PT99091A - Processo para a preparacao de composicoes farmaceuticas contendo derivados da triazina e da pirimidina, como ingredientes activos, destinadas a reverter a resistencia aos agentes anticancerosos e antimalaricos - Google Patents

Processo para a preparacao de composicoes farmaceuticas contendo derivados da triazina e da pirimidina, como ingredientes activos, destinadas a reverter a resistencia aos agentes anticancerosos e antimalaricos

Info

Publication number
PT99091A
PT99091A PT99091A PT9909191A PT99091A PT 99091 A PT99091 A PT 99091A PT 99091 A PT99091 A PT 99091A PT 9909191 A PT9909191 A PT 9909191A PT 99091 A PT99091 A PT 99091A
Authority
PT
Portugal
Prior art keywords
resistance
agents
anticanceros
antimalaric
revert
Prior art date
Application number
PT99091A
Other languages
English (en)
Other versions
PT99091B (pt
Inventor
Alain Pierre
Gilbert Regnier
Ghanem Atassi
Alain Dhainaut
Bernard Paramelle
Xavier Leverve
Original Assignee
Adir
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adir filed Critical Adir
Publication of PT99091A publication Critical patent/PT99091A/pt
Publication of PT99091B publication Critical patent/PT99091B/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT99091A 1990-09-27 1991-09-26 Processo para a preparacao de composicoes farmaceuticas contendo derivados da triazina e da pirimidina, como ingredientes activos, destinadas a reverter a resistencia aos agentes anticancerosos e antimalaricos PT99091B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9011887A FR2667243B1 (fr) 1990-09-27 1990-09-27 Utilisation de s derives de la triazine et de la pyrimidine pour l'obtention de medicaments reversant la resistance aux agents anticancereux et antimalariques.

Publications (2)

Publication Number Publication Date
PT99091A true PT99091A (pt) 1992-08-31
PT99091B PT99091B (pt) 1999-02-26

Family

ID=9400676

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99091A PT99091B (pt) 1990-09-27 1991-09-26 Processo para a preparacao de composicoes farmaceuticas contendo derivados da triazina e da pirimidina, como ingredientes activos, destinadas a reverter a resistencia aos agentes anticancerosos e antimalaricos

Country Status (14)

Country Link
US (1) US5225405A (pt)
EP (1) EP0478416B1 (pt)
JP (1) JPH0761943B2 (pt)
AT (1) ATE100711T1 (pt)
AU (1) AU648584B2 (pt)
CA (1) CA2052441A1 (pt)
DE (1) DE69101097T2 (pt)
DK (1) DK0478416T3 (pt)
ES (1) ES2062724T3 (pt)
FR (1) FR2667243B1 (pt)
IE (1) IE65594B1 (pt)
NZ (1) NZ239953A (pt)
PT (1) PT99091B (pt)
ZA (1) ZA917699B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996032945A1 (fr) * 1995-04-20 1996-10-24 Nippon Shinyaku Co., Ltd. Inhibiteur de neovascularisation
PT860170E (pt) 1996-08-13 2000-06-30 Kyowa Hakko Kogyo Kk Comprimidos a base de ureia marcada com isotopos
US6335339B1 (en) 1998-01-13 2002-01-01 Scriptgen Pharmaceuticals, Inc. Triazine antiviral compounds
US6376514B1 (en) * 2000-10-17 2002-04-23 The Procter & Gamble Co. Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof
US6693099B2 (en) 2000-10-17 2004-02-17 The Procter & Gamble Company Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
SG11202000331YA (en) * 2017-07-13 2020-02-27 Michael David Forrest Therapeutic modulators of the reverse mode of atp synthase

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1256513A (pt) * 1968-10-02 1971-12-08
FR2521560A1 (fr) * 1982-02-17 1983-08-19 Adir Nouveaux derives de piperazine et d'homopiperazine, leurs procedes de preparation et les compositions pharmaceutiques les renfermant
FR2524467A1 (fr) * 1982-03-30 1983-10-07 Adir Polymethylene-imines disubstituees, leurs procedes de preparation et les compositions pharmaceutiques les renfermant
FR2525597B1 (fr) * 1982-04-21 1985-06-07 Adir Polymethylene diamines n,n'-substituees, leurs procedes de preparation et les compositions pharmaceutiques les renfermant
FR2544315B1 (fr) * 1983-04-12 1985-07-05 Adir Polymethylene imines disubstituees, leurs procedes de preparation, et les compositions pharmaceutiques les renfermant

Also Published As

Publication number Publication date
ZA917699B (en) 1992-06-24
JPH0761943B2 (ja) 1995-07-05
FR2667243A1 (fr) 1992-04-03
EP0478416B1 (fr) 1994-01-26
DK0478416T3 (da) 1994-05-02
US5225405A (en) 1993-07-06
DE69101097D1 (de) 1994-03-10
ATE100711T1 (de) 1994-02-15
PT99091B (pt) 1999-02-26
AU8475291A (en) 1992-04-02
EP0478416A1 (fr) 1992-04-01
ES2062724T3 (es) 1994-12-16
DE69101097T2 (de) 1994-08-04
IE65594B1 (en) 1995-11-01
NZ239953A (en) 1997-06-24
CA2052441A1 (fr) 1992-03-28
AU648584B2 (en) 1994-04-28
IE913375A1 (en) 1992-04-08
JPH0672878A (ja) 1994-03-15
FR2667243B1 (fr) 1994-11-04

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BB1A Laying open of patent application

Effective date: 19920407

FG3A Patent granted, date of granting

Effective date: 19981123

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20000531