PT1082106E - Comprimido efervescente para administração subligual, bucal e gengival de fentanil - Google Patents
Comprimido efervescente para administração subligual, bucal e gengival de fentanil Download PDFInfo
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- PT1082106E PT1082106E PT00919523T PT00919523T PT1082106E PT 1082106 E PT1082106 E PT 1082106E PT 00919523 T PT00919523 T PT 00919523T PT 00919523 T PT00919523 T PT 00919523T PT 1082106 E PT1082106 E PT 1082106E
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- 239000005017 polysaccharide Substances 0.000 description 1
- 229920000036 polyvinylpyrrolidone Polymers 0.000 description 1
- 239000001267 polyvinylpyrrolidone Substances 0.000 description 1
- 235000013855 polyvinylpyrrolidone Nutrition 0.000 description 1
- XAEFZNCEHLXOMS-UHFFFAOYSA-M potassium benzoate Chemical compound [K+].[O-]C(=O)C1=CC=CC=C1 XAEFZNCEHLXOMS-UHFFFAOYSA-M 0.000 description 1
- 239000011736 potassium bicarbonate Substances 0.000 description 1
- 229910000028 potassium bicarbonate Inorganic materials 0.000 description 1
- 235000015497 potassium bicarbonate Nutrition 0.000 description 1
- TYJJADVDDVDEDZ-UHFFFAOYSA-M potassium hydrogencarbonate Chemical compound [K+].OC([O-])=O TYJJADVDDVDEDZ-UHFFFAOYSA-M 0.000 description 1
- 239000000843 powder Substances 0.000 description 1
- 230000008569 process Effects 0.000 description 1
- 230000009467 reduction Effects 0.000 description 1
- 239000010670 sage oil Substances 0.000 description 1
- 208000026451 salivation Diseases 0.000 description 1
- 150000003839 salts Chemical class 0.000 description 1
- 210000000813 small intestine Anatomy 0.000 description 1
- 229910052708 sodium Inorganic materials 0.000 description 1
- 235000015424 sodium Nutrition 0.000 description 1
- 235000017550 sodium carbonate Nutrition 0.000 description 1
- 235000019812 sodium carboxymethyl cellulose Nutrition 0.000 description 1
- 229920001027 sodium carboxymethylcellulose Polymers 0.000 description 1
- AJPJDKMHJJGVTQ-UHFFFAOYSA-M sodium dihydrogen phosphate Chemical compound [Na+].OP(O)([O-])=O AJPJDKMHJJGVTQ-UHFFFAOYSA-M 0.000 description 1
- 239000007787 solid Substances 0.000 description 1
- 239000008107 starch Substances 0.000 description 1
- 239000006190 sub-lingual tablet Substances 0.000 description 1
- 239000005720 sucrose Substances 0.000 description 1
- 230000009747 swallowing Effects 0.000 description 1
- 239000006068 taste-masking agent Substances 0.000 description 1
- 230000001225 therapeutic effect Effects 0.000 description 1
- 239000010678 thyme oil Substances 0.000 description 1
- 239000004408 titanium dioxide Substances 0.000 description 1
- 238000005550 wet granulation Methods 0.000 description 1
- 239000009637 wintergreen oil Substances 0.000 description 1
- OENHQHLEOONYIE-JLTXGRSLSA-N β-Carotene Chemical compound CC=1CCCC(C)(C)C=1\C=C\C(\C)=C\C=C\C(\C)=C\C=C\C=C(/C)\C=C\C=C(/C)\C=C\C1=C(C)CCCC1(C)C OENHQHLEOONYIE-JLTXGRSLSA-N 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4468—Non condensed piperidines, e.g. piperocaine having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0007—Effervescent
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27742499A | 1999-03-26 | 1999-03-26 | |
| US09/327,814 US6200604B1 (en) | 1998-03-27 | 1999-06-08 | Sublingual buccal effervescent |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT1082106E true PT1082106E (pt) | 2007-02-28 |
Family
ID=26958475
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT00919523T PT1082106E (pt) | 1999-03-26 | 2000-03-22 | Comprimido efervescente para administração subligual, bucal e gengival de fentanil |
| PT03029877T PT1419765E (pt) | 1999-03-26 | 2000-03-22 | Métodos de manufactura de composições farmacêuticas |
| PT03029911T PT1417959E (pt) | 1999-03-26 | 2000-03-22 | Composições farmacêuticas para a administração oral de um medicamento |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT03029877T PT1419765E (pt) | 1999-03-26 | 2000-03-22 | Métodos de manufactura de composições farmacêuticas |
| PT03029911T PT1417959E (pt) | 1999-03-26 | 2000-03-22 | Composições farmacêuticas para a administração oral de um medicamento |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US6200604B1 (enExample) |
| EP (4) | EP1417959B1 (enExample) |
| JP (2) | JP4789324B2 (enExample) |
| AT (4) | ATE350017T1 (enExample) |
| AU (1) | AU4019400A (enExample) |
| CA (2) | CA2333375C (enExample) |
| CY (3) | CY1107592T1 (enExample) |
| DE (3) | DE60042463D1 (enExample) |
| DK (3) | DK1417959T3 (enExample) |
| ES (3) | ES2324908T3 (enExample) |
| PT (3) | PT1082106E (enExample) |
| WO (1) | WO2000057858A1 (enExample) |
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|---|---|---|---|---|
| US7611533B2 (en) * | 1995-06-07 | 2009-11-03 | Cook Incorporated | Coated implantable medical device |
| US6949264B1 (en) | 1996-11-27 | 2005-09-27 | Wm. Wrigley Jr. Company | Nutraceuticals or nutritional supplements and method of making |
| US20040023948A1 (en) * | 1997-03-24 | 2004-02-05 | Green Richard David | Fast-dispersing dosage form containing 5-HT1 agonists |
| US20030091629A1 (en) * | 1998-03-27 | 2003-05-15 | Cima Labs Inc. | Sublingual buccal effervescent |
| US20030118645A1 (en) * | 1998-04-29 | 2003-06-26 | Pather S. Indiran | Pharmaceutical compositions for rectal and vaginal administration |
| US6974590B2 (en) | 1998-03-27 | 2005-12-13 | Cima Labs Inc. | Sublingual buccal effervescent |
| US6350470B1 (en) * | 1998-04-29 | 2002-02-26 | Cima Labs Inc. | Effervescent drug delivery system for oral administration |
| US6358060B2 (en) * | 1998-09-03 | 2002-03-19 | Jsr Llc | Two-stage transmucosal medicine delivery system for symptom relief |
| US7163705B2 (en) * | 1998-12-15 | 2007-01-16 | Wm. Wrigley Jr. Company | Coated chewing gum product and method of making |
| US6627234B1 (en) | 1998-12-15 | 2003-09-30 | Wm. Wrigley Jr. Company | Method of producing active agent coated chewing gum products |
| US6531114B1 (en) | 1999-04-06 | 2003-03-11 | Wm. Wrigley Jr. Company | Sildenafil citrate chewing gum formulations and methods of using the same |
| US20020159956A1 (en) * | 1999-04-06 | 2002-10-31 | Ream Ronald L. | Over-coated chewing gum formulations |
| WO2001021156A1 (en) * | 1999-04-06 | 2001-03-29 | Wm. Wrigley Jr. Company | Pharmaceutical chewing gum formulations |
| US6426090B1 (en) | 1999-04-06 | 2002-07-30 | Wm. Wrigley Jr. Company | Over-coated product including tableted center and medicament |
| US7935362B2 (en) * | 1999-04-06 | 2011-05-03 | Wm. Wrigley Jr. Company | Over-coated product including consumable center and medicament |
| US6355265B1 (en) | 1999-04-06 | 2002-03-12 | Wm. Wrigley Jr. Company | Over-coated chewing gum formulations |
| US6773716B2 (en) | 1999-04-06 | 2004-08-10 | Wm. Wrigley Jr. Company | Over-coated chewing gum formulations |
| US6663849B1 (en) | 2000-09-01 | 2003-12-16 | Wm. Wrigley Jr. Company | Antacid chewing gum products coated with high viscosity materials |
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| AU3885201A (en) * | 1999-09-20 | 2001-04-24 | Mastercare | Diet and weight control gum and sucker |
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-
1999
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-
2000
- 2000-03-22 PT PT00919523T patent/PT1082106E/pt unknown
- 2000-03-22 EP EP03029911A patent/EP1417959B1/en not_active Expired - Lifetime
- 2000-03-22 AT AT00919523T patent/ATE350017T1/de active
- 2000-03-22 PT PT03029877T patent/PT1419765E/pt unknown
- 2000-03-22 EP EP03029877A patent/EP1419765B1/en not_active Expired - Lifetime
- 2000-03-22 ES ES03029911T patent/ES2324908T3/es not_active Expired - Lifetime
- 2000-03-22 DK DK03029911T patent/DK1417959T3/da active
- 2000-03-22 AT AT03029911T patent/ATE433745T1/de active
- 2000-03-22 JP JP2000607609A patent/JP4789324B2/ja not_active Expired - Lifetime
- 2000-03-22 DE DE60042463T patent/DE60042463D1/de not_active Expired - Lifetime
- 2000-03-22 PT PT03029911T patent/PT1417959E/pt unknown
- 2000-03-22 AT AT09008228T patent/ATE548028T1/de active
- 2000-03-22 AT AT03029877T patent/ATE434432T1/de active
- 2000-03-22 ES ES00919523T patent/ES2276677T3/es not_active Expired - Lifetime
- 2000-03-22 DK DK03029877T patent/DK1419765T3/da active
- 2000-03-22 DE DE60032691T patent/DE60032691T2/de not_active Expired - Lifetime
- 2000-03-22 CA CA002333375A patent/CA2333375C/en not_active Expired - Lifetime
- 2000-03-22 AU AU40194/00A patent/AU4019400A/en not_active Abandoned
- 2000-03-22 DE DE60042427T patent/DE60042427D1/de not_active Expired - Lifetime
- 2000-03-22 EP EP00919523A patent/EP1082106B1/en not_active Expired - Lifetime
- 2000-03-22 EP EP09008228A patent/EP2095813B1/en not_active Expired - Lifetime
- 2000-03-22 CA CA2569674A patent/CA2569674C/en not_active Expired - Lifetime
- 2000-03-22 ES ES03029877T patent/ES2324907T3/es not_active Expired - Lifetime
- 2000-03-22 WO PCT/US2000/007567 patent/WO2000057858A1/en not_active Ceased
- 2000-03-22 DK DK00919523T patent/DK1082106T3/da active
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2007
- 2007-04-02 CY CY20071100454T patent/CY1107592T1/el unknown
-
2008
- 2008-09-25 JP JP2008246357A patent/JP4954170B2/ja not_active Expired - Lifetime
-
2009
- 2009-06-24 CY CY20091100668T patent/CY1109176T1/el unknown
- 2009-06-25 CY CY20091100667T patent/CY1109172T1/el unknown
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