PT1082119E - Pre-concentrados de microemulsao contendo um antagonista da substancia p da piperidina - Google Patents

Pre-concentrados de microemulsao contendo um antagonista da substancia p da piperidina

Info

Publication number
PT1082119E
PT1082119E PT99927760T PT99927760T PT1082119E PT 1082119 E PT1082119 E PT 1082119E PT 99927760 T PT99927760 T PT 99927760T PT 99927760 T PT99927760 T PT 99927760T PT 1082119 E PT1082119 E PT 1082119E
Authority
PT
Portugal
Prior art keywords
microemulation
antagonist
concentrates
piperidine substance
piperidine
Prior art date
Application number
PT99927760T
Other languages
English (en)
Portuguese (pt)
Inventor
Steffen Lang
Kurt Liechti
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9811200.6A external-priority patent/GB9811200D0/en
Priority claimed from GBGB9818105.0A external-priority patent/GB9818105D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PT1082119E publication Critical patent/PT1082119E/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Biophysics (AREA)
  • Dispersion Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT99927760T 1998-05-26 1999-05-26 Pre-concentrados de microemulsao contendo um antagonista da substancia p da piperidina PT1082119E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9811200.6A GB9811200D0 (en) 1998-05-26 1998-05-26 Organic compounds
GBGB9818105.0A GB9818105D0 (en) 1998-08-19 1998-08-19 Organic compounds

Publications (1)

Publication Number Publication Date
PT1082119E true PT1082119E (pt) 2004-05-31

Family

ID=26313736

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99927760T PT1082119E (pt) 1998-05-26 1999-05-26 Pre-concentrados de microemulsao contendo um antagonista da substancia p da piperidina

Country Status (30)

Country Link
US (2) US20020156099A1 (cg-RX-API-DMAC10.html)
EP (1) EP1082119B1 (cg-RX-API-DMAC10.html)
JP (1) JP4083985B2 (cg-RX-API-DMAC10.html)
KR (1) KR20010043669A (cg-RX-API-DMAC10.html)
CN (1) CN1270714C (cg-RX-API-DMAC10.html)
AR (1) AR018376A1 (cg-RX-API-DMAC10.html)
AT (1) ATE257380T1 (cg-RX-API-DMAC10.html)
AU (1) AU755134B2 (cg-RX-API-DMAC10.html)
BE (1) BE1012143A5 (cg-RX-API-DMAC10.html)
BR (1) BR9910696A (cg-RX-API-DMAC10.html)
CA (1) CA2333154C (cg-RX-API-DMAC10.html)
DE (2) DE19983247T1 (cg-RX-API-DMAC10.html)
DK (1) DK1082119T3 (cg-RX-API-DMAC10.html)
ES (1) ES2214859T3 (cg-RX-API-DMAC10.html)
FR (1) FR2779145B1 (cg-RX-API-DMAC10.html)
GB (1) GB2353473A (cg-RX-API-DMAC10.html)
HU (1) HUP0102202A3 (cg-RX-API-DMAC10.html)
ID (1) ID27096A (cg-RX-API-DMAC10.html)
IL (1) IL139501A0 (cg-RX-API-DMAC10.html)
IT (1) IT1313551B1 (cg-RX-API-DMAC10.html)
NO (1) NO20005920L (cg-RX-API-DMAC10.html)
NZ (1) NZ508325A (cg-RX-API-DMAC10.html)
PE (1) PE20000537A1 (cg-RX-API-DMAC10.html)
PL (1) PL344245A1 (cg-RX-API-DMAC10.html)
PT (1) PT1082119E (cg-RX-API-DMAC10.html)
RU (1) RU2240121C2 (cg-RX-API-DMAC10.html)
SK (1) SK17752000A3 (cg-RX-API-DMAC10.html)
TR (1) TR200003502T2 (cg-RX-API-DMAC10.html)
TW (1) TW537894B (cg-RX-API-DMAC10.html)
WO (1) WO1999061025A1 (cg-RX-API-DMAC10.html)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW537894B (en) 1998-05-26 2003-06-21 Novartis Ag A spontaneously dispersible pharmaceutical composition comprising a piperidine substance P antagonist
AU2003225260A1 (en) * 2002-04-22 2003-11-03 University Of Florida Microemulsions for selective molecular separation
GB0220953D0 (en) 2002-09-10 2002-10-23 Novartis Ag Organic compounds
US7842791B2 (en) 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
FR2935001B1 (fr) * 2008-08-14 2011-12-30 Commissariat Energie Atomique Emulsion fluorescente
FR2934954B1 (fr) 2008-08-14 2011-07-22 Commissariat Energie Atomique Emulsion fluorescente de vert d'indocyanine
FR2934953B1 (fr) 2008-08-14 2011-01-21 Commissariat Energie Atomique Nanoemulsions de nanocristaux
FR2934955B1 (fr) 2008-08-14 2011-07-08 Commissariat Energie Atomique Encapsulation d'agents therapeutiques lipophiles ou amphiphiles dans des nanoemulsions
EP2938324B1 (en) 2012-12-31 2023-11-08 JRX Biotechnology, Inc. Liquid topical pharmaceutical nano-emulsion formulations

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3305689A1 (de) 1983-02-18 1984-08-23 Mack Chem Pharm Pharmazeutische zubereitung mit retardwirkung
US5342625A (en) * 1988-09-16 1994-08-30 Sandoz Ltd. Pharmaceutical compositions comprising cyclosporins
MY110227A (en) * 1991-08-12 1998-03-31 Ciba Geigy Ag 1-acylpiperindine compounds.
DE4220616C2 (de) 1992-06-24 1994-12-22 Byk Gulden Lomberg Chem Fab Dexniguldipin zur intravenösen Verabreichung
DK0589843T3 (da) 1992-09-25 2002-04-02 Novartis Ag Cyclosporinholdige farmaceutiske præparater
GB2278780B (en) * 1993-05-27 1998-10-14 Sandoz Ltd Macrolide formulations
DE69535127T2 (de) * 1994-03-18 2007-02-15 Supernus Pharmaceuticals, Inc. Emulgierte arzneistoffabgabesysteme
TW397825B (en) * 1994-10-14 2000-07-11 Novartis Ag Aroyl-piperidine derivatives
GB2308545B (en) 1994-10-26 1999-06-02 Novartis Ag Pharmaceutical microemulsion preconcentrates
MY129435A (en) * 1994-10-26 2007-04-30 Novartis Ag Pharmaceutical microemulsion preconcentrates
FR2728165A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728169A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
DE69617226T2 (de) * 1995-03-27 2002-07-25 Hisamitsu Pharmaceutical Co., Inc. Piperidinderivate.
NZ280689A (en) 1995-12-15 1997-08-22 Bernard Charles Sherma Sherman Pharmaceutical composition comprising a cyclosporipharmaceutical composition comprising a cyclosporin; a tocol, tocopherol or tocotrienol; and propylen; a tocol, tocopherol or tocotrienol; and propylene carbonate or polyethylene glycol ne carbonate or polyethylene glycol
GB9601120D0 (en) 1996-01-19 1996-03-20 Sandoz Ltd Organic compounds
WO1997045119A1 (en) 1996-05-24 1997-12-04 Novartis Ag Use of substance p antagonists for treating social phobia
TW537894B (en) 1998-05-26 2003-06-21 Novartis Ag A spontaneously dispersible pharmaceutical composition comprising a piperidine substance P antagonist

Also Published As

Publication number Publication date
US20020156099A1 (en) 2002-10-24
BR9910696A (pt) 2001-01-30
HK1035137A1 (en) 2001-11-16
CA2333154A1 (en) 1999-12-02
NZ508325A (en) 2003-06-30
PL344245A1 (en) 2001-10-08
IT1313551B1 (it) 2002-09-09
PE20000537A1 (es) 2000-07-10
US6949257B2 (en) 2005-09-27
DE69914077T2 (de) 2004-06-09
SK17752000A3 (sk) 2001-05-10
CA2333154C (en) 2008-07-08
GB2353473A (en) 2001-02-28
WO1999061025A1 (en) 1999-12-02
AU4500899A (en) 1999-12-13
AR018376A1 (es) 2001-11-14
TR200003502T2 (tr) 2001-04-20
EP1082119A1 (en) 2001-03-14
NO20005920L (no) 2001-01-25
CN1270714C (zh) 2006-08-23
RU2240121C2 (ru) 2004-11-20
FR2779145A1 (fr) 1999-12-03
DE19983247T1 (de) 2001-05-31
GB0028506D0 (en) 2001-01-10
JP2002516280A (ja) 2002-06-04
ITMI991164A1 (it) 2000-11-26
KR20010043669A (ko) 2001-05-25
DE69914077D1 (de) 2004-02-12
CN1303285A (zh) 2001-07-11
HUP0102202A3 (en) 2003-01-28
FR2779145B1 (fr) 2004-07-30
BE1012143A5 (fr) 2000-05-02
EP1082119B1 (en) 2004-01-07
AU755134B2 (en) 2002-12-05
TW537894B (en) 2003-06-21
JP4083985B2 (ja) 2008-04-30
US20030152626A1 (en) 2003-08-14
ID27096A (id) 2001-03-01
ATE257380T1 (de) 2004-01-15
ES2214859T3 (es) 2004-09-16
NO20005920D0 (no) 2000-11-23
HUP0102202A2 (hu) 2001-11-28
DK1082119T3 (da) 2004-04-13
IL139501A0 (en) 2001-11-25

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