ATE3769T1 - 1-imidazol-2-yliden-3-thienyl-harnstoffderivate verfahren zu deren herstellung und pharmazeutische zusammensetzungen. - Google Patents
1-imidazol-2-yliden-3-thienyl-harnstoffderivate verfahren zu deren herstellung und pharmazeutische zusammensetzungen.Info
- Publication number
- ATE3769T1 ATE3769T1 AT79302921T AT79302921T ATE3769T1 AT E3769 T1 ATE3769 T1 AT E3769T1 AT 79302921 T AT79302921 T AT 79302921T AT 79302921 T AT79302921 T AT 79302921T AT E3769 T1 ATE3769 T1 AT E3769T1
- Authority
- AT
- Austria
- Prior art keywords
- processes
- pharmaceutical compositions
- ylidene
- imidazole
- preparation
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- FKVFQJHVQSGXMN-UHFFFAOYSA-N (1-imidazol-2-ylidenethiophen-3-yl)urea Chemical class C1=CC(NC(=O)N)=CS1=C1N=CC=N1 FKVFQJHVQSGXMN-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- 230000009858 acid secretion Effects 0.000 abstract 1
- 230000000949 anxiolytic effect Effects 0.000 abstract 1
- 239000003085 diluting agent Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
- 125000001544 thienyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Anesthesiology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/004,675 US4230713A (en) | 1979-01-19 | 1979-01-19 | Heterocyclic tetrahydro-1-alkyl-4-oxo-1H-imidazol-2-ylidene urea and phenyl esters of tetrahydro-1-alkyl-4-oxo-1H-imidazol-2-ylidene carbamic acid compounds |
| EP79302921A EP0013817B1 (de) | 1979-01-19 | 1979-12-17 | 1-Imidazol-2-yliden-3-thienyl-harnstoffderivate, Verfahren zu deren Herstellung und pharmazeutische Zusammensetzungen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE3769T1 true ATE3769T1 (de) | 1983-06-15 |
Family
ID=21711951
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT79302921T ATE3769T1 (de) | 1979-01-19 | 1979-12-17 | 1-imidazol-2-yliden-3-thienyl-harnstoffderivate verfahren zu deren herstellung und pharmazeutische zusammensetzungen. |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US4230713A (de) |
| EP (1) | EP0013817B1 (de) |
| JP (1) | JPS55100380A (de) |
| AT (1) | ATE3769T1 (de) |
| CA (1) | CA1122600A (de) |
| DE (1) | DE2965701D1 (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4472583A (en) * | 1980-02-05 | 1984-09-18 | The Dow Chemical Company | 4-Isothiocyanato-2,6-bis-(trifluoromethyl)pyridine |
| DE3674054D1 (de) * | 1985-04-26 | 1990-10-18 | Hoffmann La Roche | 1,3-disubstituierte imidazoliumsalze. |
| US4657922A (en) * | 1985-05-24 | 1987-04-14 | Mcneilab, Inc. | Anxiolytic 4,5-dihydro-4-oxo-1H-imidazol-2-yl urea derivatives |
| DE59805833D1 (de) | 1997-07-22 | 2002-11-07 | Basf Coatings Ag | Beschichtungsmittel und verfahren zu dessen herstellung |
| US20030220646A1 (en) * | 2002-05-23 | 2003-11-27 | Thelen Sarah L. | Method and apparatus for reducing femoral fractures |
| WO2007073283A1 (en) * | 2005-12-20 | 2007-06-28 | Astrazeneca Ab | Substituted cinnoline derivatives as gabaa-receptor modulators and method for their synthesis |
| US7465795B2 (en) * | 2005-12-20 | 2008-12-16 | Astrazeneca Ab | Compounds and uses thereof |
| AR067028A1 (es) * | 2007-06-19 | 2009-09-30 | Astrazeneca Ab | Compuestos y usos de los mismos 849 |
| MA53096A (fr) * | 2018-07-03 | 2021-05-12 | Ifm Due Inc | Composés et compositions destinés au traitement d'états pathologiques associés à une activité de sting |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3983135A (en) * | 1974-09-23 | 1976-09-28 | Mcneil Laboratories, Incorporated | 4-Oxo-2-imidazolidinylidene ureas |
-
1979
- 1979-01-19 US US06/004,675 patent/US4230713A/en not_active Expired - Lifetime
- 1979-12-07 CA CA341,498A patent/CA1122600A/en not_active Expired
- 1979-12-17 AT AT79302921T patent/ATE3769T1/de not_active IP Right Cessation
- 1979-12-17 DE DE7979302921T patent/DE2965701D1/de not_active Expired
- 1979-12-17 EP EP79302921A patent/EP0013817B1/de not_active Expired
-
1980
- 1980-01-18 JP JP375680A patent/JPS55100380A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| DE2965701D1 (en) | 1983-07-21 |
| JPS55100380A (en) | 1980-07-31 |
| CA1122600A (en) | 1982-04-27 |
| EP0013817B1 (de) | 1983-06-15 |
| US4230713A (en) | 1980-10-28 |
| EP0013817A1 (de) | 1980-08-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |