ES2032985T3 - Nuevos tripeptidos de estructura policiclica nitrogenada, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. - Google Patents

Nuevos tripeptidos de estructura policiclica nitrogenada, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.

Info

Publication number
ES2032985T3
ES2032985T3 ES198888401476T ES88401476T ES2032985T3 ES 2032985 T3 ES2032985 T3 ES 2032985T3 ES 198888401476 T ES198888401476 T ES 198888401476T ES 88401476 T ES88401476 T ES 88401476T ES 2032985 T3 ES2032985 T3 ES 2032985T3
Authority
ES
Spain
Prior art keywords
denotes
nitrogen
polyclic
contain
pharmaceutical compositions
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES198888401476T
Other languages
English (en)
Inventor
Michel Vincent
Georges Remond
Bernard Portevin
Claude Cudennec
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ADIR SARL
Original Assignee
ADIR SARL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ADIR SARL filed Critical ADIR SARL
Application granted granted Critical
Publication of ES2032985T3 publication Critical patent/ES2032985T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0815—Tripeptides with the first amino acid being basic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

LA INVENCION SE REFIERE A COMPUESTOS DE FORMULA GENETAL (I) EN LA QUE X REPRESENTA UN ATOMO DE OXIGENO, DOS ATOMOS DE NITROGENO; Y REPRESENTA UN ATOMO DE HIDROGENO, DOS AGRUPAMIENTOS HIDROXILO O Y REPRESENTA UN AGRUPAMIENTO AMINO CON LA CONDICION DE QUE X REPRESENTE DOS ATOMOS DE HIDROGENO; R REPRESENTA UN ATOMO DE HIDROGENO, UN AGRUPAMIENTO ALCOILO DE 1 A 6 ATOMOS DE CARBONO DE CADENA RECTA O RAMIFICADA EVENTUALMENTE SUSTITUIDA POR UNO O VARIOS AGRUPAMIENTOS HIDROXI, AMINO, MERCAPTO, METILTIO, CARBOXI O ARILO COMO FENILO, PIRIDILO O TIENILO. (II) REPRESENTA UNA ESTRCUTURA POLICICLICA NITROGENADA, SUS ENANCIOMEROS, EPIMEROS Y DIASTEREOISOMEROS ASI COMO SUS SALES DE ADICION A UN ACIDO O UNA BASE FARMACEUTICAMENTE ACEPTABLE. MEDICAMENTOS.
ES198888401476T 1987-06-16 1988-06-15 Nuevos tripeptidos de estructura policiclica nitrogenada, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. Expired - Lifetime ES2032985T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8708350A FR2616663B1 (fr) 1987-06-16 1987-06-16 Nouveaux tripeptides a structure polycyclique azotee, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
ES2032985T3 true ES2032985T3 (es) 1993-03-01

Family

ID=9352075

Family Applications (1)

Application Number Title Priority Date Filing Date
ES198888401476T Expired - Lifetime ES2032985T3 (es) 1987-06-16 1988-06-15 Nuevos tripeptidos de estructura policiclica nitrogenada, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.

Country Status (16)

Country Link
US (1) US5047400A (es)
EP (1) EP0296059B1 (es)
JP (1) JPH0637518B2 (es)
AT (1) ATE73822T1 (es)
AU (1) AU612657B2 (es)
CA (1) CA1336349C (es)
DE (1) DE3869223D1 (es)
DK (1) DK330588A (es)
ES (1) ES2032985T3 (es)
FR (1) FR2616663B1 (es)
GR (1) GR3004851T3 (es)
IE (1) IE66224B1 (es)
NZ (1) NZ225043A (es)
OA (1) OA08881A (es)
PT (1) PT87734B (es)
ZA (1) ZA884276B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0454302A3 (en) * 1990-03-30 1992-10-14 Banyu Pharmaceutical Co., Ltd. Tuftsin derivatives
FR2663336B1 (fr) * 1990-06-18 1992-09-04 Adir Nouveaux derives peptidiques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
JPH0813834B2 (ja) * 1990-08-01 1996-02-14 日東紡績株式会社 トリペプチド誘導体及びそれを有効成分とする蛋白分解酵素阻害剤
AU679474B2 (en) * 1992-11-25 1997-07-03 Merck & Co., Inc. Carboxy-peptidyl derivatives as antidegenerative active agents
US5569745A (en) * 1994-02-25 1996-10-29 Resolution Pharmaceuticals Inc. Peptide-Chelator conjugates
US5662885A (en) * 1994-07-22 1997-09-02 Resolution Pharmaceuticals Inc. Peptide derived radionuclide chelators
GB9526577D0 (en) * 1995-12-28 1996-02-28 Nat Power Plc Method for the fabrication of electrochemical cells
EP1448554A1 (en) * 2001-10-09 2004-08-25 SmithKline Beecham Corporation Propylcarbamate derivatives as inhibitors of serine and cysteine proteases

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2343034C2 (de) * 1973-08-25 1984-08-23 Hoechst Ag, 6230 Frankfurt Tetrapeptide mit phagocytose-stimulierender Wirkung, Verfahren zu deren Herstellung und deren Verwendung
IT8021120A0 (it) * 1979-04-02 1980-04-01 Inst Organicheskogo Sinteza Ak Analogo ciclico del peptide naturale stimolante la fagocitosi: treonile-ciclo (n-lisile-prolile-arginile).
FR2575753B1 (fr) * 1985-01-07 1987-02-20 Adir Nouveaux derives peptidiques a structure polycyclique azotee, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2601957B1 (fr) * 1986-07-22 1988-11-10 Pf Medicament Derives tetrapeptidiques, procede pour leur preparation, leur utilisation en tant que medicaments et compositions pharmaceutiques obtenues
FR2610934B1 (fr) * 1987-02-13 1989-05-05 Adir Nouveaux derives peptidiques a structure polycyclique azotee, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
PT87734A (pt) 1988-07-01
CA1336349C (fr) 1995-07-18
IE66224B1 (en) 1995-12-13
ATE73822T1 (de) 1992-04-15
AU612657B2 (en) 1991-07-18
JPH0637518B2 (ja) 1994-05-18
EP0296059B1 (fr) 1992-03-18
DK330588A (da) 1988-12-17
GR3004851T3 (es) 1993-04-28
OA08881A (fr) 1989-10-31
US5047400A (en) 1991-09-10
DE3869223D1 (de) 1992-04-23
FR2616663A1 (fr) 1988-12-23
IE881803L (en) 1988-12-16
ZA884276B (en) 1989-03-29
FR2616663B1 (fr) 1989-08-18
NZ225043A (en) 1990-04-26
DK330588D0 (da) 1988-06-16
AU1774188A (en) 1988-12-22
EP0296059A1 (fr) 1988-12-21
JPS6419096A (en) 1989-01-23
PT87734B (pt) 1992-10-30

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