PT96154A - Processo para a preparacao de derivados de carbamoilo e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados de carbamoilo e de composicoes farmaceuticas que os contem

Info

Publication number
PT96154A
PT96154A PT96154A PT9615490A PT96154A PT 96154 A PT96154 A PT 96154A PT 96154 A PT96154 A PT 96154A PT 9615490 A PT9615490 A PT 9615490A PT 96154 A PT96154 A PT 96154A
Authority
PT
Portugal
Prior art keywords
carbamoil
derivatives
preparing
contain
pharmaceutical compositions
Prior art date
Application number
PT96154A
Other languages
English (en)
Other versions
PT96154B (pt
Inventor
Robert Toms Jacobs
Original Assignee
Ici Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Plc filed Critical Ici Plc
Publication of PT96154A publication Critical patent/PT96154A/pt
Publication of PT96154B publication Critical patent/PT96154B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/24Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an alkyl or cycloalkyl radical attached to the ring nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/02Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C211/15Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT96154A 1989-12-11 1990-12-11 Processo para a preparacao de derivados de carbamoilo e de composicoes farmaceuticas que os contem PT96154B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898927981A GB8927981D0 (en) 1989-12-11 1989-12-11 Carbamoyl derivative

Publications (2)

Publication Number Publication Date
PT96154A true PT96154A (pt) 1991-09-30
PT96154B PT96154B (pt) 1998-05-29

Family

ID=10667774

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96154A PT96154B (pt) 1989-12-11 1990-12-11 Processo para a preparacao de derivados de carbamoilo e de composicoes farmaceuticas que os contem

Country Status (31)

Country Link
EP (1) EP0432984B1 (pt)
JP (1) JPH0822849B2 (pt)
KR (1) KR100192999B1 (pt)
CN (1) CN1025786C (pt)
AP (1) AP192A (pt)
AT (1) ATE163641T1 (pt)
AU (1) AU642182B2 (pt)
BG (2) BG60015B2 (pt)
CA (1) CA2031897C (pt)
CZ (1) CZ282068B6 (pt)
DE (1) DE69032083T2 (pt)
DK (1) DK0432984T3 (pt)
ES (1) ES2112832T3 (pt)
FI (1) FI95029C (pt)
GB (2) GB8927981D0 (pt)
GR (1) GR3026279T3 (pt)
HR (1) HRP930326B1 (pt)
HU (2) HU210441B (pt)
IE (1) IE904448A1 (pt)
IL (1) IL96621A (pt)
MY (1) MY106363A (pt)
NO (1) NO174198C (pt)
PL (2) PL166516B1 (pt)
PT (1) PT96154B (pt)
RO (1) RO108562B1 (pt)
RU (1) RU2002740C1 (pt)
SI (1) SI9012330A (pt)
SK (1) SK278528B6 (pt)
TW (1) TW219329B (pt)
YU (1) YU48218B (pt)
ZA (1) ZA909898B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0455596B1 (de) * 1990-05-04 1994-11-02 Novartis AG Substituierte Indole
GB9020338D0 (en) * 1990-09-18 1990-10-31 Lilly Industries Ltd Pharmaceutical compounds
GB9026425D0 (en) * 1990-12-05 1991-01-23 Ici Plc Process
GB9026427D0 (en) * 1990-12-05 1991-01-23 Ici Plc Chemical process
GB9119001D0 (en) * 1991-09-05 1991-10-23 Ici Plc Pharmaceutical agents
ES2050611B1 (es) * 1992-10-08 1994-12-16 Ici Plc Una nueva forma fisica de un derivado de carbamoilindol con propiedades antagonistas de leucotrienos.
GR1001368B (el) * 1992-10-08 1993-10-29 Ici Plc Φαρμακευτικοί φορείς.
WO1996008496A1 (en) * 1994-09-16 1996-03-21 Takeda Chemical Industries, Ltd. Triazolopyridazines process and intermediates for their preparation and their use as medicaments
US7166638B2 (en) * 2003-05-27 2007-01-23 Nicox S.A. Statin derivatives
AU2005296305A1 (en) * 2004-10-12 2006-04-27 Decode Genetics Ehf Sulfonamide peri-substituted bicyclics for occlusive artery disease
EP1852420B1 (en) * 2005-02-25 2012-10-17 Ono Pharmaceutical Co., Ltd. Indole compounds for treating respiratory disorders

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4524152A (en) * 1982-12-30 1985-06-18 Pennwalt Corporation 1-Cyano-3-(fluoroalkyl)guanidines for lowering blood pressure
GB8623429D0 (en) * 1985-10-17 1986-11-05 Ici America Inc Carboximide derivatives
EP0227241B1 (en) * 1985-10-17 1996-09-11 Zeneca Inc. Medicinal indole and indazole keto sulphone derivatives
MY103259A (en) * 1987-04-15 1993-05-29 Ici America Inc Aliphatic carboxamides
GB8906032D0 (en) * 1988-04-14 1989-04-26 Ici America Inc Hetera-aliphatic carboxamides
GB9026425D0 (en) * 1990-12-05 1991-01-23 Ici Plc Process

Also Published As

Publication number Publication date
CN1025786C (zh) 1994-08-31
GB8927981D0 (en) 1990-02-14
IE904448A1 (en) 1991-06-19
SK614690A3 (en) 1997-08-06
EP0432984B1 (en) 1998-03-04
SK278528B6 (en) 1997-08-06
CN1053604A (zh) 1991-08-07
HU908137D0 (en) 1991-06-28
NO174198B (no) 1993-12-20
ZA909898B (en) 1991-08-28
JPH0770061A (ja) 1995-03-14
ATE163641T1 (de) 1998-03-15
BG50606A3 (bg) 1992-09-15
BG60015B2 (bg) 1993-06-30
HK1003830A1 (en) 1998-11-06
KR910011780A (ko) 1991-08-07
JPH0822849B2 (ja) 1996-03-06
RU2002740C1 (ru) 1993-11-15
GB2238790A (en) 1991-06-12
NO905327L (no) 1991-06-12
PL166516B1 (pl) 1995-05-31
PL288184A1 (en) 1992-04-21
FI95029C (fi) 1995-12-11
MY106363A (en) 1995-05-30
YU48218B (sh) 1997-08-22
NO174198C (no) 1994-04-06
IL96621A0 (en) 1991-09-16
HRP930326A2 (en) 1996-06-30
CA2031897A1 (en) 1991-06-12
TW219329B (pt) 1994-01-21
FI906084A0 (fi) 1990-12-11
EP0432984A3 (en) 1992-04-22
RO108562B1 (ro) 1994-06-30
DE69032083D1 (de) 1998-04-09
GB2238790B (en) 1993-06-30
ES2112832T3 (es) 1998-04-16
PT96154B (pt) 1998-05-29
HRP930326B1 (en) 1998-12-31
GB9026797D0 (en) 1991-01-30
HUT56345A (en) 1991-08-28
KR100192999B1 (ko) 1999-06-15
AP192A (en) 1992-06-30
CZ614690A3 (en) 1997-05-14
EP0432984A2 (en) 1991-06-19
HU210441B (en) 1995-04-28
PL167449B1 (pl) 1995-09-30
DE69032083T2 (de) 1998-07-16
FI95029B (fi) 1995-08-31
AP9000230A0 (en) 1991-01-31
AU6791790A (en) 1991-06-13
CA2031897C (en) 2001-12-18
CZ282068B6 (cs) 1997-05-14
IL96621A (en) 1994-11-28
GR3026279T3 (en) 1998-06-30
AU642182B2 (en) 1993-10-14
SI9012330A (en) 1997-12-31
HU210877A9 (en) 1995-09-28
NO905327D0 (no) 1990-12-10
YU233090A (sh) 1993-05-28
FI906084L (fi) 1991-06-12
DK0432984T3 (da) 1998-11-30

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19910509

FG3A Patent granted, date of granting

Effective date: 19980213

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20040813