plantelor

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Publication number
RO117375B1
RO117375B1 RO96-02074A RO9602074A RO117375B1 RO 117375 B1 RO117375 B1 RO 117375B1 RO 9602074 A RO9602074 A RO 9602074A RO 117375 B1 RO117375 B1 RO 117375B1
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RO
Romania
Prior art keywords
alkyl
alpha
alkylthio
cycloalkyl
alkoxy
Prior art date
Application number
RO96-02074A
Other languages
English (en)
Inventor
Martin Zeller
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of RO117375B1 publication Critical patent/RO117375B1/ro

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C307/04—Diamides of sulfuric acids
    • C07C307/06—Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/07—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/11—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/14—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C313/02—Sulfinic acids; Derivatives thereof
    • C07C313/06—Sulfinamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C313/08—Sulfenic acids; Derivatives thereof
    • C07C313/18—Sulfenamides
    • C07C313/20—Sulfenamides having sulfur atoms of sulfenamide groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/02—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms
    • C07C317/04—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Invenţia se referă la derivaţi amidici de alfa-aminoacizi cu activitate microbicidă, cu formula generală (I):în care n este 0 sau 1; Reste alchil C-C, care este nesubstituit sau care poate să fie substituit cu alcoxi C-C, tioalchil C-C, sulfonilalchil C-C, cicloalchil C- C, ciano, alcoxicarbonil C-C, alcheniloxicarbonil C-Csau alchiniloxicarbonil C-C; cicloalchil C-C, alchenil C-C; alchinil C-C, halogenoalchil C-Csau o grupare NRR, în care Rsi R, în mod independent unul de celălalt, sunt hidrogen sau alchil C-Csau împreună sunt tetra- sau penta- metilen; Rşi Rîn mod independent, unul faţă de celălalt, sunt hidrogen; alchil C-C; alchil C-Ccare este substituit cu hidroxil, alcoxi C-Cmercapto sau tioalchil C-C; alchenil C-C; alchinil C-C; cicloalchil C-Csau cicloalchil C-C, alchil C-Csau în care cele două grupări Rşi R, împreună cu atomul de carbon la care sunt legate, formează un inel carbociclic cu trei până la opt membri; Reste hidrogen sau alchil C-C; Reste hidrogen; alchilC-Csau fenil, care este nesubstituit sau poate fi substituit cu halogen, nitro, alchil C-C, halogenalchil C-C, alcoxi C-Csau tioalchil C-C; şi Reste o rupare G:în care Rşi Rsunt, independent unul faţă de celălalt, hidrogen sau alchil C-C; p este 0 sau 1; şi R, Rşi Rsunt în mod independent, unul faţă de celălalt, hidrogen, alchil C-C, halogenoalchil C-C, alchenil C-C, alchinil C-C, alcoxi C-C, alcheniloxi C-C, alchiniloxi C-C, tioalchil C-Chalogen sau nitro.
RO96-02074A 1994-05-04 1995-04-22 Derivaţi amidici n-sulfonil şi n-sulfinil de a-aminoacizi, procedee pentru prepararea acestora, compoziţie microbicidă şi metodă de control şi prevenire a infestării plantelor RO117375B1 (ro)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH140794 1994-05-04
CH58495 1995-03-01
PCT/EP1995/001530 WO1995030651A1 (en) 1994-05-04 1995-04-22 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides

Publications (1)

Publication Number Publication Date
RO117375B1 true RO117375B1 (ro) 2002-02-28

Family

ID=25685033

Family Applications (1)

Application Number Title Priority Date Filing Date
RO96-02074A RO117375B1 (ro) 1994-05-04 1995-04-22 Derivaţi amidici n-sulfonil şi n-sulfinil de a-aminoacizi, procedee pentru prepararea acestora, compoziţie microbicidă şi metodă de control şi prevenire a infestării plantelor

Country Status (24)

Country Link
US (2) US5585519A (ro)
EP (1) EP0758317B1 (ro)
JP (1) JPH10504522A (ro)
KR (1) KR100358813B1 (ro)
CN (1) CN1064957C (ro)
AT (1) ATE178593T1 (ro)
AU (1) AU683382B2 (ro)
BG (1) BG63337B1 (ro)
BR (1) BR9507703A (ro)
CA (1) CA2186510A1 (ro)
CZ (1) CZ289778B6 (ro)
DE (1) DE69508932T2 (ro)
DK (1) DK0758317T3 (ro)
ES (1) ES2132662T3 (ro)
GR (1) GR3030368T3 (ro)
HU (1) HU216747B (ro)
IL (1) IL113577A0 (ro)
MX (1) MX9605333A (ro)
NZ (1) NZ284812A (ro)
PL (1) PL178747B1 (ro)
RO (1) RO117375B1 (ro)
RU (1) RU2140411C1 (ro)
SK (1) SK280607B6 (ro)
WO (1) WO1995030651A1 (ro)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU705463B2 (en) * 1995-10-18 1999-05-20 Novartis Ag N-sulphonyl and N-sulphinyl amino acid derivatives as microbicides
BR9807508A (pt) † 1997-01-23 2000-03-21 Hoffmann La Roche Inibidores de sulfamida da metaloprotease
GB9702194D0 (en) * 1997-02-04 1997-03-26 Lilly Co Eli Sulphonide derivatives
DE69808256T2 (de) * 1997-02-25 2003-05-28 Syngenta Participations Ag, Basel Als mikrobizide mittel verwendbare n-sulfonyl- und n-sulfinyl-aminosäureamide
PT968178E (pt) 1997-02-25 2002-11-29 Syngenta Participations Ag N-sulfonil e n-sulfinil amidas de aminoacidos como microbicidas
EP1034163A1 (en) * 1997-05-07 2000-09-13 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Berlin New cysteine derivatives, processes for their production, and pharmaceuticals containing them
GT199800109A (es) 1997-08-06 2000-01-13 Derivados de n-sulfonilglicinalquiniloxifenetilamida microbicidas.
GB9804265D0 (en) * 1998-02-27 1998-04-22 Ciba Geigy Ag Organic compounds
US6176155B1 (en) 1998-09-18 2001-01-23 Schleuniger Holding Ag Semi-automatic wire processing apparatus
GB9826649D0 (en) 1998-12-03 1999-01-27 Novartis Ag Organic compounds
TW564244B (en) * 1999-01-11 2003-12-01 Novartis Ag Novel propargylether derivatives
GB0009055D0 (en) * 2000-04-13 2000-05-31 Novartis Ag Organic compounds
GB0009053D0 (en) * 2000-04-13 2000-05-31 Novartis Ag Organic compounds
GB0009054D0 (en) 2000-04-13 2000-05-31 Novartis Ag Organic compounds
GB0011944D0 (en) * 2000-05-17 2000-07-05 Novartis Ag Organic compounds
GB0022338D0 (en) * 2000-09-12 2000-10-25 Novartis Ag Organic Compounds
GB0115602D0 (en) * 2001-06-26 2001-08-15 Syngenta Participations Ag Organic compounds
GB0127556D0 (en) 2001-11-16 2002-01-09 Syngenta Participations Ag Organic compounds
GB0223665D0 (en) * 2002-10-10 2002-11-20 Syngenta Participations Ag Organic compounds
US7868206B2 (en) 2005-12-27 2011-01-11 National University Corporation, Gunma University Trihalomethionine derivative and pharmaceutical product containing the same
EP1939157A1 (en) 2006-12-22 2008-07-02 Tradecorp, S. A. New products for the treatment of the iron chlorosis
CN112939825B (zh) * 2021-02-22 2022-07-19 浙江理工大学 一种亚磺酰胺化合物及其制备方法与应用

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Publication number Priority date Publication date Assignee Title
CA2012306A1 (en) * 1989-03-28 1990-09-28 Werner Neidhart Amino acid derivatives
JP2701932B2 (ja) * 1989-04-10 1998-01-21 サントリー株式会社 タンパク質分解酵素阻害剤
DE3915755A1 (de) * 1989-05-13 1990-11-29 Bayer Ag Fungizide mittel sowie substituierte aminosaeureamid-derivate und deren herstellung
DE3936298A1 (de) * 1989-11-01 1991-05-02 Bayer Ag Substituierte aminosaeureamid-derivate deren herstellung und verwendung
DE4026966A1 (de) * 1990-08-25 1992-02-27 Bayer Ag Substituierte valinamid-derivate
US5371267A (en) * 1990-09-22 1994-12-06 Bayer Aktiengesellschaft Substituted amino acid amide derivatives their preparation and use
US5254715A (en) * 1990-11-07 1993-10-19 Warner-Lambert Company Aminosulfonyl carbamates
US5155136A (en) * 1990-11-23 1992-10-13 Eastman Kodak Company Fungicidal, 2-acylacetanilide derivatives
EP0493683A1 (en) * 1990-12-20 1992-07-08 American Cyanamid Company Fungicidal amino acid amides
DE4102042A1 (de) * 1991-01-24 1992-07-30 Bayer Ag Substituierte aminosaeureamid-derivate deren herstellung und verwendung als fungizide
DE4203084A1 (de) * 1992-02-04 1993-08-05 Bayer Ag Substituierte aminosaeureamide

Also Published As

Publication number Publication date
MX9605333A (es) 1997-12-31
WO1995030651A1 (en) 1995-11-16
DE69508932D1 (de) 1999-05-12
BG101003A (en) 1997-08-29
DK0758317T3 (da) 1999-10-18
RU2140411C1 (ru) 1999-10-27
AU683382B2 (en) 1997-11-06
ES2132662T3 (es) 1999-08-16
CN1147247A (zh) 1997-04-09
CZ289778B6 (cs) 2002-04-17
PL178747B1 (pl) 2000-06-30
CZ319896A3 (en) 1997-02-12
KR970702847A (ko) 1997-06-10
CN1064957C (zh) 2001-04-25
HUT75049A (en) 1997-03-28
HU9603026D0 (en) 1997-01-28
JPH10504522A (ja) 1998-05-06
BR9507703A (pt) 1997-08-19
EP0758317B1 (en) 1999-04-07
ATE178593T1 (de) 1999-04-15
EP0758317A1 (en) 1997-02-19
PL316660A1 (en) 1997-02-03
NZ284812A (en) 1998-06-26
IL113577A0 (en) 1995-08-31
CA2186510A1 (en) 1995-11-16
DE69508932T2 (de) 1999-09-30
HU216747B (hu) 1999-08-30
US5728875A (en) 1998-03-17
US5585519A (en) 1996-12-17
GR3030368T3 (en) 1999-09-30
KR100358813B1 (ko) 2003-02-11
AU2345895A (en) 1995-11-29
SK141996A3 (en) 1997-05-07
SK280607B6 (sk) 2000-05-16
BG63337B1 (bg) 2001-10-31

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