PT974598E - Novos derivados da eritromicina, seu processo de preparação e sua aplicação como medicamentos - Google Patents

Novos derivados da eritromicina, seu processo de preparação e sua aplicação como medicamentos Download PDF

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Publication number
PT974598E
PT974598E PT99401706T PT99401706T PT974598E PT 974598 E PT974598 E PT 974598E PT 99401706 T PT99401706 T PT 99401706T PT 99401706 T PT99401706 T PT 99401706T PT 974598 E PT974598 E PT 974598E
Authority
PT
Portugal
Prior art keywords
radical
methyl
formula
compounds
dideoxy
Prior art date
Application number
PT99401706T
Other languages
English (en)
Portuguese (pt)
Inventor
Alexis Denis
Giuseppe Gigliotti
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9808795A external-priority patent/FR2780977B1/fr
Priority claimed from FR9905245A external-priority patent/FR2792637B1/fr
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of PT974598E publication Critical patent/PT974598E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
PT99401706T 1998-07-09 1999-07-08 Novos derivados da eritromicina, seu processo de preparação e sua aplicação como medicamentos PT974598E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9808795A FR2780977B1 (fr) 1998-07-09 1998-07-09 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR9905245A FR2792637B1 (fr) 1999-04-26 1999-04-26 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
PT974598E true PT974598E (pt) 2011-11-23

Family

ID=26234434

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99401706T PT974598E (pt) 1998-07-09 1999-07-08 Novos derivados da eritromicina, seu processo de preparação e sua aplicação como medicamentos

Country Status (8)

Country Link
US (1) US6433151B1 (enExample)
EP (1) EP0974598B1 (enExample)
JP (1) JP4573925B2 (enExample)
AT (1) ATE521619T1 (enExample)
CY (1) CY1112087T1 (enExample)
DK (1) DK0974598T3 (enExample)
ES (1) ES2372156T3 (enExample)
PT (1) PT974598E (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2273964T3 (es) * 1998-12-10 2007-05-16 Pfizer Products Inc. Antibioticos de carbamato y carbazato cetolida.
EP1794171A2 (en) * 2004-07-28 2007-06-13 Ranbaxy Laboratories, Ltd. Ketolide derivatives as antibacterial agents
EP1812455A2 (en) * 2004-09-27 2007-08-01 Ranbaxy Laboratories Limited Erythromycin a derivatives as antibacterial agents
US20090170790A1 (en) * 2004-10-25 2009-07-02 Biswajit Das Ketolide derivatives as antibacterial agents
MX2007007598A (es) * 2004-12-21 2007-07-25 Pfizer Prod Inc Macrolidos.
EP1957085A2 (en) * 2005-11-08 2008-08-20 Ranbaxy Laboratories, Ltd. Macrolides as anti-inflammatory agents
WO2007060518A2 (en) * 2005-11-23 2007-05-31 Ranbaxy Laboratories Limited Ketolide derivatives as antibacterial agents
US20090130225A1 (en) * 2005-11-23 2009-05-21 Anjan Chakrabarti Macrolides derivatives as antibacterial agents
EP1954294A2 (en) * 2005-11-23 2008-08-13 Ranbaxy Laboratories Limited Use of macrolide derivatives for treating acne
WO2008072034A1 (en) * 2006-12-12 2008-06-19 Zambon S.P.A. Macrolide compounds endowed with antiinflammatory activity
AU2019403048B2 (en) * 2018-12-17 2025-01-23 Lunella Biotech, Inc. Triple combination therapies for targeting mitochondria and killing cancer stem cells

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3725385A (en) * 1970-11-02 1973-04-03 Abbott Lab Process for the demethylation of 3-amino macrolides
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2719587B1 (fr) * 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
KR19990067492A (ko) * 1995-11-08 1999-08-25 스티븐 에프. 웨인스톡 트리사이클릭 에리트로마이신 유도체
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2745290B1 (fr) * 1996-02-28 1998-04-03 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
BR9711661A (pt) * 1996-09-04 1999-08-24 Abbott Lab Composto composi-Æo farmac-utica e processos para controlar uma infec-Æo bacteriana em um mam¡fero e para preparar um composto
JP2001518476A (ja) * 1997-09-30 2001-10-16 アボット・ラボラトリーズ 抗菌活性を有する3’−n−修飾6−o−置換エリスロマイシンケトライド誘導体

Also Published As

Publication number Publication date
EP0974598B1 (fr) 2011-08-24
EP0974598A3 (fr) 2003-12-17
EP0974598A2 (fr) 2000-01-26
ES2372156T3 (es) 2012-01-16
CY1112087T1 (el) 2015-11-04
US6433151B1 (en) 2002-08-13
ATE521619T1 (de) 2011-09-15
JP4573925B2 (ja) 2010-11-04
DK0974598T3 (da) 2011-12-19
JP2000026494A (ja) 2000-01-25

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