PT3221331T - Esteroides 6-alquil-7-hidroxi-4-en-3-ona como intermediários para a produção de moduladores de fxr esteroidais - Google Patents

Esteroides 6-alquil-7-hidroxi-4-en-3-ona como intermediários para a produção de moduladores de fxr esteroidais

Info

Publication number
PT3221331T
PT3221331T PT158009092T PT15800909T PT3221331T PT 3221331 T PT3221331 T PT 3221331T PT 158009092 T PT158009092 T PT 158009092T PT 15800909 T PT15800909 T PT 15800909T PT 3221331 T PT3221331 T PT 3221331T
Authority
PT
Portugal
Prior art keywords
steroids
intermediates
hydroxy
alkyl
production
Prior art date
Application number
PT158009092T
Other languages
English (en)
Portuguese (pt)
Inventor
Weymouth-Wilson Alexander
Komsta Zofia
Boydell James
Otter Carl
WALLIS Laura
BATCHELOR Rhys
Original Assignee
Nzp Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB1420594.2A external-priority patent/GB201420594D0/en
Priority claimed from GBGB1420593.4A external-priority patent/GB201420593D0/en
Priority claimed from GBGB1505670.8A external-priority patent/GB201505670D0/en
Application filed by Nzp Uk Ltd filed Critical Nzp Uk Ltd
Publication of PT3221331T publication Critical patent/PT3221331T/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT158009092T 2014-11-19 2015-11-19 Esteroides 6-alquil-7-hidroxi-4-en-3-ona como intermediários para a produção de moduladores de fxr esteroidais PT3221331T (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1420594.2A GB201420594D0 (en) 2014-11-19 2014-11-19 Compounds
GBGB1420593.4A GB201420593D0 (en) 2014-11-19 2014-11-19 Compounds
GBGB1505670.8A GB201505670D0 (en) 2015-04-01 2015-04-01 Compounds

Publications (1)

Publication Number Publication Date
PT3221331T true PT3221331T (pt) 2019-12-23

Family

ID=54704019

Family Applications (1)

Application Number Title Priority Date Filing Date
PT158009092T PT3221331T (pt) 2014-11-19 2015-11-19 Esteroides 6-alquil-7-hidroxi-4-en-3-ona como intermediários para a produção de moduladores de fxr esteroidais

Country Status (15)

Country Link
US (1) US10301350B2 (cg-RX-API-DMAC7.html)
EP (1) EP3221331B1 (cg-RX-API-DMAC7.html)
JP (1) JP6700274B2 (cg-RX-API-DMAC7.html)
KR (1) KR102526631B1 (cg-RX-API-DMAC7.html)
CN (1) CN107207559B (cg-RX-API-DMAC7.html)
BR (1) BR112017010319B1 (cg-RX-API-DMAC7.html)
CA (1) CA2968309A1 (cg-RX-API-DMAC7.html)
DK (1) DK3221331T3 (cg-RX-API-DMAC7.html)
EA (1) EA033427B1 (cg-RX-API-DMAC7.html)
ES (1) ES2759725T3 (cg-RX-API-DMAC7.html)
MX (1) MX375863B (cg-RX-API-DMAC7.html)
PL (1) PL3221331T3 (cg-RX-API-DMAC7.html)
PT (1) PT3221331T (cg-RX-API-DMAC7.html)
TW (1) TWI690536B (cg-RX-API-DMAC7.html)
WO (1) WO2016079517A1 (cg-RX-API-DMAC7.html)

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Also Published As

Publication number Publication date
BR112017010319B1 (pt) 2023-04-11
CN107207559B (zh) 2019-10-25
JP6700274B2 (ja) 2020-05-27
MX375863B (es) 2025-03-07
MX2017006563A (es) 2018-01-26
DK3221331T3 (da) 2019-12-02
US20170327528A1 (en) 2017-11-16
EA201790884A8 (ru) 2019-07-31
NZ731924A (en) 2020-12-18
KR20170086604A (ko) 2017-07-26
US10301350B2 (en) 2019-05-28
HK1246801A1 (en) 2018-09-14
WO2016079517A1 (en) 2016-05-26
TWI690536B (zh) 2020-04-11
JP2017534670A (ja) 2017-11-24
KR102526631B1 (ko) 2023-04-27
BR112017010319A2 (pt) 2017-12-26
EP3221331B1 (en) 2019-09-18
EA033427B1 (ru) 2019-10-31
EA201790884A1 (ru) 2017-11-30
PL3221331T3 (pl) 2020-03-31
CA2968309A1 (en) 2016-05-26
CN107207559A (zh) 2017-09-26
EP3221331A1 (en) 2017-09-27
ES2759725T3 (es) 2020-05-12
TW201632537A (zh) 2016-09-16

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