PT1166773E - Solucao de tetra-hidrato do sal monossodico da n-o(p-pivaloiloxibenzenossulfonilamino)benzoilglicina e seu produto farmaceutico - Google Patents

Solucao de tetra-hidrato do sal monossodico da n-o(p-pivaloiloxibenzenossulfonilamino)benzoilglicina e seu produto farmaceutico

Info

Publication number
PT1166773E
PT1166773E PT01305556T PT01305556T PT1166773E PT 1166773 E PT1166773 E PT 1166773E PT 01305556 T PT01305556 T PT 01305556T PT 01305556 T PT01305556 T PT 01305556T PT 1166773 E PT1166773 E PT 1166773E
Authority
PT
Portugal
Prior art keywords
pivaloyloxibenzenesulfonylamino
benzoylglycine
pharmaceutical product
hydrate solution
salt tetra
Prior art date
Application number
PT01305556T
Other languages
English (en)
Inventor
Akira Takada
Masao Sudoh
Original Assignee
Ono Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ono Pharmaceutical Co filed Critical Ono Pharmaceutical Co
Publication of PT1166773E publication Critical patent/PT1166773E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/37Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • C07C311/38Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton
    • C07C311/44Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pulmonology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT01305556T 2000-06-29 2001-06-27 Solucao de tetra-hidrato do sal monossodico da n-o(p-pivaloiloxibenzenossulfonilamino)benzoilglicina e seu produto farmaceutico PT1166773E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000195853 2000-06-29
JP2000195852 2000-06-29

Publications (1)

Publication Number Publication Date
PT1166773E true PT1166773E (pt) 2004-05-31

Family

ID=26594951

Family Applications (1)

Application Number Title Priority Date Filing Date
PT01305556T PT1166773E (pt) 2000-06-29 2001-06-27 Solucao de tetra-hidrato do sal monossodico da n-o(p-pivaloiloxibenzenossulfonilamino)benzoilglicina e seu produto farmaceutico

Country Status (19)

Country Link
US (1) US6552082B2 (pt)
EP (1) EP1166773B1 (pt)
KR (1) KR100725076B1 (pt)
CN (1) CN1263736C (pt)
AT (1) ATE259218T1 (pt)
AU (1) AU782838B2 (pt)
BR (1) BR0102604B1 (pt)
CA (1) CA2351273C (pt)
DE (1) DE60101979T2 (pt)
DK (1) DK1166773T3 (pt)
ES (1) ES2215856T3 (pt)
HU (1) HUP0102699A2 (pt)
MX (1) MXPA01006698A (pt)
NO (1) NO330296B1 (pt)
NZ (1) NZ512486A (pt)
PT (1) PT1166773E (pt)
RU (1) RU2272623C2 (pt)
TR (1) TR200400585T4 (pt)
TW (1) TWI246925B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2416600A1 (en) * 2000-07-24 2003-01-20 Ono Pharmaceutical Co., Ltd. Freeze-dried preparation of n-¬o-(p-pivaloyloxybenzenesulfonylamino)benzoyl|glycine monosodium salt tetrahydrate and a process for the maufacture thereof
US20050101633A1 (en) * 2001-05-17 2005-05-12 Takeharu Tonai Remedial agent for myelopathic disease
TW200519080A (en) * 2003-10-03 2005-06-16 Ono Pharmaceutical Co Agent containinf (2R)-2-propyloctanic acid as effective component
CA2707484C (en) 2007-12-04 2021-08-10 Remedy Pharmaceuticals, Inc. Improved formulations and methods for lyophilization and lyophilates provided thereby
KR101247137B1 (ko) * 2011-03-23 2013-04-01 주식회사 엠씨켐 N-[o-(p-피발로일옥시벤젠술포닐아미노)벤조일]글리신의 신규 제조 방법 및 그 모노나트륨염ㆍ4 수화물의 동결 건조 제제의 제조 방법
KR101366706B1 (ko) 2012-12-06 2014-02-24 상명대학교서울산학협력단 N-[o-(p-피발로일옥시벤젠술포닐아미노)벤조일]글리신의 신규 제조 방법 및 그 모노나트륨염ㆍ4 수화물의 동결 건조 제제의 제조 방법
CN104107172B (zh) * 2013-04-18 2017-11-28 上海汇伦生命科技有限公司 西维来司钠注射用冻干粉的制备方法
CN114681435A (zh) * 2020-12-31 2022-07-01 上海汇伦生物科技有限公司 吸入用药物组合物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0320253A (ja) 1988-06-13 1991-01-29 Ono Pharmaceut Co Ltd ピバル酸 p―置換フェニルエステル誘導体、それらの製造方法およびそれらを有効成分として含有するエラスターゼ阻害剤
CA1340191C (en) 1988-06-13 1998-12-15 Katsuhiro Imaki Derivatives of p-substituted phenyl ester of pivalic acid
IT1242642B (it) * 1990-04-17 1994-05-16 Alfa Wassermann Spa Formulazioni iniettabili contenenti naproxen sale sodico.
JP3020253B2 (ja) 1990-05-02 2000-03-15 松下電工株式会社 配線器具の取付枠への取付構造
EP0539223A1 (en) 1991-10-25 1993-04-28 Ono Pharmaceutical Co., Ltd. Glycine derivative monosodium salt tetrahydrate having an inhibitory effect on elastase
JPH05194366A (ja) 1991-10-25 1993-08-03 Ono Pharmaceut Co Ltd グリシン誘導体・モノナトリウム塩・4水和物、その製造方法、それを含有する薬剤および該誘導体の中間体の製造方法
JP3193597B2 (ja) 1995-07-28 2001-07-30 小野薬品工業株式会社 グリシン誘導体の製造方法
AU5528299A (en) 1998-09-15 2000-04-03 Naeja Pharmaceutical Inc. Combined therapy for treatment of inflammation using elastase inhibitor(s) and antibacterial agent(s)
AU6870800A (en) * 1999-09-06 2001-04-10 Ono Pharmaceutical Co. Ltd. Preventive and therapeutic agents for eye diseases

Also Published As

Publication number Publication date
KR100725076B1 (ko) 2007-06-08
RU2272623C2 (ru) 2006-03-27
NO20013223D0 (no) 2001-06-27
ES2215856T3 (es) 2004-10-16
DE60101979D1 (de) 2004-03-18
NO20013223L (no) 2001-12-31
AU782838B2 (en) 2005-09-01
NZ512486A (en) 2001-12-21
KR20020002242A (ko) 2002-01-09
US20020022738A1 (en) 2002-02-21
BR0102604A (pt) 2002-02-13
CA2351273A1 (en) 2001-12-29
TR200400585T4 (tr) 2004-04-21
CN1263736C (zh) 2006-07-12
BR0102604B1 (pt) 2012-06-26
CN1341591A (zh) 2002-03-27
DE60101979T2 (de) 2005-01-05
AU5409201A (en) 2002-03-28
CA2351273C (en) 2010-09-07
MXPA01006698A (es) 2004-07-30
US6552082B2 (en) 2003-04-22
HU0102699D0 (en) 2001-08-28
NO330296B1 (no) 2011-03-21
TWI246925B (en) 2006-01-11
DK1166773T3 (da) 2004-06-07
ATE259218T1 (de) 2004-02-15
EP1166773A1 (en) 2002-01-02
HUP0102699A2 (en) 2002-06-29
EP1166773B1 (en) 2004-02-11

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