PT87734A - Procede de preparation de nouveaux tripeptides a structure polycyclique azotee et de compositions pharmaceutiques les contenant - Google Patents
Procede de preparation de nouveaux tripeptides a structure polycyclique azotee et de compositions pharmaceutiques les contenantInfo
- Publication number
- PT87734A PT87734A PT87734A PT8773488A PT87734A PT 87734 A PT87734 A PT 87734A PT 87734 A PT87734 A PT 87734A PT 8773488 A PT8773488 A PT 8773488A PT 87734 A PT87734 A PT 87734A
- Authority
- PT
- Portugal
- Prior art keywords
- denotes
- azotee
- polycyclique
- nouveaux
- procede
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000003277 amino group Chemical group 0.000 abstract 1
- -1 amino, mercapto, methylthio, carboxyl Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 238000002483 medication Methods 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001544 thienyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0815—Tripeptides with the first amino acid being basic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Communicable Diseases (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Transplantation (AREA)
- Virology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8708350A FR2616663B1 (fr) | 1987-06-16 | 1987-06-16 | Nouveaux tripeptides a structure polycyclique azotee, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT87734A true PT87734A (pt) | 1988-07-01 |
| PT87734B PT87734B (pt) | 1992-10-30 |
Family
ID=9352075
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT87734A PT87734B (pt) | 1987-06-16 | 1988-06-15 | Processo para a preparacao de novos tripeptidos com estrutura policiclica azotada e de composicoes farmaceuticas que os contem |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US5047400A (pt) |
| EP (1) | EP0296059B1 (pt) |
| JP (1) | JPH0637518B2 (pt) |
| AT (1) | ATE73822T1 (pt) |
| AU (1) | AU612657B2 (pt) |
| CA (1) | CA1336349C (pt) |
| DE (1) | DE3869223D1 (pt) |
| DK (1) | DK330588A (pt) |
| ES (1) | ES2032985T3 (pt) |
| FR (1) | FR2616663B1 (pt) |
| GR (1) | GR3004851T3 (pt) |
| IE (1) | IE66224B1 (pt) |
| NZ (1) | NZ225043A (pt) |
| OA (1) | OA08881A (pt) |
| PT (1) | PT87734B (pt) |
| ZA (1) | ZA884276B (pt) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0454302A3 (en) * | 1990-03-30 | 1992-10-14 | Banyu Pharmaceutical Co., Ltd. | Tuftsin derivatives |
| FR2663336B1 (fr) * | 1990-06-18 | 1992-09-04 | Adir | Nouveaux derives peptidiques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| JPH0813834B2 (ja) * | 1990-08-01 | 1996-02-14 | 日東紡績株式会社 | トリペプチド誘導体及びそれを有効成分とする蛋白分解酵素阻害剤 |
| JPH08503475A (ja) * | 1992-11-25 | 1996-04-16 | メルク エンド カンパニー インコーポレーテッド | 抗変性活性剤としてのカルボキシ−ペプチジル誘導体 |
| US5569745A (en) * | 1994-02-25 | 1996-10-29 | Resolution Pharmaceuticals Inc. | Peptide-Chelator conjugates |
| US5662885A (en) * | 1994-07-22 | 1997-09-02 | Resolution Pharmaceuticals Inc. | Peptide derived radionuclide chelators |
| GB9526577D0 (en) * | 1995-12-28 | 1996-02-28 | Nat Power Plc | Method for the fabrication of electrochemical cells |
| WO2003031437A1 (en) * | 2001-10-09 | 2003-04-17 | Smithkline Beecham Corporation | Propylcarbamate derivatives as inhibitors of serine and cysteine proteases |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2343034C2 (de) * | 1973-08-25 | 1984-08-23 | Hoechst Ag, 6230 Frankfurt | Tetrapeptide mit phagocytose-stimulierender Wirkung, Verfahren zu deren Herstellung und deren Verwendung |
| IT8021120A0 (it) * | 1979-04-02 | 1980-04-01 | Inst Organicheskogo Sinteza Ak | Analogo ciclico del peptide naturale stimolante la fagocitosi: treonile-ciclo (n-lisile-prolile-arginile). |
| FR2575753B1 (fr) * | 1985-01-07 | 1987-02-20 | Adir | Nouveaux derives peptidiques a structure polycyclique azotee, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| FR2601957B1 (fr) * | 1986-07-22 | 1988-11-10 | Pf Medicament | Derives tetrapeptidiques, procede pour leur preparation, leur utilisation en tant que medicaments et compositions pharmaceutiques obtenues |
| FR2610934B1 (fr) * | 1987-02-13 | 1989-05-05 | Adir | Nouveaux derives peptidiques a structure polycyclique azotee, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
1987
- 1987-06-16 FR FR8708350A patent/FR2616663B1/fr not_active Expired
-
1988
- 1988-06-15 PT PT87734A patent/PT87734B/pt not_active IP Right Cessation
- 1988-06-15 EP EP88401476A patent/EP0296059B1/fr not_active Expired - Lifetime
- 1988-06-15 JP JP63147930A patent/JPH0637518B2/ja not_active Expired - Lifetime
- 1988-06-15 AU AU17741/88A patent/AU612657B2/en not_active Ceased
- 1988-06-15 ES ES198888401476T patent/ES2032985T3/es not_active Expired - Lifetime
- 1988-06-15 IE IE180388A patent/IE66224B1/en not_active IP Right Cessation
- 1988-06-15 NZ NZ225043A patent/NZ225043A/en unknown
- 1988-06-15 DE DE8888401476T patent/DE3869223D1/de not_active Expired - Lifetime
- 1988-06-15 AT AT88401476T patent/ATE73822T1/de not_active IP Right Cessation
- 1988-06-15 OA OA59375A patent/OA08881A/xx unknown
- 1988-06-15 ZA ZA884276A patent/ZA884276B/xx unknown
- 1988-06-16 DK DK330588A patent/DK330588A/da not_active Application Discontinuation
- 1988-06-16 US US07/207,710 patent/US5047400A/en not_active Expired - Fee Related
- 1988-06-16 CA CA000569700A patent/CA1336349C/fr not_active Expired - Fee Related
-
1992
- 1992-06-10 GR GR920401204T patent/GR3004851T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2032985T3 (es) | 1993-03-01 |
| JPH0637518B2 (ja) | 1994-05-18 |
| NZ225043A (en) | 1990-04-26 |
| FR2616663A1 (fr) | 1988-12-23 |
| AU1774188A (en) | 1988-12-22 |
| CA1336349C (fr) | 1995-07-18 |
| OA08881A (fr) | 1989-10-31 |
| IE66224B1 (en) | 1995-12-13 |
| ZA884276B (en) | 1989-03-29 |
| AU612657B2 (en) | 1991-07-18 |
| DK330588A (da) | 1988-12-17 |
| EP0296059A1 (fr) | 1988-12-21 |
| US5047400A (en) | 1991-09-10 |
| DK330588D0 (da) | 1988-06-16 |
| DE3869223D1 (de) | 1992-04-23 |
| PT87734B (pt) | 1992-10-30 |
| EP0296059B1 (fr) | 1992-03-18 |
| IE881803L (en) | 1988-12-16 |
| JPS6419096A (en) | 1989-01-23 |
| GR3004851T3 (pt) | 1993-04-28 |
| ATE73822T1 (de) | 1992-04-15 |
| FR2616663B1 (fr) | 1989-08-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG3A | Patent granted, date of granting |
Effective date: 19920423 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19961031 |